Quick view Biovision | Thiazovivin | 1681 Cell-permeable. Helps in promoting human embryonic stem cell (hESC) survival by > 30-fold. Thiazovivin enhances the efficiency of fibroblast reprogramming to generate induced pluripotent stem cells... MSRP: Was: Now: $1,152 - $3,504 Choose Options Compare
Quick view Biovision | TAME Hydrochloride | 2050 A small molecule anaphase-promoting complex/cyclosome (APC/C) inhibitor that stabilizes APC/C substrates in mitotic Xenopus extracts. TAME binds to APC and prevents its activation by Cdc20 and Cdh1... MSRP: Was: Now: $690 - $2,555 Choose Options Compare
Quick view Biovision | A-674563 | B1761 A-674563 is a potent, orally available Akt1 inhibitor with an IC50 value of 11nM. Also displays activity against PKA and CDK2 with IC50 values of 16nM and 46nM respectively.A-674563 is a potent,... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Biovision | MK-5108 | B1344 MK-5108 is a highly selective Aurora A inhibitor with IC50 of 0.064 nMMK-5108 is a highly selective Aurora A inhibitor with IC50 of 0.064 nMBiovision | B1344 | MK-5108 DataSheetAlternate... MSRP: Was: Now: $1,411 - $4,018 Choose Options Compare
Quick view Biovision | LY2886721 | 2299 Cell-permeable. A potent and selective β-secretase (BACE-1) inhibitor (IC₅₀ = 20 nM for recombinant hBACE1). Does not inhibit other aspartyl proteases such as cathepsin D, pepsin, and renin. A... MSRP: Was: Now: $1,180 - $3,129 Choose Options Compare
Quick view Biovision | GSK2578215A | 2845 GSK2578215A is a potent and highly selective leucine-rich repeat kinase 2 (LRRK2) inhibitor (IC₅₀ values are 8.9 and 10.1 nM for LRRK2[G2019S] mutant and wild-type LRRK2 respectively). Shows... MSRP: Was: Now: $749 - $2,125 Choose Options Compare
Quick view Biovision | I-BET151 | 2220 A BET bromodomain inhibitor that interacts with BRD4 and BRD3 BET proteins and displaces them from chromatin; displays highefficacy against human and murine MLL-fusion leukemic cell lines, through... MSRP: Was: Now: $665 - $1,754 Choose Options Compare
Quick view Biovision | Boc-D-FMK | 1160 A synthetic peptide that irreversibly inhibits activity of caspase family proteases and blocks apoptosis. The inhibitor is designed as a methyl ester to facilitate cell permeability. The product can... MSRP: Was: Now: $1,180 - $2,842 Choose Options Compare
Quick view Biovision | Crenolanib | 9679 Crenolanib is a highly selective and potent FLT3 tyrosine kinase inhibitor (TKI) with activity against the internal tandem duplication (FLT3/ITD) mutants and the FLT3/D835 point mutants. Also... MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Biovision | Avasimibe | 9506 Avasimibe is an orally bioavailable inhibitor of the acyl coenzyme A: cholesterol acyltransferase (ACAT) (IC₅₀ = 60 nM). Avasimibe also inhibits major drug metabolizing enzymes such as CYP2C9 (IC₅₀ =... MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Biovision | Zanamivir | B1900 Zanamivir is a potent and selective inhibitor of influenza A and B virus neuraminidases with IC₅₀ values of 0.95 nM and 2.7 nM, respectively. It interacts with a group of amino acids in the active... MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Biovision | ONX-0914 | 2555 A potent and selective immunoproteasome inhibitor with minimal cross-reactivity for the constitutive proteasome. It selectively inhibits low–molecular mass polypeptide-7 (LMP7, encoded by Psmb8), the... MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare
Quick view Biovision | T0070907 | 2095 T0070907 is a potent and selective antagonist of the human PPARγ (IC50 = 1 nM). T0070907 suppresses breast cancer cell proliferation and motility via both PPARγ-dependent and –independent mechanisms... MSRP: Now: $980 Add to Cart Compare Quick view Biovision | CHIR-98014 | 2595 Cell-permeable. CHIR-98014 is a potent, selective and ATP-competitive inhibitor of GSK3α and GSK3β (IC₅₀ = 0.65 and 0.58 nM, respectively). In addition, CHIR-98014 displays 500 to greater than... MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Biovision | Golvatinib | 2655 Golvatinib ( E7050) is an orally bioavailable dual kinase inhibitor of c-Met (hepatocyte growth factor receptor) and VEGFR-2 (vascular endothelial growth factor receptor-2) tyrosine kinases with... MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare Quick view Biovision | Cobimetinib | B1689 Cobimetinib(GDC-0973; XL518) is a potent, highly selective inhibitor of mitogen-activated protein kinase kinase(MEK1/2).Cobimetinib(GDC-0973; XL518) is a potent, highly selective inhibitor of... MSRP: Was: Now: $949 - $2,783 Choose Options Compare Quick view Biovision | ADX-47273 | 9562 ADX-47273 is a potent and selective mGluR5 receptor PAM (positive allosteric modulator), EC₅₀ = 0.17 μm, with no effect on other mGluR subtypes. ADX-47273 elevates extracellular signal-regulated... MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Biovision | Fostamatinib Disodium | 1936 A potent, ATP-competitive and selective Syk (Spleen tyrosine kinase) inhibitor (IC₅₀ = 41 nM). Inhibits tumor growth in the Eμ- TCL1 transgenic mouse model of CLL by blocking antigen-dependent B-cell... MSRP: Was: Now: $865 - $2,555 Choose Options Compare Quick view Biovision | DAPT | 1855 Cell permeable. A potent inhibitor of γ-secretase (IC₅₀ = 115 nM for total β-amyloid, IC₅₀ = 200 nM for β-amyloid 1-42). It reduces Aβ levels in vivo in plasma and cerebrospinal fluid in young and... MSRP: Now: $1,351 Add to Cart Compare Quick view Biovision | MRT67307 | B1604 MRT67307 is a dual inhibitor of the IKKe and TBK-1MRT67307 is a dual inhibitor of the IKKe and TBK-1Biovision | B1604 | MRT67307 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Biovision | Ivacaftor | 9582 Ivacaftor (VX-770) is a potent, cell-permeable small molecule potentiator of cystic fibrosis transmembrane conductance regulator (CFTR). It increases the forskolin-induced CFTR-mediated epithelial... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | RepSox | 1894 Cell-permeable. A TGF-β type I receptor (ALK5) inhibitor. Inhibits ALK5 autophosphorylation (IC₅₀ = 4 nM). Can replace one of the four reprogramming factors Sox-2. RepSox has been successfully used... MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Biovision | Laquinimod | 2332 A potent immunomodulator. Also displays anti-inflammatory properties.Laquinimod is a potent immunomodulator. Also displays anti-inflammatory properties.Biovision | 2332 | Laquinimod... MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Biovision | Torin 1 | 2273 A potent, selective and ATP-competitive mTOR inhibitor, with IC₅₀ values of 2 and 10 nM for mTORC1 and mTORC2 respectively; Torin1 displays 1000-fold selectivity for mTOR over PI3K (EC₅₀ = 1800 nM)... MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Biovision | Torin 2 | 2274 A potent, selective and ATP-competitive mTOR inhibitor (IC₅₀ = 2.1 nM for mTORC1). Torin 2 displays 800-fold selectivity for mTOR over PI3K (cellular EC₅₀ values of 0.25 nM and 200 nM, respectively)... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | Quizartinib | 2008 Cell-permeable. A second generation FLT3 receptor tyrosine kinase inhibitor. Quizartinib displays high affinity for FLT3 in a binding assay (Kd = 1.6 nM) and is a potent inhibitor in cellular... MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Biovision | Spautin-1 | 2037 Cell-permeable. A specific and potent autophagy inhibitor in mammalian cells. It promotes the degradation of Vps34 PI3 kinase complexes by inhibiting two ubiquitin specific peptidases, USP10 and... MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Biovision | Pimozide | 1887 Cell-permeable. An antipsychotic drug and D2 dopamine receptor antagonist; binds with high affinity to the cloned 5-HT7 receptor. A Stat5 inhibitor; decreases Stat5 tyrosine phosphorylation, but does... MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Biovision | PRT-060318 | B1911 PR-060318 is a potent and selective Syk inhibtor. It prevents both HIT (Heparin-induced thrombocytopenia) immune complex-induced thrombocytopenia and thrombosis in vivo.PR-060318 is a potent and... MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Biovision | Nampt-IN-1 | B1171 Nampt-IN-1 is a potent and selective NAMPT (Nicotinamide phosphoribosyltransferase) inhibitor. Displays potent anticancer properties. NAMPT is found to be upregulated in various cancer cells and... MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Biovision | SGI-7079 | B1202 SGI-7079 is a potent and selective Axl inhibitor with potential anticancer activity. SGI-7079 significantly inhibits the proliferation of SUM149 or KPL-4 cells with an IC₅₀ of 0.43 or 0.16 μM,... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | AMG319 | B1663 AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ with IC50 of 850 nM.AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ... MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Biovision | GNE-3511 | B1341 GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.Biovision | B1341 | GNE-3511 DataSheetAlternate... MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Biovision | OAC2 | B1080 OAC2 is an Oct4-activating compound that activates expression through the Oct4 gene promoter. In cells expressing Oct4 with Sox2, Klf4, and c-Myc, OAC2 (1 μM) enhances reprogramming efficiency by... MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Biovision | IWP-4 | 2650 IWP-4 is a potent inhibitor of Wnt production that blocks Wnt pathway activity in vitro (IC₅₀ = 25 nM). IWP-4 inactivates Porcupine (porcn), a membrane-bound O-acyltransferase responsible for... MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Biovision | BQU57 | 9576 BQU57 is a GTPase Ral inhibitor. Displays selectivity for Ral relative to the GTPases Ras and RhoA and inhibits tumor xenograft growth to a similar extent to the depletion of Ral using RNA... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | RBC8 | B1136 RBC8 is cell-permeable small molecule that inhibits the binding of Ras-like GTPases A and B ( RalA and RalB GTPase ) to RaLBP1 and shown to suppress growth of xenograft tumors in mice. It reduces the... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | Nazartinib | B2288 Nazartinib is a potent, irreversible, third-generation, mutant-selective epidermal growth factor receptor (EGFR) inhibitor, with potential antineoplastic activity. It covalently binds to and inhibits... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | AZD9496 | B1652 AZD9496 is a potent and orally bioavailable selective estrogen receptor down regulator (Ki=0.7 nM) and antagonist.AZD9496 is a potent and orally bioavailable selective estrogen receptor down... MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Biovision | PT-2385 | B1920 PT-2385 is a potent ad selective inhibitor of hypoxia inducible factor (HIF-2α) with potential antineoplastic activity. PT-2385 selectively disrupts the heterodimerization of HIF-2α with HIF-1β. Very... MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Biovision | JNJ-42041935 | B1072 JNJ-42041935 is a HIF-PHD (Hypoxia-inducible factor- prolyl hydroxylase) inhibitor. JNJ-42041935 is a selective, 2-OG (2-oxoglutarate) competitive, and reversible inhibitor of PHD enzymes (pKis = 7... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | BLU9931 | 9639 BLU9931 is a potent and irreversible small-molecule inhibitor of FGFR4. It potently inhibits FGFR4 activity (IC₅₀ = 3 nM), but only weakly inhibits FGFR1 (IC₅₀ = 591 nM), FGFR2 (IC₅₀ = 493 nM), and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | EHop-016 | 9595 EHop-016 is an analog of NSC-23766 (Cat. No. 1941) that acts as a potent inhibitor of Rac GTPase (IC₅₀ = 1.1 µM for Rac1). The IC₅₀ of 1.1 μM for Rac inhibition by EHop-016 is ∼100-fold lower than... MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Biovision | Optovin | 9594 Optovin is a reversible photoactive TRPA1 activator. It specifically activates TRPA1 (EC₅₀ = 2 μM) but not TRPV1 or TRPM8. Optovin activates human TRPA1 via structure-dependent photochemical... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | STF-118804 | 9552 STF-118804 is a potent and highly specific inhibitor of Nampt (nicotinamide phosphoribosyl transferase) (IC₅₀s = 3-6 nM) that prevents NAD⁺ synthesis from nicotinamide. It inhibits the viability of... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | FIPI | 9593 FIPI is a potent phospholipase D (PLD) inhibitor. FIPI inhibits both PLD1 (IC₅₀ = 25 nM) and PLD2 (IC₅₀ = 20 nM); prevents PLD regulation of F-actin cytoskeleton reorganization, cell spreading, and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | Etrasimod | B2319 A potent and selective sphingosine-1-phosphate-1 (S1P1) receptor antagonist (IC₅₀ =1.88 nM in CHO cells).Etrasimod (APD334) is a potent and selective sphingosine-1-phosphate-1 (S1P1) receptor... MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Biovision | L-779450 | B1709 L-779450 is a potent, ATP-competitive Raf kinase inhibitor (IC50 =10 nM) that displays > 7, > 30 and > 70-fold selectivity over p38α, GSK3β and Lck respectively.L-779450 is a potent, ATP-competitive... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | Cyantraniliprole | B1648 Cyantraniliprole (HGW-86) is an insecticide of the ryanoid class; has activity against pests such as Diaphorina citri that have developed resistance to other classes insecticides.Cyantraniliprole... MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Biovision | IC261 | 9669 IC261 is a reversible, ATP-competitive inhibitor of casein kinase 1 (CK1) (IC₅₀ = ~1 µM for CK1δ and CK1ɛ and 16 µM for CK1α). It is at least 100-fold less effective against PKA, p34cdc2, and p55fyn... MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Biovision | BLZ945 | B1651 BLZ945 is a brain-penetrant CSF-1R kinase inhibitor. The biochemical IC50 for CSF-1R is 1 nM, which is >3200-fold higher than its affinity for other kinases.BLZ945 is a brain-penetrant CSF-1R kinase... MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Biovision | GNE-317 | B1716 GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.Biovision | B1716 | GNE-317... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Thiazovivin | 1681 MSRP: Was: Now: $1,152 - $3,504 Choose Options Compare Quick view Details Biovision | TAME Hydrochloride | 2050 MSRP: Was: Now: $690 - $2,555 Choose Options Compare Quick view Details Biovision | A-674563 | B1761 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | MK-5108 | B1344 MSRP: Was: Now: $1,411 - $4,018 Choose Options Compare Quick view Details Biovision | LY2886721 | 2299 MSRP: Was: Now: $1,180 - $3,129 Choose Options Compare Quick view Details Biovision | GSK2578215A | 2845 MSRP: Was: Now: $749 - $2,125 Choose Options Compare Quick view Details Biovision | I-BET151 | 2220 MSRP: Was: Now: $665 - $1,754 Choose Options Compare Quick view Details Biovision | Boc-D-FMK | 1160 MSRP: Was: Now: $1,180 - $2,842 Choose Options Compare Quick view Details Biovision | Crenolanib | 9679 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Avasimibe | 9506 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Zanamivir | B1900 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | ONX-0914 | 2555 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | T0070907 | 2095 MSRP: Now: $980 Add to Cart Compare Quick view Details Biovision | CHIR-98014 | 2595 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Golvatinib | 2655 MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare Quick view Details Biovision | Cobimetinib | B1689 MSRP: Was: Now: $949 - $2,783 Choose Options Compare Quick view Details Biovision | ADX-47273 | 9562 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Fostamatinib Disodium | 1936 MSRP: Was: Now: $865 - $2,555 Choose Options Compare Quick view Details Biovision | DAPT | 1855 MSRP: Now: $1,351 Add to Cart Compare Quick view Details Biovision | MRT67307 | B1604 MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Details Biovision | Ivacaftor | 9582 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RepSox | 1894 MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Details Biovision | Laquinimod | 2332 MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Details Biovision | Torin 1 | 2273 MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Details Biovision | Torin 2 | 2274 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Quizartinib | 2008 MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Details Biovision | Spautin-1 | 2037 MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Details Biovision | Pimozide | 1887 MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Details Biovision | PRT-060318 | B1911 MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Details Biovision | Nampt-IN-1 | B1171 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | SGI-7079 | B1202 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | AMG319 | B1663 MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Details Biovision | GNE-3511 | B1341 MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Details Biovision | OAC2 | B1080 MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Details Biovision | IWP-4 | 2650 MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Details Biovision | BQU57 | 9576 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RBC8 | B1136 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Nazartinib | B2288 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | AZD9496 | B1652 MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Details Biovision | PT-2385 | B1920 MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Details Biovision | JNJ-42041935 | B1072 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | BLU9931 | 9639 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | EHop-016 | 9595 MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Details Biovision | Optovin | 9594 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | STF-118804 | 9552 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | FIPI | 9593 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | Etrasimod | B2319 MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Details Biovision | L-779450 | B1709 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Cyantraniliprole | B1648 MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Details Biovision | IC261 | 9669 MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Details Biovision | BLZ945 | B1651 MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Details Biovision | GNE-317 | B1716 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Previous 186 187 188 189 190 191 192 193 194 195 196 Next Previous 186 187 188 189 190 191 192 193 194 195 196 Next Compare Selected × OK
Quick view Biovision | CHIR-98014 | 2595 Cell-permeable. CHIR-98014 is a potent, selective and ATP-competitive inhibitor of GSK3α and GSK3β (IC₅₀ = 0.65 and 0.58 nM, respectively). In addition, CHIR-98014 displays 500 to greater than... MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Biovision | Golvatinib | 2655 Golvatinib ( E7050) is an orally bioavailable dual kinase inhibitor of c-Met (hepatocyte growth factor receptor) and VEGFR-2 (vascular endothelial growth factor receptor-2) tyrosine kinases with... MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare
Quick view Biovision | Cobimetinib | B1689 Cobimetinib(GDC-0973; XL518) is a potent, highly selective inhibitor of mitogen-activated protein kinase kinase(MEK1/2).Cobimetinib(GDC-0973; XL518) is a potent, highly selective inhibitor of... MSRP: Was: Now: $949 - $2,783 Choose Options Compare
Quick view Biovision | ADX-47273 | 9562 ADX-47273 is a potent and selective mGluR5 receptor PAM (positive allosteric modulator), EC₅₀ = 0.17 μm, with no effect on other mGluR subtypes. ADX-47273 elevates extracellular signal-regulated... MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Biovision | Fostamatinib Disodium | 1936 A potent, ATP-competitive and selective Syk (Spleen tyrosine kinase) inhibitor (IC₅₀ = 41 nM). Inhibits tumor growth in the Eμ- TCL1 transgenic mouse model of CLL by blocking antigen-dependent B-cell... MSRP: Was: Now: $865 - $2,555 Choose Options Compare
Quick view Biovision | DAPT | 1855 Cell permeable. A potent inhibitor of γ-secretase (IC₅₀ = 115 nM for total β-amyloid, IC₅₀ = 200 nM for β-amyloid 1-42). It reduces Aβ levels in vivo in plasma and cerebrospinal fluid in young and... MSRP: Now: $1,351 Add to Cart Compare Quick view Biovision | MRT67307 | B1604 MRT67307 is a dual inhibitor of the IKKe and TBK-1MRT67307 is a dual inhibitor of the IKKe and TBK-1Biovision | B1604 | MRT67307 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Biovision | Ivacaftor | 9582 Ivacaftor (VX-770) is a potent, cell-permeable small molecule potentiator of cystic fibrosis transmembrane conductance regulator (CFTR). It increases the forskolin-induced CFTR-mediated epithelial... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | RepSox | 1894 Cell-permeable. A TGF-β type I receptor (ALK5) inhibitor. Inhibits ALK5 autophosphorylation (IC₅₀ = 4 nM). Can replace one of the four reprogramming factors Sox-2. RepSox has been successfully used... MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Biovision | Laquinimod | 2332 A potent immunomodulator. Also displays anti-inflammatory properties.Laquinimod is a potent immunomodulator. Also displays anti-inflammatory properties.Biovision | 2332 | Laquinimod... MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Biovision | Torin 1 | 2273 A potent, selective and ATP-competitive mTOR inhibitor, with IC₅₀ values of 2 and 10 nM for mTORC1 and mTORC2 respectively; Torin1 displays 1000-fold selectivity for mTOR over PI3K (EC₅₀ = 1800 nM)... MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Biovision | Torin 2 | 2274 A potent, selective and ATP-competitive mTOR inhibitor (IC₅₀ = 2.1 nM for mTORC1). Torin 2 displays 800-fold selectivity for mTOR over PI3K (cellular EC₅₀ values of 0.25 nM and 200 nM, respectively)... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | Quizartinib | 2008 Cell-permeable. A second generation FLT3 receptor tyrosine kinase inhibitor. Quizartinib displays high affinity for FLT3 in a binding assay (Kd = 1.6 nM) and is a potent inhibitor in cellular... MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Biovision | Spautin-1 | 2037 Cell-permeable. A specific and potent autophagy inhibitor in mammalian cells. It promotes the degradation of Vps34 PI3 kinase complexes by inhibiting two ubiquitin specific peptidases, USP10 and... MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Biovision | Pimozide | 1887 Cell-permeable. An antipsychotic drug and D2 dopamine receptor antagonist; binds with high affinity to the cloned 5-HT7 receptor. A Stat5 inhibitor; decreases Stat5 tyrosine phosphorylation, but does... MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Biovision | PRT-060318 | B1911 PR-060318 is a potent and selective Syk inhibtor. It prevents both HIT (Heparin-induced thrombocytopenia) immune complex-induced thrombocytopenia and thrombosis in vivo.PR-060318 is a potent and... MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Biovision | Nampt-IN-1 | B1171 Nampt-IN-1 is a potent and selective NAMPT (Nicotinamide phosphoribosyltransferase) inhibitor. Displays potent anticancer properties. NAMPT is found to be upregulated in various cancer cells and... MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Biovision | SGI-7079 | B1202 SGI-7079 is a potent and selective Axl inhibitor with potential anticancer activity. SGI-7079 significantly inhibits the proliferation of SUM149 or KPL-4 cells with an IC₅₀ of 0.43 or 0.16 μM,... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | AMG319 | B1663 AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ with IC50 of 850 nM.AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ... MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Biovision | GNE-3511 | B1341 GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.Biovision | B1341 | GNE-3511 DataSheetAlternate... MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Biovision | OAC2 | B1080 OAC2 is an Oct4-activating compound that activates expression through the Oct4 gene promoter. In cells expressing Oct4 with Sox2, Klf4, and c-Myc, OAC2 (1 μM) enhances reprogramming efficiency by... MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Biovision | IWP-4 | 2650 IWP-4 is a potent inhibitor of Wnt production that blocks Wnt pathway activity in vitro (IC₅₀ = 25 nM). IWP-4 inactivates Porcupine (porcn), a membrane-bound O-acyltransferase responsible for... MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Biovision | BQU57 | 9576 BQU57 is a GTPase Ral inhibitor. Displays selectivity for Ral relative to the GTPases Ras and RhoA and inhibits tumor xenograft growth to a similar extent to the depletion of Ral using RNA... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | RBC8 | B1136 RBC8 is cell-permeable small molecule that inhibits the binding of Ras-like GTPases A and B ( RalA and RalB GTPase ) to RaLBP1 and shown to suppress growth of xenograft tumors in mice. It reduces the... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | Nazartinib | B2288 Nazartinib is a potent, irreversible, third-generation, mutant-selective epidermal growth factor receptor (EGFR) inhibitor, with potential antineoplastic activity. It covalently binds to and inhibits... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | AZD9496 | B1652 AZD9496 is a potent and orally bioavailable selective estrogen receptor down regulator (Ki=0.7 nM) and antagonist.AZD9496 is a potent and orally bioavailable selective estrogen receptor down... MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Biovision | PT-2385 | B1920 PT-2385 is a potent ad selective inhibitor of hypoxia inducible factor (HIF-2α) with potential antineoplastic activity. PT-2385 selectively disrupts the heterodimerization of HIF-2α with HIF-1β. Very... MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Biovision | JNJ-42041935 | B1072 JNJ-42041935 is a HIF-PHD (Hypoxia-inducible factor- prolyl hydroxylase) inhibitor. JNJ-42041935 is a selective, 2-OG (2-oxoglutarate) competitive, and reversible inhibitor of PHD enzymes (pKis = 7... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | BLU9931 | 9639 BLU9931 is a potent and irreversible small-molecule inhibitor of FGFR4. It potently inhibits FGFR4 activity (IC₅₀ = 3 nM), but only weakly inhibits FGFR1 (IC₅₀ = 591 nM), FGFR2 (IC₅₀ = 493 nM), and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | EHop-016 | 9595 EHop-016 is an analog of NSC-23766 (Cat. No. 1941) that acts as a potent inhibitor of Rac GTPase (IC₅₀ = 1.1 µM for Rac1). The IC₅₀ of 1.1 μM for Rac inhibition by EHop-016 is ∼100-fold lower than... MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Biovision | Optovin | 9594 Optovin is a reversible photoactive TRPA1 activator. It specifically activates TRPA1 (EC₅₀ = 2 μM) but not TRPV1 or TRPM8. Optovin activates human TRPA1 via structure-dependent photochemical... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | STF-118804 | 9552 STF-118804 is a potent and highly specific inhibitor of Nampt (nicotinamide phosphoribosyl transferase) (IC₅₀s = 3-6 nM) that prevents NAD⁺ synthesis from nicotinamide. It inhibits the viability of... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Biovision | FIPI | 9593 FIPI is a potent phospholipase D (PLD) inhibitor. FIPI inhibits both PLD1 (IC₅₀ = 25 nM) and PLD2 (IC₅₀ = 20 nM); prevents PLD regulation of F-actin cytoskeleton reorganization, cell spreading, and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Biovision | Etrasimod | B2319 A potent and selective sphingosine-1-phosphate-1 (S1P1) receptor antagonist (IC₅₀ =1.88 nM in CHO cells).Etrasimod (APD334) is a potent and selective sphingosine-1-phosphate-1 (S1P1) receptor... MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Biovision | L-779450 | B1709 L-779450 is a potent, ATP-competitive Raf kinase inhibitor (IC50 =10 nM) that displays > 7, > 30 and > 70-fold selectivity over p38α, GSK3β and Lck respectively.L-779450 is a potent, ATP-competitive... MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Biovision | Cyantraniliprole | B1648 Cyantraniliprole (HGW-86) is an insecticide of the ryanoid class; has activity against pests such as Diaphorina citri that have developed resistance to other classes insecticides.Cyantraniliprole... MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Biovision | IC261 | 9669 IC261 is a reversible, ATP-competitive inhibitor of casein kinase 1 (CK1) (IC₅₀ = ~1 µM for CK1δ and CK1ɛ and 16 µM for CK1α). It is at least 100-fold less effective against PKA, p34cdc2, and p55fyn... MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Biovision | BLZ945 | B1651 BLZ945 is a brain-penetrant CSF-1R kinase inhibitor. The biochemical IC50 for CSF-1R is 1 nM, which is >3200-fold higher than its affinity for other kinases.BLZ945 is a brain-penetrant CSF-1R kinase... MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Biovision | GNE-317 | B1716 GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.Biovision | B1716 | GNE-317... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Thiazovivin | 1681 MSRP: Was: Now: $1,152 - $3,504 Choose Options Compare Quick view Details Biovision | TAME Hydrochloride | 2050 MSRP: Was: Now: $690 - $2,555 Choose Options Compare Quick view Details Biovision | A-674563 | B1761 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | MK-5108 | B1344 MSRP: Was: Now: $1,411 - $4,018 Choose Options Compare Quick view Details Biovision | LY2886721 | 2299 MSRP: Was: Now: $1,180 - $3,129 Choose Options Compare Quick view Details Biovision | GSK2578215A | 2845 MSRP: Was: Now: $749 - $2,125 Choose Options Compare Quick view Details Biovision | I-BET151 | 2220 MSRP: Was: Now: $665 - $1,754 Choose Options Compare Quick view Details Biovision | Boc-D-FMK | 1160 MSRP: Was: Now: $1,180 - $2,842 Choose Options Compare Quick view Details Biovision | Crenolanib | 9679 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Avasimibe | 9506 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Zanamivir | B1900 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | ONX-0914 | 2555 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | T0070907 | 2095 MSRP: Now: $980 Add to Cart Compare Quick view Details Biovision | CHIR-98014 | 2595 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Golvatinib | 2655 MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare Quick view Details Biovision | Cobimetinib | B1689 MSRP: Was: Now: $949 - $2,783 Choose Options Compare Quick view Details Biovision | ADX-47273 | 9562 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Fostamatinib Disodium | 1936 MSRP: Was: Now: $865 - $2,555 Choose Options Compare Quick view Details Biovision | DAPT | 1855 MSRP: Now: $1,351 Add to Cart Compare Quick view Details Biovision | MRT67307 | B1604 MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Details Biovision | Ivacaftor | 9582 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RepSox | 1894 MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Details Biovision | Laquinimod | 2332 MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Details Biovision | Torin 1 | 2273 MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Details Biovision | Torin 2 | 2274 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Quizartinib | 2008 MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Details Biovision | Spautin-1 | 2037 MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Details Biovision | Pimozide | 1887 MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Details Biovision | PRT-060318 | B1911 MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Details Biovision | Nampt-IN-1 | B1171 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | SGI-7079 | B1202 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | AMG319 | B1663 MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Details Biovision | GNE-3511 | B1341 MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Details Biovision | OAC2 | B1080 MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Details Biovision | IWP-4 | 2650 MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Details Biovision | BQU57 | 9576 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RBC8 | B1136 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Nazartinib | B2288 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | AZD9496 | B1652 MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Details Biovision | PT-2385 | B1920 MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Details Biovision | JNJ-42041935 | B1072 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | BLU9931 | 9639 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | EHop-016 | 9595 MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Details Biovision | Optovin | 9594 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | STF-118804 | 9552 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | FIPI | 9593 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | Etrasimod | B2319 MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Details Biovision | L-779450 | B1709 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Cyantraniliprole | B1648 MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Details Biovision | IC261 | 9669 MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Details Biovision | BLZ945 | B1651 MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Details Biovision | GNE-317 | B1716 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Previous 186 187 188 189 190 191 192 193 194 195 196 Next Previous 186 187 188 189 190 191 192 193 194 195 196 Next Compare Selected × OK
Quick view Biovision | MRT67307 | B1604 MRT67307 is a dual inhibitor of the IKKe and TBK-1MRT67307 is a dual inhibitor of the IKKe and TBK-1Biovision | B1604 | MRT67307 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare
Quick view Biovision | Ivacaftor | 9582 Ivacaftor (VX-770) is a potent, cell-permeable small molecule potentiator of cystic fibrosis transmembrane conductance regulator (CFTR). It increases the forskolin-induced CFTR-mediated epithelial... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare
Quick view Biovision | RepSox | 1894 Cell-permeable. A TGF-β type I receptor (ALK5) inhibitor. Inhibits ALK5 autophosphorylation (IC₅₀ = 4 nM). Can replace one of the four reprogramming factors Sox-2. RepSox has been successfully used... MSRP: Was: Now: $837 - $2,209 Choose Options Compare
Quick view Biovision | Laquinimod | 2332 A potent immunomodulator. Also displays anti-inflammatory properties.Laquinimod is a potent immunomodulator. Also displays anti-inflammatory properties.Biovision | 2332 | Laquinimod... MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare
Quick view Biovision | Torin 1 | 2273 A potent, selective and ATP-competitive mTOR inhibitor, with IC₅₀ values of 2 and 10 nM for mTORC1 and mTORC2 respectively; Torin1 displays 1000-fold selectivity for mTOR over PI3K (EC₅₀ = 1800 nM)... MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare
Quick view Biovision | Torin 2 | 2274 A potent, selective and ATP-competitive mTOR inhibitor (IC₅₀ = 2.1 nM for mTORC1). Torin 2 displays 800-fold selectivity for mTOR over PI3K (cellular EC₅₀ values of 0.25 nM and 200 nM, respectively)... MSRP: Was: Now: $949 - $2,898 Choose Options Compare
Quick view Biovision | Quizartinib | 2008 Cell-permeable. A second generation FLT3 receptor tyrosine kinase inhibitor. Quizartinib displays high affinity for FLT3 in a binding assay (Kd = 1.6 nM) and is a potent inhibitor in cellular... MSRP: Was: Now: $809 - $2,237 Choose Options Compare
Quick view Biovision | Spautin-1 | 2037 Cell-permeable. A specific and potent autophagy inhibitor in mammalian cells. It promotes the degradation of Vps34 PI3 kinase complexes by inhibiting two ubiquitin specific peptidases, USP10 and... MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare
Quick view Biovision | Pimozide | 1887 Cell-permeable. An antipsychotic drug and D2 dopamine receptor antagonist; binds with high affinity to the cloned 5-HT7 receptor. A Stat5 inhibitor; decreases Stat5 tyrosine phosphorylation, but does... MSRP: Was: Now: $690 - $1,813 Choose Options Compare
Quick view Biovision | PRT-060318 | B1911 PR-060318 is a potent and selective Syk inhibtor. It prevents both HIT (Heparin-induced thrombocytopenia) immune complex-induced thrombocytopenia and thrombosis in vivo.PR-060318 is a potent and... MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare
Quick view Biovision | Nampt-IN-1 | B1171 Nampt-IN-1 is a potent and selective NAMPT (Nicotinamide phosphoribosyltransferase) inhibitor. Displays potent anticancer properties. NAMPT is found to be upregulated in various cancer cells and... MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare
Quick view Biovision | SGI-7079 | B1202 SGI-7079 is a potent and selective Axl inhibitor with potential anticancer activity. SGI-7079 significantly inhibits the proliferation of SUM149 or KPL-4 cells with an IC₅₀ of 0.43 or 0.16 μM,... MSRP: Was: Now: $949 - $2,898 Choose Options Compare
Quick view Biovision | AMG319 | B1663 AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ with IC50 of 850 nM.AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, also inhibits PI3Kγ... MSRP: Was: Now: $949 - $2,870 Choose Options Compare
Quick view Biovision | GNE-3511 | B1341 GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.GNE-3511 is a potent and selective zipper kinase (DLK, MAP3K12) inhibitors.Biovision | B1341 | GNE-3511 DataSheetAlternate... MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare
Quick view Biovision | OAC2 | B1080 OAC2 is an Oct4-activating compound that activates expression through the Oct4 gene promoter. In cells expressing Oct4 with Sox2, Klf4, and c-Myc, OAC2 (1 μM) enhances reprogramming efficiency by... MSRP: Was: Now: $718 - $1,925 Choose Options Compare
Quick view Biovision | IWP-4 | 2650 IWP-4 is a potent inhibitor of Wnt production that blocks Wnt pathway activity in vitro (IC₅₀ = 25 nM). IWP-4 inactivates Porcupine (porcn), a membrane-bound O-acyltransferase responsible for... MSRP: Was: Now: $718 - $1,985 Choose Options Compare
Quick view Biovision | BQU57 | 9576 BQU57 is a GTPase Ral inhibitor. Displays selectivity for Ral relative to the GTPases Ras and RhoA and inhibits tumor xenograft growth to a similar extent to the depletion of Ral using RNA... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare
Quick view Biovision | RBC8 | B1136 RBC8 is cell-permeable small molecule that inhibits the binding of Ras-like GTPases A and B ( RalA and RalB GTPase ) to RaLBP1 and shown to suppress growth of xenograft tumors in mice. It reduces the... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Biovision | Nazartinib | B2288 Nazartinib is a potent, irreversible, third-generation, mutant-selective epidermal growth factor receptor (EGFR) inhibitor, with potential antineoplastic activity. It covalently binds to and inhibits... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Biovision | AZD9496 | B1652 AZD9496 is a potent and orally bioavailable selective estrogen receptor down regulator (Ki=0.7 nM) and antagonist.AZD9496 is a potent and orally bioavailable selective estrogen receptor down... MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare
Quick view Biovision | PT-2385 | B1920 PT-2385 is a potent ad selective inhibitor of hypoxia inducible factor (HIF-2α) with potential antineoplastic activity. PT-2385 selectively disrupts the heterodimerization of HIF-2α with HIF-1β. Very... MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare
Quick view Biovision | JNJ-42041935 | B1072 JNJ-42041935 is a HIF-PHD (Hypoxia-inducible factor- prolyl hydroxylase) inhibitor. JNJ-42041935 is a selective, 2-OG (2-oxoglutarate) competitive, and reversible inhibitor of PHD enzymes (pKis = 7... MSRP: Was: Now: $949 - $2,898 Choose Options Compare
Quick view Biovision | BLU9931 | 9639 BLU9931 is a potent and irreversible small-molecule inhibitor of FGFR4. It potently inhibits FGFR4 activity (IC₅₀ = 3 nM), but only weakly inhibits FGFR1 (IC₅₀ = 591 nM), FGFR2 (IC₅₀ = 493 nM), and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare
Quick view Biovision | EHop-016 | 9595 EHop-016 is an analog of NSC-23766 (Cat. No. 1941) that acts as a potent inhibitor of Rac GTPase (IC₅₀ = 1.1 µM for Rac1). The IC₅₀ of 1.1 μM for Rac inhibition by EHop-016 is ∼100-fold lower than... MSRP: Was: Now: $837 - $2,440 Choose Options Compare
Quick view Biovision | Optovin | 9594 Optovin is a reversible photoactive TRPA1 activator. It specifically activates TRPA1 (EC₅₀ = 2 μM) but not TRPV1 or TRPM8. Optovin activates human TRPA1 via structure-dependent photochemical... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Biovision | STF-118804 | 9552 STF-118804 is a potent and highly specific inhibitor of Nampt (nicotinamide phosphoribosyl transferase) (IC₅₀s = 3-6 nM) that prevents NAD⁺ synthesis from nicotinamide. It inhibits the viability of... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Biovision | FIPI | 9593 FIPI is a potent phospholipase D (PLD) inhibitor. FIPI inhibits both PLD1 (IC₅₀ = 25 nM) and PLD2 (IC₅₀ = 20 nM); prevents PLD regulation of F-actin cytoskeleton reorganization, cell spreading, and... MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare
Quick view Biovision | Etrasimod | B2319 A potent and selective sphingosine-1-phosphate-1 (S1P1) receptor antagonist (IC₅₀ =1.88 nM in CHO cells).Etrasimod (APD334) is a potent and selective sphingosine-1-phosphate-1 (S1P1) receptor... MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare
Quick view Biovision | L-779450 | B1709 L-779450 is a potent, ATP-competitive Raf kinase inhibitor (IC50 =10 nM) that displays > 7, > 30 and > 70-fold selectivity over p38α, GSK3β and Lck respectively.L-779450 is a potent, ATP-competitive... MSRP: Was: Now: $949 - $2,898 Choose Options Compare
Quick view Biovision | Cyantraniliprole | B1648 Cyantraniliprole (HGW-86) is an insecticide of the ryanoid class; has activity against pests such as Diaphorina citri that have developed resistance to other classes insecticides.Cyantraniliprole... MSRP: Was: Now: $809 - $2,328 Choose Options Compare
Quick view Biovision | IC261 | 9669 IC261 is a reversible, ATP-competitive inhibitor of casein kinase 1 (CK1) (IC₅₀ = ~1 µM for CK1δ and CK1ɛ and 16 µM for CK1α). It is at least 100-fold less effective against PKA, p34cdc2, and p55fyn... MSRP: Was: Now: $949 - $2,727 Choose Options Compare
Quick view Biovision | BLZ945 | B1651 BLZ945 is a brain-penetrant CSF-1R kinase inhibitor. The biochemical IC50 for CSF-1R is 1 nM, which is >3200-fold higher than its affinity for other kinases.BLZ945 is a brain-penetrant CSF-1R kinase... MSRP: Was: Now: $777 - $2,184 Choose Options Compare
Quick view Biovision | GNE-317 | B1716 GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.GNE-317 is a potent and selective PI3K inhibitor with potential anticancer activity.Biovision | B1716 | GNE-317... MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Details Biovision | Thiazovivin | 1681 MSRP: Was: Now: $1,152 - $3,504 Choose Options Compare
Quick view Details Biovision | TAME Hydrochloride | 2050 MSRP: Was: Now: $690 - $2,555 Choose Options Compare
Quick view Details Biovision | A-674563 | B1761 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Details Biovision | MK-5108 | B1344 MSRP: Was: Now: $1,411 - $4,018 Choose Options Compare
Quick view Details Biovision | LY2886721 | 2299 MSRP: Was: Now: $1,180 - $3,129 Choose Options Compare
Quick view Details Biovision | GSK2578215A | 2845 MSRP: Was: Now: $749 - $2,125 Choose Options Compare
Quick view Details Biovision | Boc-D-FMK | 1160 MSRP: Was: Now: $1,180 - $2,842 Choose Options Compare
Quick view Details Biovision | Crenolanib | 9679 MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Details Biovision | Zanamivir | B1900 MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Details Biovision | ONX-0914 | 2555 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare
Quick view Details Biovision | T0070907 | 2095 MSRP: Now: $980 Add to Cart Compare Quick view Details Biovision | CHIR-98014 | 2595 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Golvatinib | 2655 MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare Quick view Details Biovision | Cobimetinib | B1689 MSRP: Was: Now: $949 - $2,783 Choose Options Compare Quick view Details Biovision | ADX-47273 | 9562 MSRP: Was: Now: $777 - $2,209 Choose Options Compare Quick view Details Biovision | Fostamatinib Disodium | 1936 MSRP: Was: Now: $865 - $2,555 Choose Options Compare Quick view Details Biovision | DAPT | 1855 MSRP: Now: $1,351 Add to Cart Compare Quick view Details Biovision | MRT67307 | B1604 MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Details Biovision | Ivacaftor | 9582 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RepSox | 1894 MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Details Biovision | Laquinimod | 2332 MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Details Biovision | Torin 1 | 2273 MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Details Biovision | Torin 2 | 2274 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Quizartinib | 2008 MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Details Biovision | Spautin-1 | 2037 MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Details Biovision | Pimozide | 1887 MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Details Biovision | PRT-060318 | B1911 MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Details Biovision | Nampt-IN-1 | B1171 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | SGI-7079 | B1202 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | AMG319 | B1663 MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Details Biovision | GNE-3511 | B1341 MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Details Biovision | OAC2 | B1080 MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Details Biovision | IWP-4 | 2650 MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Details Biovision | BQU57 | 9576 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RBC8 | B1136 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Nazartinib | B2288 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | AZD9496 | B1652 MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Details Biovision | PT-2385 | B1920 MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Details Biovision | JNJ-42041935 | B1072 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | BLU9931 | 9639 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | EHop-016 | 9595 MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Details Biovision | Optovin | 9594 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | STF-118804 | 9552 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | FIPI | 9593 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | Etrasimod | B2319 MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Details Biovision | L-779450 | B1709 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Cyantraniliprole | B1648 MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Details Biovision | IC261 | 9669 MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Details Biovision | BLZ945 | B1651 MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Details Biovision | GNE-317 | B1716 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Previous 186 187 188 189 190 191 192 193 194 195 196 Next Previous 186 187 188 189 190 191 192 193 194 195 196 Next Compare Selected
Quick view Details Biovision | CHIR-98014 | 2595 MSRP: Was: Now: $777 - $2,209 Choose Options Compare
Quick view Details Biovision | Golvatinib | 2655 MSRP: Was: Now: $1,120 - $3,444 Choose Options Compare
Quick view Details Biovision | Cobimetinib | B1689 MSRP: Was: Now: $949 - $2,783 Choose Options Compare
Quick view Details Biovision | Fostamatinib Disodium | 1936 MSRP: Was: Now: $865 - $2,555 Choose Options Compare
Quick view Details Biovision | DAPT | 1855 MSRP: Now: $1,351 Add to Cart Compare Quick view Details Biovision | MRT67307 | B1604 MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare Quick view Details Biovision | Ivacaftor | 9582 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RepSox | 1894 MSRP: Was: Now: $837 - $2,209 Choose Options Compare Quick view Details Biovision | Laquinimod | 2332 MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare Quick view Details Biovision | Torin 1 | 2273 MSRP: Was: Now: $1,092 - $3,213 Choose Options Compare Quick view Details Biovision | Torin 2 | 2274 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Quizartinib | 2008 MSRP: Was: Now: $809 - $2,237 Choose Options Compare Quick view Details Biovision | Spautin-1 | 2037 MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare Quick view Details Biovision | Pimozide | 1887 MSRP: Was: Now: $690 - $1,813 Choose Options Compare Quick view Details Biovision | PRT-060318 | B1911 MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare Quick view Details Biovision | Nampt-IN-1 | B1171 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare Quick view Details Biovision | SGI-7079 | B1202 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | AMG319 | B1663 MSRP: Was: Now: $949 - $2,870 Choose Options Compare Quick view Details Biovision | GNE-3511 | B1341 MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare Quick view Details Biovision | OAC2 | B1080 MSRP: Was: Now: $718 - $1,925 Choose Options Compare Quick view Details Biovision | IWP-4 | 2650 MSRP: Was: Now: $718 - $1,985 Choose Options Compare Quick view Details Biovision | BQU57 | 9576 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | RBC8 | B1136 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | Nazartinib | B2288 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | AZD9496 | B1652 MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare Quick view Details Biovision | PT-2385 | B1920 MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare Quick view Details Biovision | JNJ-42041935 | B1072 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | BLU9931 | 9639 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | EHop-016 | 9595 MSRP: Was: Now: $837 - $2,440 Choose Options Compare Quick view Details Biovision | Optovin | 9594 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | STF-118804 | 9552 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Quick view Details Biovision | FIPI | 9593 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare Quick view Details Biovision | Etrasimod | B2319 MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare Quick view Details Biovision | L-779450 | B1709 MSRP: Was: Now: $949 - $2,898 Choose Options Compare Quick view Details Biovision | Cyantraniliprole | B1648 MSRP: Was: Now: $809 - $2,328 Choose Options Compare Quick view Details Biovision | IC261 | 9669 MSRP: Was: Now: $949 - $2,727 Choose Options Compare Quick view Details Biovision | BLZ945 | B1651 MSRP: Was: Now: $777 - $2,184 Choose Options Compare Quick view Details Biovision | GNE-317 | B1716 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare Previous 186 187 188 189 190 191 192 193 194 195 196 Next Previous 186 187 188 189 190 191 192 193 194 195 196 Next Compare Selected
Quick view Details Biovision | MRT67307 | B1604 MSRP: Was: Now: $1,411 - $4,158 Choose Options Compare
Quick view Details Biovision | Ivacaftor | 9582 MSRP: Was: Now: $1,061 - $3,357 Choose Options Compare
Quick view Details Biovision | Laquinimod | 2332 MSRP: Was: Now: $1,120 - $3,644 Choose Options Compare
Quick view Details Biovision | Quizartinib | 2008 MSRP: Was: Now: $809 - $2,237 Choose Options Compare
Quick view Details Biovision | Spautin-1 | 2037 MSRP: Was: Now: $1,180 - $3,584 Choose Options Compare
Quick view Details Biovision | PRT-060318 | B1911 MSRP: Was: Now: $1,582 - $5,422 Choose Options Compare
Quick view Details Biovision | Nampt-IN-1 | B1171 MSRP: Was: Now: $1,120 - $3,584 Choose Options Compare
Quick view Details Biovision | GNE-3511 | B1341 MSRP: Was: Now: $1,866 - $6,311 Choose Options Compare
Quick view Details Biovision | Nazartinib | B2288 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Details Biovision | AZD9496 | B1652 MSRP: Was: Now: $2,184 - $7,515 Choose Options Compare
Quick view Details Biovision | PT-2385 | B1920 MSRP: Was: Now: $1,495 - $4,851 Choose Options Compare
Quick view Details Biovision | JNJ-42041935 | B1072 MSRP: Was: Now: $949 - $2,898 Choose Options Compare
Quick view Details Biovision | STF-118804 | 9552 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare
Quick view Details Biovision | Etrasimod | B2319 MSRP: Was: Now: $1,061 - $3,129 Choose Options Compare
Quick view Details Biovision | Cyantraniliprole | B1648 MSRP: Was: Now: $809 - $2,328 Choose Options Compare
Quick view Details Biovision | GNE-317 | B1716 MSRP: Was: Now: $1,008 - $3,129 Choose Options Compare