Quick view Biovision | BV6 | B1332 BV6 is a selective inhibitor of IAP proteinsBV6 is a selective inhibitor of IAP proteinsBiovision | B1332 | BV6 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: £738 - £2,214 Choose Options Compare
Quick view Biovision | Nexturastat A | 2098 Nexturastat A is an aryl urea derivative that acts as a potent and highly selective inhibitor of histone deacetylase 6 (HDAC6) (IC₅₀ = 5.02 ± 0.60 nM). Displays 600-, 1380-, 1330-, 1870-, -2330,... MSRP: Now: £592 Add to Cart Compare Quick view Biovision | TAPI-1 | 2068 Inhibitor of TNF-α processing (IC₅₀ = 100 nM), similar to TAPI-0 (Cat. No. 2067-1), but more stable in tissue culture and in vivo. Inhibits TACE and other metalloproteases. Blocks release of TNF- α... MSRP: Now: £1,214 Add to Cart Compare Quick view Biovision | CNX-1351 | B1673 CNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMCNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMBiovision | B1673 | CNX-1351... MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Biovision | Brefeldin A | 1560 Brefeldin A has been shown to induce apoptosis in human tumor cells through caspase activation. It has also been shown to block translocation of proteins from the endoplasmic reticulum to the Golgi... MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Biovision | Birinapant | 2597 Birinapant is a SMAC (synthetic small molecule and peptidomimetic of second mitochondrial-derived activator of caspases) mimetic and IAP (Inhibitor of Apoptosis Protein) antagonist with potential... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | PFI-1 | 2203 PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC₅₀... MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Biovision | VS-5584 | 9603 VS-5584 is a potent and selective PI3K/mTOR kinase inhibitor. It inhibits mTOR (IC₅₀ = 37 nM) and PI3K (IC₅₀s = 16, 68, 25, and 42 nM for the α, β, γ, and δ isoforms, respectively) without relevant... MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Biovision | Sapacitabine | B2002 Sapacitabine is an orally bioavailable nucleoside analog prodrug that is potentially useful for treatment of hematologic malignancies and solid tumors. The active metabolite of sapacitabine, CNDAC... MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Biovision | Briciclib | B1140 Briciclib is a small molecule that suppresses cyclin D1 accumulation in cancer cells. Cyclin D, a member of the cyclin family of cell cycle regulators, plays a key role in cell cycle division and is... MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Biovision | Nimorazole | 9521 Nimorazole is a 5-nitroimidazole derivative that displays antimicrobial activity. Used in the treatment of intestinal protozoal infections. Also acts as a hypoxic radiosensitizer.Nimorazole is a... MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Biovision | Kartogenin | 2066 Cell-permeable. Kartogenin promotes the selective differentiation of multipotent mesenchymal stem cells into chondrocytes (EC₅₀ = 100 nM). Displays chondroprotective effects in vitro and is... MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Biovision | Ethynylcytidine | B1266 Ethynylcytidine is a synthetic cytidine nucleoside containing a covalently bound ethynyl group with potential antineoplastic and radiosensitizing activities. Ethynylcytidine is metabolized in tumor... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | Cilengitide | B2365 Cilengitide is a cyclo-(Arg-Gly-Asp-D-Phe-Val) (cRGDfV) peptide that acts as an integrin αVβ3 receptor antagonist. It inhibits adhesion and induces apoptosis of U87MG and U373MG malignant glioma (MG)... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | BMS-303141 | 2821 BMS-303141 is a potent inhibitor of ATP citrate lyase (ACL) (IC₅₀ = 0.13 µM for human recombinant ACL). BMS-303141 inhibits lipid synthesis in HepG2 cells with an IC₅₀ of 8 μM, and lowers plasma... MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Biovision | Arglabin | 9691 Arglabin is a potent anti-inflammatory and anticancer agent. It also acts as a Farnesyltransferase inhibitor and antiatherogenic compound. Prevents the accumulation of lipid containing plaques in... MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Biovision | ACTB-1003 | B2016 ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2 and 4 nM for FGFR1, VEGFR2 and Tie-2, respectively. Displays anticancer activities.ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2... MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Biovision | Citarinostat | B1560 Citarinostat (ACY-241), is a potent, selective and orally available histone deacetylase 6 (HDAC6) inhibitor with IC₅₀ values of 4 nM and 76 nM for HDAC6 and HDAC3, respectively. Displays... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | SM-164 | B1816 SM-164 is a potent cell-permeable and bivalent Smac mimetic which binds to a XIAP protein with a Ki value of 0.56 nM, and binds to cIAP-1 and cIAP-2 proteins with Ki values of 0.31 and 1.1 nM,... MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Biovision | CTx-0294885 | 9435 CTx-0294885 is a broad-spectrum kinase inhibitor. CTx-0294885 displays inhibitory activity against a broad range of kinases in vitro. CTx-0294885 could be a potentially powerful new tool for analysis... MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Biovision | P7C3-A20 | 2850 P7C3-A20 is a derivative of P7C3 (Cat. No. 2849), and is a proneurogenic, neuroprotective agent. P7C3-A20 displays increased activity and an improved toxicity profile compared to P7C3... MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Biovision | P7C3 | 2849 P7C3 is an aminopropyl carbazole derivative that acts as a proneurogenic, neuroprotective compound. Protects newborn neurons in the dentate gyrus by mitigating cell death. Also enhances learning and... MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Biovision | Uprosertib | B1760 Uprosertib, also known as GSK2141795 and GSK795, is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity.Uprosertib,... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | DBeQ | 1858 Cell- permeable. A potent, selective, reversible, and ATP-competitive p97 inhibitor. DBeQ blocks both ubiquitin-dependent and autophagic protein clearance pathways and rapidly promotes executioner... MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Biovision | X-GAL | 2671 X-GAL is a useful chromogenic substrate for β-galactosidase that produces a rich blue color that can easily be detected visually over background. X-GAL is used to indicate whether a cell expresses... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | Luminol | B1807 Luminol is a useful probe that displays chemiluminescence upon oxidation. Horseradish peroxidase (HRP), combined with hydrogen peroxide as an activator, causes luminescent peroxidation of luminol... MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Biovision | DTT | 1201 An excellent reagent for maintaining SH groups in reduced state. DTT quantitatively reduces disulfides. It is effective in sample buffers for reducing protein disulfide bonds prior to SDSPAGE.DTT is... MSRP: Now: £462 Add to Cart Compare Quick view Biovision | DTE | B2410 A useful reagent for maintaining sulfhydryl groups in the reduced stateDTE is a useful reagent for maintaining sulfhydryl groups in the reduced stateBiovision | B2410 | DTE DataSheetAlternate... MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Biovision | Y-320 | B1164 Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T cells stimulated with IL-15 with IC50 values of 20 to 60 nM.Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | DMOG | 2216 A cell-permeable prolyl 4-hydroxylase (P4H) inhibitor; inhibits hypoxia-inducible factor α (HIF-α) prolyl hydroxylase (HIF-PH). Increases levels of HIF-1α; promotes cell survival under hypoxic... MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Biovision | PTC-209 | B1055 PTC-209 is a potent, cell-permeable, BMI-1 inhibitor (IC₅₀ = 0.5 µM) with potential anticancer activity. PTC-209 lowers the self-renewal properties of colorectal cancer-initiating cells (CICs)... MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Biovision | TCS JNK 5a | B1688 TCS JNK 5a (JNK Inhibitor IX) is a selective inhibitor of JNK2 and JNK3; displays no significant activity at a range of other protein kinases including EGFR, ErbB2, cdk2, PLK-1 and Src (pIC50 < 5.0)... MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Biovision | Inauhzin | 9555 Inauhzin is a potent SIRT inhibitor that effectively reactivates p53 by inhibiting SIRT1 activity. Inauhzin inhibits cell proliferation, induces senescence, and p53-dependent apoptosis of human... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | HS-173 | B1627 HS-173 is a novel PI3K inhibitor, that is used for cancer treatment. HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on cancer cells.HS-173 is a novel PI3K... MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Biovision | FLI-06 | 2603 A potent Notch signaling (EC₅₀ = 2.3 µM) as well as the early secretory pathway inhibitor. FLI-06 leads to a disruption of the Golgi by a mechanism different from Brefeldin A (Cat. No. 1560) or other... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Atglistatin | B1864 Atglistatin is a potent, and selective inhibitor of adipose triglyceride lipase (ATGL) the rate limiting enzyme involved in fatty acid mobilization and prevention of lipolysis. It does not inhibit... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | AdipoRon | 2565 A potent and selective adiponectin receptor agonist (Kd = 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively). Displays similar effects to adiponectin in muscle and liver such as activation of... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | CPI-203 | 9404 CPI-203 is an analog of (+)-JQ1 (Cat. No. 2070). Acts as a BET bromodomain inhibitor. It is comparable or superior to (+)-JQ1 in inhibiting BRD4 binding and action in vitro or in cells.CPI-203... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SF1670 | 2774 SF1670 is a selective PTEN (phosphatase and tensin homolog) inhibitor (IC₅₀ = 2 µM). It specifically binds to the active site of PTEN. At nanomolar concentrations it increases cellular... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | ID-8 | 2562 ID-8 is a cell culture supplement that can sustain self-renewal and pluripotency of mouse embryonic stem cells in vitro. At 10 μM it stimulates proliferation in serum-free media at a steady rate for... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | SAR-260301 | B1263 SAR260301 is a potent and selective Class I phosphatidylinositol-3-kinase-β (PI3K-β) specific inhibitor with an IC₅₀ of 52 nM for this isoform. SAR260301 displays improved physicochemical and in... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | BAY 87-2243 | B1878 BAY 87-2243 is a highly potent and selective inhibitor of hypoxia-induced gene activation. It inhibits HIF-1α and HIF-2α protein accumulation under hypoxic conditions in non-small cell lung cancer... MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Biovision | NSC 405020 | 2682 NSC-405020 is a membrane type-I matrix metalloproteinase (MT1-MMP) inhibitor that specifically targets the hemopexin (PEX) domain rather than the catalytic domain of MT1-MMP (IC₅₀ >100 μmol/L). It... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SGC-CBP30 | 9554 SGC-CBP30 is a potent and selective CREBBP/EP300 bromodomain inhibitor with IC values of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively. SGC-CBP30 has little activity against other... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | Bromosporine | 2652 Bromosporine is a broad spectrum bromodomain inhibitor (IC₅₀s = 0.41 µM, 0.29 µM, 0.122 µM and 0.017 µM for BRD2, BRD4, BRD9 and CECR2, respectively). At 1 µM, Bromosporine accelerates FRAP recovery... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | UNC2881 | 2837 UNC2881 is a potent Mer kinase inhibitor. It inhibits steady-state Mer kinase phosphorylation with an IC₅₀ value of 22 nM. Treatment with UNC2281 is also sufficient to block EGF-mediated stimulation... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | HG-9-91-01 | B1849 HG-9-91-01 is a potent, selective, ATP-competitive, pan-SIK (salt-inducible kinases) inhibitor with IC₅₀ values of 0.92 nM, 6.6n M and 9.6 nM for SIK1, SIK2, SIK3, respectively.HG-9-91-01 is a... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | PF-4708671 | 9460 PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) with a Ki of 20 nM and IC₅₀ of 160 nM. PF-4708671 prevents the S6K1-mediated phosphorylation of S6 protein in... MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Biovision | TAK-632 | 2473 A selective pan-RAF inhibitor with IC₅₀ Values: 2.4 nM (BRAF V600E); 1.4 nM (C-RAF); 160 nM (VEGFR). TAK-632 displays significant cellular activity against mutated BRAF or mutated NRAS cancer cell... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Erastin | 2231 Erastin is a selective antitumor agent that displays greater lethality in human tumour cells harbouring mutations in the oncogenes HRAS, KRAS or BRAF. It binds to mitochondrial volatage-dependent... MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Biovision | Valdecoxib | B1991 Valdecoxib is a non-steroidal anti-inflammatory drug (NSAID), that acts as a potent and selective inhibitor of cyclooxygenase-2 (COX-2) (IC₅₀ = 5 nM).Valdecoxib is a non-steroidal anti-inflammatory... MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Biovision | Necrostatin-1 | 1864 Inhibits necroptosis, a non-apoptotic cell death pathway. Does not inhibit FAS-induced apoptosis and has no effect on apoptotic morphology. Inhibits RIP1 kinase, the key upstream kinase involved in... MSRP: Was: Now: £410 - £968 Choose Options Compare Quick view Details Biovision | BV6 | B1332 MSRP: Was: Now: £738 - £2,214 Choose Options Compare Quick view Details Biovision | Nexturastat A | 2098 MSRP: Now: £592 Add to Cart Compare Quick view Details Biovision | TAPI-1 | 2068 MSRP: Now: £1,214 Add to Cart Compare Quick view Details Biovision | CNX-1351 | B1673 MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | PFI-1 | 2203 MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Details Biovision | VS-5584 | 9603 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Details Biovision | Nimorazole | 9521 MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Details Biovision | Arglabin | 9691 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | SM-164 | B1816 MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3-A20 | 2850 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3 | 2849 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | DBeQ | 1858 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | X-GAL | 2671 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Luminol | B1807 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected × OK
Quick view Biovision | TAPI-1 | 2068 Inhibitor of TNF-α processing (IC₅₀ = 100 nM), similar to TAPI-0 (Cat. No. 2067-1), but more stable in tissue culture and in vivo. Inhibits TACE and other metalloproteases. Blocks release of TNF- α... MSRP: Now: £1,214 Add to Cart Compare Quick view Biovision | CNX-1351 | B1673 CNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMCNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMBiovision | B1673 | CNX-1351... MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Biovision | Brefeldin A | 1560 Brefeldin A has been shown to induce apoptosis in human tumor cells through caspase activation. It has also been shown to block translocation of proteins from the endoplasmic reticulum to the Golgi... MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Biovision | Birinapant | 2597 Birinapant is a SMAC (synthetic small molecule and peptidomimetic of second mitochondrial-derived activator of caspases) mimetic and IAP (Inhibitor of Apoptosis Protein) antagonist with potential... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | PFI-1 | 2203 PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC₅₀... MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Biovision | VS-5584 | 9603 VS-5584 is a potent and selective PI3K/mTOR kinase inhibitor. It inhibits mTOR (IC₅₀ = 37 nM) and PI3K (IC₅₀s = 16, 68, 25, and 42 nM for the α, β, γ, and δ isoforms, respectively) without relevant... MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Biovision | Sapacitabine | B2002 Sapacitabine is an orally bioavailable nucleoside analog prodrug that is potentially useful for treatment of hematologic malignancies and solid tumors. The active metabolite of sapacitabine, CNDAC... MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Biovision | Briciclib | B1140 Briciclib is a small molecule that suppresses cyclin D1 accumulation in cancer cells. Cyclin D, a member of the cyclin family of cell cycle regulators, plays a key role in cell cycle division and is... MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Biovision | Nimorazole | 9521 Nimorazole is a 5-nitroimidazole derivative that displays antimicrobial activity. Used in the treatment of intestinal protozoal infections. Also acts as a hypoxic radiosensitizer.Nimorazole is a... MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Biovision | Kartogenin | 2066 Cell-permeable. Kartogenin promotes the selective differentiation of multipotent mesenchymal stem cells into chondrocytes (EC₅₀ = 100 nM). Displays chondroprotective effects in vitro and is... MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Biovision | Ethynylcytidine | B1266 Ethynylcytidine is a synthetic cytidine nucleoside containing a covalently bound ethynyl group with potential antineoplastic and radiosensitizing activities. Ethynylcytidine is metabolized in tumor... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | Cilengitide | B2365 Cilengitide is a cyclo-(Arg-Gly-Asp-D-Phe-Val) (cRGDfV) peptide that acts as an integrin αVβ3 receptor antagonist. It inhibits adhesion and induces apoptosis of U87MG and U373MG malignant glioma (MG)... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | BMS-303141 | 2821 BMS-303141 is a potent inhibitor of ATP citrate lyase (ACL) (IC₅₀ = 0.13 µM for human recombinant ACL). BMS-303141 inhibits lipid synthesis in HepG2 cells with an IC₅₀ of 8 μM, and lowers plasma... MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Biovision | Arglabin | 9691 Arglabin is a potent anti-inflammatory and anticancer agent. It also acts as a Farnesyltransferase inhibitor and antiatherogenic compound. Prevents the accumulation of lipid containing plaques in... MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Biovision | ACTB-1003 | B2016 ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2 and 4 nM for FGFR1, VEGFR2 and Tie-2, respectively. Displays anticancer activities.ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2... MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Biovision | Citarinostat | B1560 Citarinostat (ACY-241), is a potent, selective and orally available histone deacetylase 6 (HDAC6) inhibitor with IC₅₀ values of 4 nM and 76 nM for HDAC6 and HDAC3, respectively. Displays... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | SM-164 | B1816 SM-164 is a potent cell-permeable and bivalent Smac mimetic which binds to a XIAP protein with a Ki value of 0.56 nM, and binds to cIAP-1 and cIAP-2 proteins with Ki values of 0.31 and 1.1 nM,... MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Biovision | CTx-0294885 | 9435 CTx-0294885 is a broad-spectrum kinase inhibitor. CTx-0294885 displays inhibitory activity against a broad range of kinases in vitro. CTx-0294885 could be a potentially powerful new tool for analysis... MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Biovision | P7C3-A20 | 2850 P7C3-A20 is a derivative of P7C3 (Cat. No. 2849), and is a proneurogenic, neuroprotective agent. P7C3-A20 displays increased activity and an improved toxicity profile compared to P7C3... MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Biovision | P7C3 | 2849 P7C3 is an aminopropyl carbazole derivative that acts as a proneurogenic, neuroprotective compound. Protects newborn neurons in the dentate gyrus by mitigating cell death. Also enhances learning and... MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Biovision | Uprosertib | B1760 Uprosertib, also known as GSK2141795 and GSK795, is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity.Uprosertib,... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | DBeQ | 1858 Cell- permeable. A potent, selective, reversible, and ATP-competitive p97 inhibitor. DBeQ blocks both ubiquitin-dependent and autophagic protein clearance pathways and rapidly promotes executioner... MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Biovision | X-GAL | 2671 X-GAL is a useful chromogenic substrate for β-galactosidase that produces a rich blue color that can easily be detected visually over background. X-GAL is used to indicate whether a cell expresses... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | Luminol | B1807 Luminol is a useful probe that displays chemiluminescence upon oxidation. Horseradish peroxidase (HRP), combined with hydrogen peroxide as an activator, causes luminescent peroxidation of luminol... MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Biovision | DTT | 1201 An excellent reagent for maintaining SH groups in reduced state. DTT quantitatively reduces disulfides. It is effective in sample buffers for reducing protein disulfide bonds prior to SDSPAGE.DTT is... MSRP: Now: £462 Add to Cart Compare Quick view Biovision | DTE | B2410 A useful reagent for maintaining sulfhydryl groups in the reduced stateDTE is a useful reagent for maintaining sulfhydryl groups in the reduced stateBiovision | B2410 | DTE DataSheetAlternate... MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Biovision | Y-320 | B1164 Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T cells stimulated with IL-15 with IC50 values of 20 to 60 nM.Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | DMOG | 2216 A cell-permeable prolyl 4-hydroxylase (P4H) inhibitor; inhibits hypoxia-inducible factor α (HIF-α) prolyl hydroxylase (HIF-PH). Increases levels of HIF-1α; promotes cell survival under hypoxic... MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Biovision | PTC-209 | B1055 PTC-209 is a potent, cell-permeable, BMI-1 inhibitor (IC₅₀ = 0.5 µM) with potential anticancer activity. PTC-209 lowers the self-renewal properties of colorectal cancer-initiating cells (CICs)... MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Biovision | TCS JNK 5a | B1688 TCS JNK 5a (JNK Inhibitor IX) is a selective inhibitor of JNK2 and JNK3; displays no significant activity at a range of other protein kinases including EGFR, ErbB2, cdk2, PLK-1 and Src (pIC50 < 5.0)... MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Biovision | Inauhzin | 9555 Inauhzin is a potent SIRT inhibitor that effectively reactivates p53 by inhibiting SIRT1 activity. Inauhzin inhibits cell proliferation, induces senescence, and p53-dependent apoptosis of human... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | HS-173 | B1627 HS-173 is a novel PI3K inhibitor, that is used for cancer treatment. HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on cancer cells.HS-173 is a novel PI3K... MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Biovision | FLI-06 | 2603 A potent Notch signaling (EC₅₀ = 2.3 µM) as well as the early secretory pathway inhibitor. FLI-06 leads to a disruption of the Golgi by a mechanism different from Brefeldin A (Cat. No. 1560) or other... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Atglistatin | B1864 Atglistatin is a potent, and selective inhibitor of adipose triglyceride lipase (ATGL) the rate limiting enzyme involved in fatty acid mobilization and prevention of lipolysis. It does not inhibit... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | AdipoRon | 2565 A potent and selective adiponectin receptor agonist (Kd = 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively). Displays similar effects to adiponectin in muscle and liver such as activation of... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | CPI-203 | 9404 CPI-203 is an analog of (+)-JQ1 (Cat. No. 2070). Acts as a BET bromodomain inhibitor. It is comparable or superior to (+)-JQ1 in inhibiting BRD4 binding and action in vitro or in cells.CPI-203... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SF1670 | 2774 SF1670 is a selective PTEN (phosphatase and tensin homolog) inhibitor (IC₅₀ = 2 µM). It specifically binds to the active site of PTEN. At nanomolar concentrations it increases cellular... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | ID-8 | 2562 ID-8 is a cell culture supplement that can sustain self-renewal and pluripotency of mouse embryonic stem cells in vitro. At 10 μM it stimulates proliferation in serum-free media at a steady rate for... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | SAR-260301 | B1263 SAR260301 is a potent and selective Class I phosphatidylinositol-3-kinase-β (PI3K-β) specific inhibitor with an IC₅₀ of 52 nM for this isoform. SAR260301 displays improved physicochemical and in... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | BAY 87-2243 | B1878 BAY 87-2243 is a highly potent and selective inhibitor of hypoxia-induced gene activation. It inhibits HIF-1α and HIF-2α protein accumulation under hypoxic conditions in non-small cell lung cancer... MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Biovision | NSC 405020 | 2682 NSC-405020 is a membrane type-I matrix metalloproteinase (MT1-MMP) inhibitor that specifically targets the hemopexin (PEX) domain rather than the catalytic domain of MT1-MMP (IC₅₀ >100 μmol/L). It... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SGC-CBP30 | 9554 SGC-CBP30 is a potent and selective CREBBP/EP300 bromodomain inhibitor with IC values of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively. SGC-CBP30 has little activity against other... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | Bromosporine | 2652 Bromosporine is a broad spectrum bromodomain inhibitor (IC₅₀s = 0.41 µM, 0.29 µM, 0.122 µM and 0.017 µM for BRD2, BRD4, BRD9 and CECR2, respectively). At 1 µM, Bromosporine accelerates FRAP recovery... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | UNC2881 | 2837 UNC2881 is a potent Mer kinase inhibitor. It inhibits steady-state Mer kinase phosphorylation with an IC₅₀ value of 22 nM. Treatment with UNC2281 is also sufficient to block EGF-mediated stimulation... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | HG-9-91-01 | B1849 HG-9-91-01 is a potent, selective, ATP-competitive, pan-SIK (salt-inducible kinases) inhibitor with IC₅₀ values of 0.92 nM, 6.6n M and 9.6 nM for SIK1, SIK2, SIK3, respectively.HG-9-91-01 is a... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | PF-4708671 | 9460 PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) with a Ki of 20 nM and IC₅₀ of 160 nM. PF-4708671 prevents the S6K1-mediated phosphorylation of S6 protein in... MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Biovision | TAK-632 | 2473 A selective pan-RAF inhibitor with IC₅₀ Values: 2.4 nM (BRAF V600E); 1.4 nM (C-RAF); 160 nM (VEGFR). TAK-632 displays significant cellular activity against mutated BRAF or mutated NRAS cancer cell... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Erastin | 2231 Erastin is a selective antitumor agent that displays greater lethality in human tumour cells harbouring mutations in the oncogenes HRAS, KRAS or BRAF. It binds to mitochondrial volatage-dependent... MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Biovision | Valdecoxib | B1991 Valdecoxib is a non-steroidal anti-inflammatory drug (NSAID), that acts as a potent and selective inhibitor of cyclooxygenase-2 (COX-2) (IC₅₀ = 5 nM).Valdecoxib is a non-steroidal anti-inflammatory... MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Biovision | Necrostatin-1 | 1864 Inhibits necroptosis, a non-apoptotic cell death pathway. Does not inhibit FAS-induced apoptosis and has no effect on apoptotic morphology. Inhibits RIP1 kinase, the key upstream kinase involved in... MSRP: Was: Now: £410 - £968 Choose Options Compare Quick view Details Biovision | BV6 | B1332 MSRP: Was: Now: £738 - £2,214 Choose Options Compare Quick view Details Biovision | Nexturastat A | 2098 MSRP: Now: £592 Add to Cart Compare Quick view Details Biovision | TAPI-1 | 2068 MSRP: Now: £1,214 Add to Cart Compare Quick view Details Biovision | CNX-1351 | B1673 MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | PFI-1 | 2203 MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Details Biovision | VS-5584 | 9603 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Details Biovision | Nimorazole | 9521 MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Details Biovision | Arglabin | 9691 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | SM-164 | B1816 MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3-A20 | 2850 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3 | 2849 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | DBeQ | 1858 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | X-GAL | 2671 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Luminol | B1807 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected × OK
Quick view Biovision | CNX-1351 | B1673 CNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMCNX1351 is a potent and selective inhibitor of PI3Kα with IC50 value of 6.8 nMBiovision | B1673 | CNX-1351... MSRP: Was: Now: £494 - £1,478 Choose Options Compare
Quick view Biovision | Brefeldin A | 1560 Brefeldin A has been shown to induce apoptosis in human tumor cells through caspase activation. It has also been shown to block translocation of proteins from the endoplasmic reticulum to the Golgi... MSRP: Was: Now: £486 - £1,428 Choose Options Compare
Quick view Biovision | Birinapant | 2597 Birinapant is a SMAC (synthetic small molecule and peptidomimetic of second mitochondrial-derived activator of caspases) mimetic and IAP (Inhibitor of Apoptosis Protein) antagonist with potential... MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Biovision | PFI-1 | 2203 PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC₅₀... MSRP: Was: Now: £364 - £836 Choose Options Compare
Quick view Biovision | VS-5584 | 9603 VS-5584 is a potent and selective PI3K/mTOR kinase inhibitor. It inhibits mTOR (IC₅₀ = 37 nM) and PI3K (IC₅₀s = 16, 68, 25, and 42 nM for the α, β, γ, and δ isoforms, respectively) without relevant... MSRP: Was: Now: £444 - £1,262 Choose Options Compare
Quick view Biovision | Sapacitabine | B2002 Sapacitabine is an orally bioavailable nucleoside analog prodrug that is potentially useful for treatment of hematologic malignancies and solid tumors. The active metabolite of sapacitabine, CNDAC... MSRP: Was: Now: £904 - £3,098 Choose Options Compare
Quick view Biovision | Briciclib | B1140 Briciclib is a small molecule that suppresses cyclin D1 accumulation in cancer cells. Cyclin D, a member of the cyclin family of cell cycle regulators, plays a key role in cell cycle division and is... MSRP: Was: Now: £708 - £2,214 Choose Options Compare
Quick view Biovision | Nimorazole | 9521 Nimorazole is a 5-nitroimidazole derivative that displays antimicrobial activity. Used in the treatment of intestinal protozoal infections. Also acts as a hypoxic radiosensitizer.Nimorazole is a... MSRP: Was: Now: £410 - £806 Choose Options Compare
Quick view Biovision | Kartogenin | 2066 Cell-permeable. Kartogenin promotes the selective differentiation of multipotent mesenchymal stem cells into chondrocytes (EC₅₀ = 100 nM). Displays chondroprotective effects in vitro and is... MSRP: Was: Now: £462 - £1,344 Choose Options Compare
Quick view Biovision | Ethynylcytidine | B1266 Ethynylcytidine is a synthetic cytidine nucleoside containing a covalently bound ethynyl group with potential antineoplastic and radiosensitizing activities. Ethynylcytidine is metabolized in tumor... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | Cilengitide | B2365 Cilengitide is a cyclo-(Arg-Gly-Asp-D-Phe-Val) (cRGDfV) peptide that acts as an integrin αVβ3 receptor antagonist. It inhibits adhesion and induces apoptosis of U87MG and U373MG malignant glioma (MG)... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Biovision | BMS-303141 | 2821 BMS-303141 is a potent inhibitor of ATP citrate lyase (ACL) (IC₅₀ = 0.13 µM for human recombinant ACL). BMS-303141 inhibits lipid synthesis in HepG2 cells with an IC₅₀ of 8 μM, and lowers plasma... MSRP: Was: Now: £640 - £2,082 Choose Options Compare
Quick view Biovision | Arglabin | 9691 Arglabin is a potent anti-inflammatory and anticancer agent. It also acts as a Farnesyltransferase inhibitor and antiatherogenic compound. Prevents the accumulation of lipid containing plaques in... MSRP: Was: Now: £772 - £2,572 Choose Options Compare
Quick view Biovision | ACTB-1003 | B2016 ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2 and 4 nM for FGFR1, VEGFR2 and Tie-2, respectively. Displays anticancer activities.ACTB-1003 is a potent kinase inhibitor with IC₅₀s of 6, 2... MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Biovision | Citarinostat | B1560 Citarinostat (ACY-241), is a potent, selective and orally available histone deacetylase 6 (HDAC6) inhibitor with IC₅₀ values of 4 nM and 76 nM for HDAC6 and HDAC3, respectively. Displays... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | SM-164 | B1816 SM-164 is a potent cell-permeable and bivalent Smac mimetic which binds to a XIAP protein with a Ki value of 0.56 nM, and binds to cIAP-1 and cIAP-2 proteins with Ki values of 0.31 and 1.1 nM,... MSRP: Was: Now: £508 - £1,082 Choose Options Compare
Quick view Biovision | CTx-0294885 | 9435 CTx-0294885 is a broad-spectrum kinase inhibitor. CTx-0294885 displays inhibitory activity against a broad range of kinases in vitro. CTx-0294885 could be a potentially powerful new tool for analysis... MSRP: Was: Now: £576 - £1,690 Choose Options Compare
Quick view Biovision | P7C3-A20 | 2850 P7C3-A20 is a derivative of P7C3 (Cat. No. 2849), and is a proneurogenic, neuroprotective agent. P7C3-A20 displays increased activity and an improved toxicity profile compared to P7C3... MSRP: Was: Now: £576 - £1,690 Choose Options Compare
Quick view Biovision | P7C3 | 2849 P7C3 is an aminopropyl carbazole derivative that acts as a proneurogenic, neuroprotective compound. Protects newborn neurons in the dentate gyrus by mitigating cell death. Also enhances learning and... MSRP: Was: Now: £606 - £1,788 Choose Options Compare
Quick view Biovision | Uprosertib | B1760 Uprosertib, also known as GSK2141795 and GSK795, is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity.Uprosertib,... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | DBeQ | 1858 Cell- permeable. A potent, selective, reversible, and ATP-competitive p97 inhibitor. DBeQ blocks both ubiquitin-dependent and autophagic protein clearance pathways and rapidly promotes executioner... MSRP: Was: Now: £478 - £1,362 Choose Options Compare
Quick view Biovision | X-GAL | 2671 X-GAL is a useful chromogenic substrate for β-galactosidase that produces a rich blue color that can easily be detected visually over background. X-GAL is used to indicate whether a cell expresses... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | Luminol | B1807 Luminol is a useful probe that displays chemiluminescence upon oxidation. Horseradish peroxidase (HRP), combined with hydrogen peroxide as an activator, causes luminescent peroxidation of luminol... MSRP: Was: Now: £380 - £904 Choose Options Compare
Quick view Biovision | DTT | 1201 An excellent reagent for maintaining SH groups in reduced state. DTT quantitatively reduces disulfides. It is effective in sample buffers for reducing protein disulfide bonds prior to SDSPAGE.DTT is... MSRP: Now: £462 Add to Cart Compare Quick view Biovision | DTE | B2410 A useful reagent for maintaining sulfhydryl groups in the reduced stateDTE is a useful reagent for maintaining sulfhydryl groups in the reduced stateBiovision | B2410 | DTE DataSheetAlternate... MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Biovision | Y-320 | B1164 Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T cells stimulated with IL-15 with IC50 values of 20 to 60 nM.Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | DMOG | 2216 A cell-permeable prolyl 4-hydroxylase (P4H) inhibitor; inhibits hypoxia-inducible factor α (HIF-α) prolyl hydroxylase (HIF-PH). Increases levels of HIF-1α; promotes cell survival under hypoxic... MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Biovision | PTC-209 | B1055 PTC-209 is a potent, cell-permeable, BMI-1 inhibitor (IC₅₀ = 0.5 µM) with potential anticancer activity. PTC-209 lowers the self-renewal properties of colorectal cancer-initiating cells (CICs)... MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Biovision | TCS JNK 5a | B1688 TCS JNK 5a (JNK Inhibitor IX) is a selective inhibitor of JNK2 and JNK3; displays no significant activity at a range of other protein kinases including EGFR, ErbB2, cdk2, PLK-1 and Src (pIC50 < 5.0)... MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Biovision | Inauhzin | 9555 Inauhzin is a potent SIRT inhibitor that effectively reactivates p53 by inhibiting SIRT1 activity. Inauhzin inhibits cell proliferation, induces senescence, and p53-dependent apoptosis of human... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | HS-173 | B1627 HS-173 is a novel PI3K inhibitor, that is used for cancer treatment. HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on cancer cells.HS-173 is a novel PI3K... MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Biovision | FLI-06 | 2603 A potent Notch signaling (EC₅₀ = 2.3 µM) as well as the early secretory pathway inhibitor. FLI-06 leads to a disruption of the Golgi by a mechanism different from Brefeldin A (Cat. No. 1560) or other... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Atglistatin | B1864 Atglistatin is a potent, and selective inhibitor of adipose triglyceride lipase (ATGL) the rate limiting enzyme involved in fatty acid mobilization and prevention of lipolysis. It does not inhibit... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | AdipoRon | 2565 A potent and selective adiponectin receptor agonist (Kd = 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively). Displays similar effects to adiponectin in muscle and liver such as activation of... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | CPI-203 | 9404 CPI-203 is an analog of (+)-JQ1 (Cat. No. 2070). Acts as a BET bromodomain inhibitor. It is comparable or superior to (+)-JQ1 in inhibiting BRD4 binding and action in vitro or in cells.CPI-203... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SF1670 | 2774 SF1670 is a selective PTEN (phosphatase and tensin homolog) inhibitor (IC₅₀ = 2 µM). It specifically binds to the active site of PTEN. At nanomolar concentrations it increases cellular... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | ID-8 | 2562 ID-8 is a cell culture supplement that can sustain self-renewal and pluripotency of mouse embryonic stem cells in vitro. At 10 μM it stimulates proliferation in serum-free media at a steady rate for... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | SAR-260301 | B1263 SAR260301 is a potent and selective Class I phosphatidylinositol-3-kinase-β (PI3K-β) specific inhibitor with an IC₅₀ of 52 nM for this isoform. SAR260301 displays improved physicochemical and in... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | BAY 87-2243 | B1878 BAY 87-2243 is a highly potent and selective inhibitor of hypoxia-induced gene activation. It inhibits HIF-1α and HIF-2α protein accumulation under hypoxic conditions in non-small cell lung cancer... MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Biovision | NSC 405020 | 2682 NSC-405020 is a membrane type-I matrix metalloproteinase (MT1-MMP) inhibitor that specifically targets the hemopexin (PEX) domain rather than the catalytic domain of MT1-MMP (IC₅₀ >100 μmol/L). It... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | SGC-CBP30 | 9554 SGC-CBP30 is a potent and selective CREBBP/EP300 bromodomain inhibitor with IC values of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively. SGC-CBP30 has little activity against other... MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Biovision | Bromosporine | 2652 Bromosporine is a broad spectrum bromodomain inhibitor (IC₅₀s = 0.41 µM, 0.29 µM, 0.122 µM and 0.017 µM for BRD2, BRD4, BRD9 and CECR2, respectively). At 1 µM, Bromosporine accelerates FRAP recovery... MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Biovision | UNC2881 | 2837 UNC2881 is a potent Mer kinase inhibitor. It inhibits steady-state Mer kinase phosphorylation with an IC₅₀ value of 22 nM. Treatment with UNC2281 is also sufficient to block EGF-mediated stimulation... MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Biovision | HG-9-91-01 | B1849 HG-9-91-01 is a potent, selective, ATP-competitive, pan-SIK (salt-inducible kinases) inhibitor with IC₅₀ values of 0.92 nM, 6.6n M and 9.6 nM for SIK1, SIK2, SIK3, respectively.HG-9-91-01 is a... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | PF-4708671 | 9460 PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) with a Ki of 20 nM and IC₅₀ of 160 nM. PF-4708671 prevents the S6K1-mediated phosphorylation of S6 protein in... MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Biovision | TAK-632 | 2473 A selective pan-RAF inhibitor with IC₅₀ Values: 2.4 nM (BRAF V600E); 1.4 nM (C-RAF); 160 nM (VEGFR). TAK-632 displays significant cellular activity against mutated BRAF or mutated NRAS cancer cell... MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Biovision | Erastin | 2231 Erastin is a selective antitumor agent that displays greater lethality in human tumour cells harbouring mutations in the oncogenes HRAS, KRAS or BRAF. It binds to mitochondrial volatage-dependent... MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Biovision | Valdecoxib | B1991 Valdecoxib is a non-steroidal anti-inflammatory drug (NSAID), that acts as a potent and selective inhibitor of cyclooxygenase-2 (COX-2) (IC₅₀ = 5 nM).Valdecoxib is a non-steroidal anti-inflammatory... MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Biovision | Necrostatin-1 | 1864 Inhibits necroptosis, a non-apoptotic cell death pathway. Does not inhibit FAS-induced apoptosis and has no effect on apoptotic morphology. Inhibits RIP1 kinase, the key upstream kinase involved in... MSRP: Was: Now: £410 - £968 Choose Options Compare Quick view Details Biovision | BV6 | B1332 MSRP: Was: Now: £738 - £2,214 Choose Options Compare Quick view Details Biovision | Nexturastat A | 2098 MSRP: Now: £592 Add to Cart Compare Quick view Details Biovision | TAPI-1 | 2068 MSRP: Now: £1,214 Add to Cart Compare Quick view Details Biovision | CNX-1351 | B1673 MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | PFI-1 | 2203 MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Details Biovision | VS-5584 | 9603 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Details Biovision | Nimorazole | 9521 MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Details Biovision | Arglabin | 9691 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | SM-164 | B1816 MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3-A20 | 2850 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3 | 2849 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | DBeQ | 1858 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | X-GAL | 2671 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Luminol | B1807 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected × OK
Quick view Biovision | DTE | B2410 A useful reagent for maintaining sulfhydryl groups in the reduced stateDTE is a useful reagent for maintaining sulfhydryl groups in the reduced stateBiovision | B2410 | DTE DataSheetAlternate... MSRP: Was: Now: £444 - £2,278 Choose Options Compare
Quick view Biovision | Y-320 | B1164 Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T cells stimulated with IL-15 with IC50 values of 20 to 60 nM.Y-320 is an immunomodulator. Y-320 inhibits IL-17 production by CD4 T... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | DMOG | 2216 A cell-permeable prolyl 4-hydroxylase (P4H) inhibitor; inhibits hypoxia-inducible factor α (HIF-α) prolyl hydroxylase (HIF-PH). Increases levels of HIF-1α; promotes cell survival under hypoxic... MSRP: Was: Now: £364 - £904 Choose Options Compare
Quick view Biovision | PTC-209 | B1055 PTC-209 is a potent, cell-permeable, BMI-1 inhibitor (IC₅₀ = 0.5 µM) with potential anticancer activity. PTC-209 lowers the self-renewal properties of colorectal cancer-initiating cells (CICs)... MSRP: Was: Now: £606 - £1,788 Choose Options Compare
Quick view Biovision | TCS JNK 5a | B1688 TCS JNK 5a (JNK Inhibitor IX) is a selective inhibitor of JNK2 and JNK3; displays no significant activity at a range of other protein kinases including EGFR, ErbB2, cdk2, PLK-1 and Src (pIC50 < 5.0)... MSRP: Was: Now: £380 - £1,164 Choose Options Compare
Quick view Biovision | Inauhzin | 9555 Inauhzin is a potent SIRT inhibitor that effectively reactivates p53 by inhibiting SIRT1 activity. Inauhzin inhibits cell proliferation, induces senescence, and p53-dependent apoptosis of human... MSRP: Was: Now: £806 - £2,772 Choose Options Compare
Quick view Biovision | HS-173 | B1627 HS-173 is a novel PI3K inhibitor, that is used for cancer treatment. HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on cancer cells.HS-173 is a novel PI3K... MSRP: Was: Now: £462 - £1,330 Choose Options Compare
Quick view Biovision | FLI-06 | 2603 A potent Notch signaling (EC₅₀ = 2.3 µM) as well as the early secretory pathway inhibitor. FLI-06 leads to a disruption of the Golgi by a mechanism different from Brefeldin A (Cat. No. 1560) or other... MSRP: Was: Now: £576 - £1,754 Choose Options Compare
Quick view Biovision | Atglistatin | B1864 Atglistatin is a potent, and selective inhibitor of adipose triglyceride lipase (ATGL) the rate limiting enzyme involved in fatty acid mobilization and prevention of lipolysis. It does not inhibit... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | AdipoRon | 2565 A potent and selective adiponectin receptor agonist (Kd = 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively). Displays similar effects to adiponectin in muscle and liver such as activation of... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | CPI-203 | 9404 CPI-203 is an analog of (+)-JQ1 (Cat. No. 2070). Acts as a BET bromodomain inhibitor. It is comparable or superior to (+)-JQ1 in inhibiting BRD4 binding and action in vitro or in cells.CPI-203... MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Biovision | SF1670 | 2774 SF1670 is a selective PTEN (phosphatase and tensin homolog) inhibitor (IC₅₀ = 2 µM). It specifically binds to the active site of PTEN. At nanomolar concentrations it increases cellular... MSRP: Was: Now: £478 - £1,394 Choose Options Compare
Quick view Biovision | ID-8 | 2562 ID-8 is a cell culture supplement that can sustain self-renewal and pluripotency of mouse embryonic stem cells in vitro. At 10 μM it stimulates proliferation in serum-free media at a steady rate for... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | SAR-260301 | B1263 SAR260301 is a potent and selective Class I phosphatidylinositol-3-kinase-β (PI3K-β) specific inhibitor with an IC₅₀ of 52 nM for this isoform. SAR260301 displays improved physicochemical and in... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | BAY 87-2243 | B1878 BAY 87-2243 is a highly potent and selective inhibitor of hypoxia-induced gene activation. It inhibits HIF-1α and HIF-2α protein accumulation under hypoxic conditions in non-small cell lung cancer... MSRP: Was: Now: £806 - £2,704 Choose Options Compare
Quick view Biovision | NSC 405020 | 2682 NSC-405020 is a membrane type-I matrix metalloproteinase (MT1-MMP) inhibitor that specifically targets the hemopexin (PEX) domain rather than the catalytic domain of MT1-MMP (IC₅₀ >100 μmol/L). It... MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Biovision | SGC-CBP30 | 9554 SGC-CBP30 is a potent and selective CREBBP/EP300 bromodomain inhibitor with IC values of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively. SGC-CBP30 has little activity against other... MSRP: Was: Now: £806 - £2,772 Choose Options Compare
Quick view Biovision | Bromosporine | 2652 Bromosporine is a broad spectrum bromodomain inhibitor (IC₅₀s = 0.41 µM, 0.29 µM, 0.122 µM and 0.017 µM for BRD2, BRD4, BRD9 and CECR2, respectively). At 1 µM, Bromosporine accelerates FRAP recovery... MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Biovision | UNC2881 | 2837 UNC2881 is a potent Mer kinase inhibitor. It inhibits steady-state Mer kinase phosphorylation with an IC₅₀ value of 22 nM. Treatment with UNC2281 is also sufficient to block EGF-mediated stimulation... MSRP: Was: Now: £478 - £1,394 Choose Options Compare
Quick view Biovision | HG-9-91-01 | B1849 HG-9-91-01 is a potent, selective, ATP-competitive, pan-SIK (salt-inducible kinases) inhibitor with IC₅₀ values of 0.92 nM, 6.6n M and 9.6 nM for SIK1, SIK2, SIK3, respectively.HG-9-91-01 is a... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Biovision | PF-4708671 | 9460 PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) with a Ki of 20 nM and IC₅₀ of 160 nM. PF-4708671 prevents the S6K1-mediated phosphorylation of S6 protein in... MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Biovision | TAK-632 | 2473 A selective pan-RAF inhibitor with IC₅₀ Values: 2.4 nM (BRAF V600E); 1.4 nM (C-RAF); 160 nM (VEGFR). TAK-632 displays significant cellular activity against mutated BRAF or mutated NRAS cancer cell... MSRP: Was: Now: £576 - £1,754 Choose Options Compare
Quick view Biovision | Erastin | 2231 Erastin is a selective antitumor agent that displays greater lethality in human tumour cells harbouring mutations in the oncogenes HRAS, KRAS or BRAF. It binds to mitochondrial volatage-dependent... MSRP: Was: Now: £606 - £16,240 Choose Options Compare
Quick view Biovision | Valdecoxib | B1991 Valdecoxib is a non-steroidal anti-inflammatory drug (NSAID), that acts as a potent and selective inhibitor of cyclooxygenase-2 (COX-2) (IC₅₀ = 5 nM).Valdecoxib is a non-steroidal anti-inflammatory... MSRP: Was: Now: £576 - £1,722 Choose Options Compare
Quick view Biovision | Necrostatin-1 | 1864 Inhibits necroptosis, a non-apoptotic cell death pathway. Does not inhibit FAS-induced apoptosis and has no effect on apoptotic morphology. Inhibits RIP1 kinase, the key upstream kinase involved in... MSRP: Was: Now: £410 - £968 Choose Options Compare
Quick view Details Biovision | Nexturastat A | 2098 MSRP: Now: £592 Add to Cart Compare Quick view Details Biovision | TAPI-1 | 2068 MSRP: Now: £1,214 Add to Cart Compare Quick view Details Biovision | CNX-1351 | B1673 MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | PFI-1 | 2203 MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Details Biovision | VS-5584 | 9603 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Details Biovision | Nimorazole | 9521 MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Details Biovision | Arglabin | 9691 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | SM-164 | B1816 MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3-A20 | 2850 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3 | 2849 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | DBeQ | 1858 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | X-GAL | 2671 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Luminol | B1807 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected × OK
Quick view Details Biovision | TAPI-1 | 2068 MSRP: Now: £1,214 Add to Cart Compare Quick view Details Biovision | CNX-1351 | B1673 MSRP: Was: Now: £494 - £1,478 Choose Options Compare Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | PFI-1 | 2203 MSRP: Was: Now: £364 - £836 Choose Options Compare Quick view Details Biovision | VS-5584 | 9603 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare Quick view Details Biovision | Nimorazole | 9521 MSRP: Was: Now: £410 - £806 Choose Options Compare Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare Quick view Details Biovision | Arglabin | 9691 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | SM-164 | B1816 MSRP: Was: Now: £508 - £1,082 Choose Options Compare Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3-A20 | 2850 MSRP: Was: Now: £576 - £1,690 Choose Options Compare Quick view Details Biovision | P7C3 | 2849 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | DBeQ | 1858 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | X-GAL | 2671 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Luminol | B1807 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected
Quick view Details Biovision | Brefeldin A | 1560 MSRP: Was: Now: £486 - £1,428 Choose Options Compare
Quick view Details Biovision | Birinapant | 2597 MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Details Biovision | Sapacitabine | B2002 MSRP: Was: Now: £904 - £3,098 Choose Options Compare
Quick view Details Biovision | Briciclib | B1140 MSRP: Was: Now: £708 - £2,214 Choose Options Compare
Quick view Details Biovision | Kartogenin | 2066 MSRP: Was: Now: £462 - £1,344 Choose Options Compare
Quick view Details Biovision | Ethynylcytidine | B1266 MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Details Biovision | Cilengitide | B2365 MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Details Biovision | BMS-303141 | 2821 MSRP: Was: Now: £640 - £2,082 Choose Options Compare
Quick view Details Biovision | ACTB-1003 | B2016 MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Details Biovision | Citarinostat | B1560 MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Details Biovision | CTx-0294885 | 9435 MSRP: Was: Now: £576 - £1,690 Choose Options Compare
Quick view Details Biovision | Uprosertib | B1760 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | DTT | 1201 MSRP: Now: £462 Add to Cart Compare Quick view Details Biovision | DTE | B2410 MSRP: Was: Now: £444 - £2,278 Choose Options Compare Quick view Details Biovision | Y-320 | B1164 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | DMOG | 2216 MSRP: Was: Now: £364 - £904 Choose Options Compare Quick view Details Biovision | PTC-209 | B1055 MSRP: Was: Now: £606 - £1,788 Choose Options Compare Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare Quick view Details Biovision | Inauhzin | 9555 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | HS-173 | B1627 MSRP: Was: Now: £462 - £1,330 Choose Options Compare Quick view Details Biovision | FLI-06 | 2603 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | AdipoRon | 2565 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | CPI-203 | 9404 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SF1670 | 2774 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | ID-8 | 2562 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | SGC-CBP30 | 9554 MSRP: Was: Now: £806 - £2,772 Choose Options Compare Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare Quick view Details Biovision | UNC2881 | 2837 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | TAK-632 | 2473 MSRP: Was: Now: £576 - £1,754 Choose Options Compare Quick view Details Biovision | Erastin | 2231 MSRP: Was: Now: £606 - £16,240 Choose Options Compare Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare Previous 180 181 182 183 184 185 186 187 188 189 190 Next Previous 180 181 182 183 184 185 186 187 188 189 190 Next Compare Selected
Quick view Details Biovision | TCS JNK 5a | B1688 MSRP: Was: Now: £380 - £1,164 Choose Options Compare
Quick view Details Biovision | Atglistatin | B1864 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | SAR-260301 | B1263 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | BAY 87-2243 | B1878 MSRP: Was: Now: £806 - £2,704 Choose Options Compare
Quick view Details Biovision | NSC 405020 | 2682 MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Details Biovision | Bromosporine | 2652 MSRP: Was: Now: £410 - £1,134 Choose Options Compare
Quick view Details Biovision | HG-9-91-01 | B1849 MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Details Biovision | PF-4708671 | 9460 MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Details Biovision | Valdecoxib | B1991 MSRP: Was: Now: £576 - £1,722 Choose Options Compare
Quick view Details Biovision | Necrostatin-1 | 1864 MSRP: Was: Now: £410 - £968 Choose Options Compare