Quick view Biovision | GSK-J4 hydrochloride | 2259 Cell-permeable. An ethyl ester derivative of the JMJD3 selective histone demethylase inhibitor GSK-J1 (Cat. No. 2260-1, 5) (IC₅₀> 50 μM in vitro. When administered to human primary macrophages,... MSRP: Was: Now: £364 - £806 Choose Options Compare
Quick view Biovision | GSK-J4 (Free base) | 2762 GSK- J4 is cell-permeable ethyl ester of GSK-J1 (Cat. Nos. 2260 & 2761). Acts as a histone demethylase JMJD3/UTX inhibitor. Inhibits demethylation of histone H3K27. Reduces LPS-induced... MSRP: Was: Now: £380 - £806 Choose Options Compare
Quick view Biovision | GSK-J1 sodium salt | 2260 A potent and selective inhibitor of the H3K27 histone demethylases JMJD3 and UTX (IC₅₀ = 60 nM for human JMJD3 in vitro). It is inactive against a panel of other JMJ family demethylases, including... MSRP: Was: Now: £364 - £806 Choose Options Compare
Quick view Biovision | GSK-J1 (Free acid) | 2761 GSK-J1 is a potent and selective inhibitor of jumonji H3K27 histone demethylases JMJD3 and UTX (IC₅₀ = 60 nM, human JMJD3). This is the first known inhibitor selective for the H3K27me3-specific JMJ... MSRP: Was: Now: £380 - £806 Choose Options Compare
Quick view Biovision | GSK-961081 | B1590 GSK-961081 is a bi-functional molecule with both muscarinic antagonism and β2-agonism (MABA) properties. GSK-961081 displays high affinity for hM2 (Ki = 1.4 nM), hM3 muscarinic receptors (Ki = 1.3... MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Biovision | GSK-650394 | B2093 GSK-650394 is a potent inhibitor of serum- and glucocorticoid-regulated kinase (IC₅₀s = 62 and 103 nM for SGK1 and SGK2, respectively). It demonstrates greater than 30-fold selectivity for SGK1 over... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Biovision | GSK-583 | B1301 GSK-583 is a highly potent and selective Inhibitor of RIP2 Kinase (IC₅₀ = 5 nM). RIP2 kinase is a central component of the innate immune system and enables downstream signaling following activation... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | GSK-503 | 9538 GSK-503 is a potent EZH2 inhibitor with potential anticancer activity. Increased activity of the epigenetic modifier EZH2 has been associated with different cancers. In a melanoma mouse model,... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GSK-484 hydrochloride | B1035 GSK-484 is a potent and reversible inhibitor of PAD4 (Protein Arginine Deiminase 4) (IC₅₀ = 50 nM) that binds to the low-calcium form of the enzyme. It is selective for PAD4 over PAD1-3. GSK-484... MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Biovision | GSK-4112 | 9663 GSK-4112 is a selective agonist for REV-ERBα (EC₅₀ = 0.4 μM). At 10 μM, GSK-4112 can reset the circadian rhythm in a phasic manner by inhibiting expression of the circadian target gene bmal1 and... MSRP: Was: Now: £542 - £1,558 Choose Options Compare
Quick view Biovision | GSK-3787 | 2400 GSK-3787 is a selective and irreversible antagonist of the peroxisome proliferator-activated receptor delta (PPARδ) (plC₅₀ = 6.6). It covalently binds to Cys 249 in the PPARδ binding site.GSK-3787 is... MSRP: Was: Now: £478 - £1,394 Choose Options Compare
Quick view Biovision | GSK-3117391 | B2375 GSK-3117391 is a potent histone deacetylase (HDAC) inhibitorGSK-3117391 is a potent histone deacetylase (HDAC) inhibitorBiovision | B2375 | GSK-3117391 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Biovision | GSK-3039294 | B2374 GSK-3039294 is a potent small molecule inhibitor of serum amyloid P component (SAP) binding to amyloid fibrils for the depletion of serum amyloid-P (SAP) component from the circulation.GSK-3039294 is... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | GSK-3 Inhibitor, AR-A014418 | 1953 Cell-permeable. A selective glycogen synthase kinase 3 (GSK-3) inhibitor (IC₅₀ = 104 nM). Inhibition is competitive with respect to ATP (Ki = 38nM). Exhibits specificity for GSK-3 over cdk2 and cdk5... MSRP: Was: Now: £394 - £606 Choose Options Compare
Quick view Biovision | GSK-2982772 | B2232 GSK-2982772 is a potent and ATP-competitive receptor-interacting protein-1 (RIP1) kinase inhibitor (IC₅₀ = 1 nM).GSK-2982772 is a potent and ATP-competitive receptor-interacting protein-1 (RIP1)... MSRP: Was: Now: £478 - £1,394 Choose Options Compare
Quick view Biovision | GSK-2879552 | B1044 GSK-2879552 is a potent, selective, mechanism-based inactivator of Lysine Specific Demethylase 1 (LSD1)/ CoRepressor for Element-1-Silencing Transcription factor (CoREST) activity. GSK-2879552 binds... MSRP: Was: Now: £772 - £2,572 Choose Options Compare
Quick view Biovision | GSK2830371 | 2578 GSK2830371 is an allosteric Wip1 (Wild type p53-induced phosphatase) inhibitor (IC₅₀ of 6 nM). It binds to a flap subdomain that regulates Wip1's enzymatic activity and substrate recognition. Due to... MSRP: Was: Now: £444 - £1,262 Choose Options Compare
Quick view Biovision | GSK-2801 | 9553 GSK-2801 is a potent, selective and cell-permeable inhibitor of the BAZ2 family of bromodomain containing proteins. GSK-2801 binds to BAZ2 bromodomains with dissociation constants (KD) of 136 and 257... MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Biovision | GSK-269962 | 9654 GSK-269962 is a potent Rho kinase (ROCK) inhibitor (IC₅₀ values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively). Displays greater than 30-fold selectivity for ROCK against a... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | GSK-2656157 | 9466 GSK-2656157 is a potent, selective and ATP-competitive inhibitor of PERK (protein kinase R-like ER kinase) enzyme activity with an IC₅₀ of 0.9 nM; displays high selectivity for PERK against a panel... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GSK-2606414 | 9467 GSK-2606414 is a potent and selective inhibitor of protein kinase R-like ER kinase (PERK) with IC₅₀ value of 0.4 nM. Displays >1000-fold selectivity for PERK over HR1 and PKR. GSK-2606414 inhibits... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | GSK-2334470 | B1555 GSK-2334470 is a highly specific and potent inhibitor of PDK1 (3-Phosphoinositide dependent protein kinase-1) (IC₅₀ = 10 nM). It does not suppress activity on other 96 kinases, including Aurora,... MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Biovision | GSK2330672 | B1102 GSK2330672 is a highly selective, potent, nonabsorbable ASBT(Apical Sodium dependent bile acid transporter) inhibitor (IC₅₀ = 42 nM). It lowers glucose in an animal model of type 2 diabetes... MSRP: Was: Now: £640 - £1,950 Choose Options Compare
Quick view Biovision | GSK2292767 | B1660 Biovision | GSK2292767 | B1660 MSRP: Now: £372 Add to Cart Compare Quick view Biovision | GSK-2194069 | B1571 GSK-2194069 is a potent and specific inhibitor of the β-ketoacyl reductase (KR) activity of hFAS (human Fatty Acid Synthase).GSK-2194069 is a potent and specific inhibitor of the β-ketoacyl reductase... MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Biovision | GSK2190915 | B1891 GSK2190915 (Fiboflapon) is a potent FLAP (5-lipoxygenase-activating protein) inhibitor (IC₅₀ = 2.9 nM).GSK2190915 (Fiboflapon) is a potent FLAP (5-lipoxygenase-activating protein) inhibitor (IC₅₀ = 2... MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Biovision | GSK-2126458 | 1961 Cell-permeable. A highly potent, pan phosphoinositide 3-kinase (PI 3-K) family kinase inhibitor with biochemical Ki’s of 0.019 nM (PI 3-K⍺), 0.13 nM (PI 3-Kβ), 0.024 nM (PI 3-Kδ), 0.06 nM (PI 3-Kɣ),... MSRP: Was: Now: £494 - £1,460 Choose Options Compare Quick view Biovision | GSK-2118436 mesylate | 2800 GSK2118436 is a selective BRAF V600E inhibitor. GSK2118436 binds to Raf family kinases and inhibits their activity. It is highly selective against B-Raf V600E with IC₅₀ of 0.8 nM, compared to wild... MSRP: Was: Now: £444 - £1,232 Choose Options Compare Quick view Biovision | GSK-2110183 | B1089 GSK-2110183 is a potent, selective, and ATP-competitive pan-Akt inhibitor with IC₅₀s of 0.08, 2 and 2.6 nM for Akt1, Akt2, and Akt3 respectively.GSK-2110183 is a potent, selective, and... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | GSK-2018682 | B1967 GSK-2018682 is a potent sphingosine -1 phosphate receptor (S1PR)-1 agonist; useful for the treatment of multiple sclerosis. GSK-2018682 induces acute, transient and non-symptomatic decreases in heart... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | GSK-199 hydrochloride | B1037 GSK-199 is a potent, reversible inhibitor of PAD4 (IC₅₀ = 200 nM. It binds to the low-calcium form of the enzyme and is selective for PAD4 over PAD1-3. It is less potent than the related PAD4... MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Biovision | GSK-1940029 | B2373 GSK-1940029 is a potent stearoyl-coA desaturase (SCD) inhibitorGSK-1940029 is a potent stearoyl-coA desaturase (SCD) inhibitorBiovision | B2373 | GSK-1940029 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: £674 - £2,116 Choose Options Compare Quick view Biovision | GSK1349572 | 2288 A potent, second generation HIV integrase inhibitor (IC₅₀ = 2.7 nM) that displays potent antiviral activity.GSK1349572 is a potent, second generation HIV integrase inhibitor (IC₅₀ = 2.7 nM) that... MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Biovision | GSK1325756 | B1103 GSK1325756 is a selective and reversible CXCR2 antagonist with IC₅₀ value of 12.5 nM. GSK1325756 displays anti-inflammatory effects in various preclinical and clinical models.GSK1325756 is a... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | GSK-1292263 | B1556 GSK-1292263 is a novel GPR119 receptor agonist and is used for the treatment of type 2 diabetes. GSK1292263 improves glucose regulation in animal models of diabetes, but has no effect on plasma... MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Biovision | GSK1278863 | B1107 GSK-1278863 is a novel Hypoxia-Inducible Factor-Prolyl Hydroxylase Inhibitor (HIF-PHI). Hypoxia-inducible factor−prolyl hydroxylase inhibitors stimulate endogenous EPO synthesis and induce effective... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | GSK-121 trifluoroacetate | B1034 GSK-121 is a novel protein arginine deiminase 4 (PAD4) inhibitor. GSK-121 was shown to inhibit the citrullination of PAD4 target proteins in a functional assay with an IC₅₀ value of 3.2 µM.GSK-121 is... MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Biovision | GSK-1120212 | 1960 A potent and selective allosteric inhibitor of the MEK1 (IC₅₀ = 0.7 nM) and MEK2 (IC₅₀ = 0.9 nM) enzymes with potential antineoplastic activity.GSK-1120212 is a potent and selective allosteric... MSRP: Was: Now: £428 - £1,180 Choose Options Compare Quick view Biovision | GSK-106 hydrochloride | B1036 GSK-106 is a useful negative control for PAD4 inhibitors (GSK-121 and GSK-484). It does not inhibit PAD4 nor does it prevent the citrullination of PAD4 target proteins or the formation of neutrophil... MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Biovision | GSK-1059615 | 9450 GSK-1059615 is a potent, reversible, ATP-competitive inhibitor of PI3Kα (IC₅₀ = 2 nM). It inhibits proliferation in BT474 cells and attenuates MAPK signaling.GSK-1059615 is a potent, reversible,... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | GSK-0660 | 2897 GSK-0660 is a selective PPARδ antagonist (IC₅₀ values are 0.155, > 10 and ≥ 10 μM at PPARδ, PPARα and PPARγ, respectively).GSK-0660 is a selective PPARδ antagonist (IC₅₀ values are 0.155, > 10 and ≥... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Biovision | GS-9973 | 2669 GS-9973 is a potent and highly selective Syk (spleen tyrosine kinase) inhibitor (IC₅₀ = 7.7 nM).GS-9973 is a potent and highly selective Syk (spleen tyrosine kinase) inhibitor (IC₅₀ = 7.7 nM)... MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Biovision | Grazoprevir (MK-5172) | B2337 Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV)... MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Biovision | GPNA (monohydrate) | B2150 GPNA is a substrate for γ-glutamyl transpeptidase. GPNA has also been shown to be an inhibitor of glutamine uptake - solute-linked carrier family A1 member 5 (SLC1A5). Cellular uptake of L-glutamine... MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Biovision | Gossypin | 2374 A glucoside occurring in cotton and Hubiscus flowers that acts as a potent antimelanoma agent. Gossypin inhibits human melanoma cell proliferation, in vitro, in melanoma cell lines that harbors both... MSRP: Was: Now: £444 - £3,700 Choose Options Compare Quick view Biovision | GNE 477 | B1657 GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor with IC50 of 4 nM for PI3Kα, Kiapp is 21 nM for mTOR.GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor with IC50 of 4 nM for... MSRP: Was: Now: £658 - £2,032 Choose Options Compare Quick view Biovision | GN25 | 9430 GN25 blocks Snail binding to p53 and induces p53 expression in cancer cells in a KRas dependent manner. Oncogenic KRas has been shown to inhibit p53 function by inducing Snail to bind and eliminate... MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Biovision | GLYX13 | B2287 GLYX-13 is an N-methyl-D-aspartate receptor (NMDAR) modulator that has characteristics of a glycine site partial agonist. Displays nootropic, neuroprotective and antinociceptive activity, and... MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Biovision | GLX-351322 | B2340 GLX-351322 is a potent NADPH oxidase-4 (NOX-4) inhibitor. Displays selectivity for NOX-4 over NOX-2. GLX-351322 inhibits hydrogen peroxide production from tetracycline inducible NOX4-overexpressing... MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Biovision | Glutathione ethyl ester | B2307 Glutathione (GSH) ethyl ester is a cell-permeable derivative of GSH that undergoes hydrolysis by intracellular esterases to release GSH. Effective transport of GSH ethyl ester has been used to... MSRP: Was: Now: £410 - £904 Choose Options Compare Quick view Biovision | Glutaminase C-IN-1 (968) | B1198 Glutaminase C-IN-1 (968) a cell-permeable, reversible inhibitor of a mitochrondrial glutaminase splice variant, glutaminase C (IC₅₀ = ~2.5 µM), which is commonly found in cancer cells. Glutaminase... MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Biovision | GLPG-1690 | B1850 GLPG-1690 is a selective autotaxin inhibitor with potential application in idiopathic pulmonary disease (IPF).GLPG-1690 is a selective autotaxin inhibitor with potential application in idiopathic... MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GSK-J4 hydrochloride | 2259 MSRP: Was: Now: £364 - £806 Choose Options Compare Quick view Details Biovision | GSK-J4 (Free base) | 2762 MSRP: Was: Now: £380 - £806 Choose Options Compare Quick view Details Biovision | GSK-J1 sodium salt | 2260 MSRP: Was: Now: £364 - £806 Choose Options Compare Quick view Details Biovision | GSK-J1 (Free acid) | 2761 MSRP: Was: Now: £380 - £806 Choose Options Compare Quick view Details Biovision | GSK-961081 | B1590 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | GSK-650394 | B2093 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GSK-583 | B1301 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GSK-503 | 9538 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-484 hydrochloride | B1035 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-4112 | 9663 MSRP: Was: Now: £542 - £1,558 Choose Options Compare Quick view Details Biovision | GSK-3787 | 2400 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | GSK-3117391 | B2375 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GSK-3039294 | B2374 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | GSK-3 Inhibitor, AR-A014418 | 1953 MSRP: Was: Now: £394 - £606 Choose Options Compare Quick view Details Biovision | GSK-2982772 | B2232 MSRP: Was: Now: £478 - £1,394 Choose Options Compare Quick view Details Biovision | GSK-2879552 | B1044 MSRP: Was: Now: £772 - £2,572 Choose Options Compare Quick view Details Biovision | GSK2830371 | 2578 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | GSK-2801 | 9553 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | GSK-269962 | 9654 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | GSK-2656157 | 9466 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-2606414 | 9467 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GSK-2334470 | B1555 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GSK2330672 | B1102 MSRP: Was: Now: £640 - £1,950 Choose Options Compare Quick view Details Biovision | GSK2292767 | B1660 MSRP: Now: £372 Add to Cart Compare Quick view Details Biovision | GSK-2194069 | B1571 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | GSK2190915 | B1891 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | GSK-2126458 | 1961 MSRP: Was: Now: £494 - £1,460 Choose Options Compare Quick view Details Biovision | GSK-2118436 mesylate | 2800 MSRP: Was: Now: £444 - £1,232 Choose Options Compare Quick view Details Biovision | GSK-2110183 | B1089 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-2018682 | B1967 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GSK-199 hydrochloride | B1037 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1940029 | B2373 MSRP: Was: Now: £674 - £2,116 Choose Options Compare Quick view Details Biovision | GSK1349572 | 2288 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | GSK1325756 | B1103 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-1292263 | B1556 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GSK1278863 | B1107 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-121 trifluoroacetate | B1034 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1120212 | 1960 MSRP: Was: Now: £428 - £1,180 Choose Options Compare Quick view Details Biovision | GSK-106 hydrochloride | B1036 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1059615 | 9450 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GSK-0660 | 2897 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GS-9973 | 2669 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Grazoprevir (MK-5172) | B2337 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GPNA (monohydrate) | B2150 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | Gossypin | 2374 MSRP: Was: Now: £444 - £3,700 Choose Options Compare Quick view Details Biovision | GNE 477 | B1657 MSRP: Was: Now: £658 - £2,032 Choose Options Compare Quick view Details Biovision | GN25 | 9430 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | GLYX13 | B2287 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GLX-351322 | B2340 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Glutathione ethyl ester | B2307 MSRP: Was: Now: £410 - £904 Choose Options Compare Quick view Details Biovision | Glutaminase C-IN-1 (968) | B1198 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GLPG-1690 | B1850 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Previous 74 75 76 77 78 79 80 81 82 83 84 Next Previous 74 75 76 77 78 79 80 81 82 83 84 Next Compare Selected
Quick view Biovision | GSK-2194069 | B1571 GSK-2194069 is a potent and specific inhibitor of the β-ketoacyl reductase (KR) activity of hFAS (human Fatty Acid Synthase).GSK-2194069 is a potent and specific inhibitor of the β-ketoacyl reductase... MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Biovision | GSK2190915 | B1891 GSK2190915 (Fiboflapon) is a potent FLAP (5-lipoxygenase-activating protein) inhibitor (IC₅₀ = 2.9 nM).GSK2190915 (Fiboflapon) is a potent FLAP (5-lipoxygenase-activating protein) inhibitor (IC₅₀ = 2... MSRP: Was: Now: £478 - £1,362 Choose Options Compare
Quick view Biovision | GSK-2126458 | 1961 Cell-permeable. A highly potent, pan phosphoinositide 3-kinase (PI 3-K) family kinase inhibitor with biochemical Ki’s of 0.019 nM (PI 3-K⍺), 0.13 nM (PI 3-Kβ), 0.024 nM (PI 3-Kδ), 0.06 nM (PI 3-Kɣ),... MSRP: Was: Now: £494 - £1,460 Choose Options Compare
Quick view Biovision | GSK-2118436 mesylate | 2800 GSK2118436 is a selective BRAF V600E inhibitor. GSK2118436 binds to Raf family kinases and inhibits their activity. It is highly selective against B-Raf V600E with IC₅₀ of 0.8 nM, compared to wild... MSRP: Was: Now: £444 - £1,232 Choose Options Compare
Quick view Biovision | GSK-2110183 | B1089 GSK-2110183 is a potent, selective, and ATP-competitive pan-Akt inhibitor with IC₅₀s of 0.08, 2 and 2.6 nM for Akt1, Akt2, and Akt3 respectively.GSK-2110183 is a potent, selective, and... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GSK-2018682 | B1967 GSK-2018682 is a potent sphingosine -1 phosphate receptor (S1PR)-1 agonist; useful for the treatment of multiple sclerosis. GSK-2018682 induces acute, transient and non-symptomatic decreases in heart... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | GSK-199 hydrochloride | B1037 GSK-199 is a potent, reversible inhibitor of PAD4 (IC₅₀ = 200 nM. It binds to the low-calcium form of the enzyme and is selective for PAD4 over PAD1-3. It is less potent than the related PAD4... MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Biovision | GSK-1940029 | B2373 GSK-1940029 is a potent stearoyl-coA desaturase (SCD) inhibitorGSK-1940029 is a potent stearoyl-coA desaturase (SCD) inhibitorBiovision | B2373 | GSK-1940029 DataSheetAlternate Name/Synonyms:... MSRP: Was: Now: £674 - £2,116 Choose Options Compare
Quick view Biovision | GSK1349572 | 2288 A potent, second generation HIV integrase inhibitor (IC₅₀ = 2.7 nM) that displays potent antiviral activity.GSK1349572 is a potent, second generation HIV integrase inhibitor (IC₅₀ = 2.7 nM) that... MSRP: Was: Now: £806 - £2,704 Choose Options Compare
Quick view Biovision | GSK1325756 | B1103 GSK1325756 is a selective and reversible CXCR2 antagonist with IC₅₀ value of 12.5 nM. GSK1325756 displays anti-inflammatory effects in various preclinical and clinical models.GSK1325756 is a... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GSK-1292263 | B1556 GSK-1292263 is a novel GPR119 receptor agonist and is used for the treatment of type 2 diabetes. GSK1292263 improves glucose regulation in animal models of diabetes, but has no effect on plasma... MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Biovision | GSK1278863 | B1107 GSK-1278863 is a novel Hypoxia-Inducible Factor-Prolyl Hydroxylase Inhibitor (HIF-PHI). Hypoxia-inducible factor−prolyl hydroxylase inhibitors stimulate endogenous EPO synthesis and induce effective... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GSK-121 trifluoroacetate | B1034 GSK-121 is a novel protein arginine deiminase 4 (PAD4) inhibitor. GSK-121 was shown to inhibit the citrullination of PAD4 target proteins in a functional assay with an IC₅₀ value of 3.2 µM.GSK-121 is... MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Biovision | GSK-1120212 | 1960 A potent and selective allosteric inhibitor of the MEK1 (IC₅₀ = 0.7 nM) and MEK2 (IC₅₀ = 0.9 nM) enzymes with potential antineoplastic activity.GSK-1120212 is a potent and selective allosteric... MSRP: Was: Now: £428 - £1,180 Choose Options Compare
Quick view Biovision | GSK-106 hydrochloride | B1036 GSK-106 is a useful negative control for PAD4 inhibitors (GSK-121 and GSK-484). It does not inhibit PAD4 nor does it prevent the citrullination of PAD4 target proteins or the formation of neutrophil... MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Biovision | GSK-1059615 | 9450 GSK-1059615 is a potent, reversible, ATP-competitive inhibitor of PI3Kα (IC₅₀ = 2 nM). It inhibits proliferation in BT474 cells and attenuates MAPK signaling.GSK-1059615 is a potent, reversible,... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Biovision | GSK-0660 | 2897 GSK-0660 is a selective PPARδ antagonist (IC₅₀ values are 0.155, > 10 and ≥ 10 μM at PPARδ, PPARα and PPARγ, respectively).GSK-0660 is a selective PPARδ antagonist (IC₅₀ values are 0.155, > 10 and ≥... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Biovision | GS-9973 | 2669 GS-9973 is a potent and highly selective Syk (spleen tyrosine kinase) inhibitor (IC₅₀ = 7.7 nM).GS-9973 is a potent and highly selective Syk (spleen tyrosine kinase) inhibitor (IC₅₀ = 7.7 nM)... MSRP: Was: Now: £444 - £1,262 Choose Options Compare
Quick view Biovision | Grazoprevir (MK-5172) | B2337 Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV)... MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Biovision | GPNA (monohydrate) | B2150 GPNA is a substrate for γ-glutamyl transpeptidase. GPNA has also been shown to be an inhibitor of glutamine uptake - solute-linked carrier family A1 member 5 (SLC1A5). Cellular uptake of L-glutamine... MSRP: Was: Now: £380 - £904 Choose Options Compare
Quick view Biovision | Gossypin | 2374 A glucoside occurring in cotton and Hubiscus flowers that acts as a potent antimelanoma agent. Gossypin inhibits human melanoma cell proliferation, in vitro, in melanoma cell lines that harbors both... MSRP: Was: Now: £444 - £3,700 Choose Options Compare
Quick view Biovision | GNE 477 | B1657 GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor with IC50 of 4 nM for PI3Kα, Kiapp is 21 nM for mTOR.GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor with IC50 of 4 nM for... MSRP: Was: Now: £658 - £2,032 Choose Options Compare
Quick view Biovision | GN25 | 9430 GN25 blocks Snail binding to p53 and induces p53 expression in cancer cells in a KRas dependent manner. Oncogenic KRas has been shown to inhibit p53 function by inducing Snail to bind and eliminate... MSRP: Was: Now: £444 - £1,262 Choose Options Compare
Quick view Biovision | GLYX13 | B2287 GLYX-13 is an N-methyl-D-aspartate receptor (NMDAR) modulator that has characteristics of a glycine site partial agonist. Displays nootropic, neuroprotective and antinociceptive activity, and... MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Biovision | GLX-351322 | B2340 GLX-351322 is a potent NADPH oxidase-4 (NOX-4) inhibitor. Displays selectivity for NOX-4 over NOX-2. GLX-351322 inhibits hydrogen peroxide production from tetracycline inducible NOX4-overexpressing... MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Biovision | Glutathione ethyl ester | B2307 Glutathione (GSH) ethyl ester is a cell-permeable derivative of GSH that undergoes hydrolysis by intracellular esterases to release GSH. Effective transport of GSH ethyl ester has been used to... MSRP: Was: Now: £410 - £904 Choose Options Compare
Quick view Biovision | Glutaminase C-IN-1 (968) | B1198 Glutaminase C-IN-1 (968) a cell-permeable, reversible inhibitor of a mitochrondrial glutaminase splice variant, glutaminase C (IC₅₀ = ~2.5 µM), which is commonly found in cancer cells. Glutaminase... MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Biovision | GLPG-1690 | B1850 GLPG-1690 is a selective autotaxin inhibitor with potential application in idiopathic pulmonary disease (IPF).GLPG-1690 is a selective autotaxin inhibitor with potential application in idiopathic... MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Details Biovision | GSK-J4 hydrochloride | 2259 MSRP: Was: Now: £364 - £806 Choose Options Compare
Quick view Details Biovision | GSK-J4 (Free base) | 2762 MSRP: Was: Now: £380 - £806 Choose Options Compare
Quick view Details Biovision | GSK-J1 sodium salt | 2260 MSRP: Was: Now: £364 - £806 Choose Options Compare
Quick view Details Biovision | GSK-J1 (Free acid) | 2761 MSRP: Was: Now: £380 - £806 Choose Options Compare
Quick view Details Biovision | GSK-961081 | B1590 MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Details Biovision | GSK-650394 | B2093 MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Details Biovision | GSK-484 hydrochloride | B1035 MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Details Biovision | GSK-3117391 | B2375 MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Details Biovision | GSK-3039294 | B2374 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | GSK-3 Inhibitor, AR-A014418 | 1953 MSRP: Was: Now: £394 - £606 Choose Options Compare
Quick view Details Biovision | GSK-2982772 | B2232 MSRP: Was: Now: £478 - £1,394 Choose Options Compare
Quick view Details Biovision | GSK-2879552 | B1044 MSRP: Was: Now: £772 - £2,572 Choose Options Compare
Quick view Details Biovision | GSK2830371 | 2578 MSRP: Was: Now: £444 - £1,262 Choose Options Compare
Quick view Details Biovision | GSK-269962 | 9654 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | GSK-2656157 | 9466 MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Details Biovision | GSK-2606414 | 9467 MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Details Biovision | GSK-2334470 | B1555 MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Details Biovision | GSK2330672 | B1102 MSRP: Was: Now: £640 - £1,950 Choose Options Compare
Quick view Details Biovision | GSK2292767 | B1660 MSRP: Now: £372 Add to Cart Compare Quick view Details Biovision | GSK-2194069 | B1571 MSRP: Was: Now: £738 - £2,444 Choose Options Compare Quick view Details Biovision | GSK2190915 | B1891 MSRP: Was: Now: £478 - £1,362 Choose Options Compare Quick view Details Biovision | GSK-2126458 | 1961 MSRP: Was: Now: £494 - £1,460 Choose Options Compare Quick view Details Biovision | GSK-2118436 mesylate | 2800 MSRP: Was: Now: £444 - £1,232 Choose Options Compare Quick view Details Biovision | GSK-2110183 | B1089 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-2018682 | B1967 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GSK-199 hydrochloride | B1037 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1940029 | B2373 MSRP: Was: Now: £674 - £2,116 Choose Options Compare Quick view Details Biovision | GSK1349572 | 2288 MSRP: Was: Now: £806 - £2,704 Choose Options Compare Quick view Details Biovision | GSK1325756 | B1103 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-1292263 | B1556 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GSK1278863 | B1107 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GSK-121 trifluoroacetate | B1034 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1120212 | 1960 MSRP: Was: Now: £428 - £1,180 Choose Options Compare Quick view Details Biovision | GSK-106 hydrochloride | B1036 MSRP: Was: Now: £410 - £576 Choose Options Compare Quick view Details Biovision | GSK-1059615 | 9450 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GSK-0660 | 2897 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Quick view Details Biovision | GS-9973 | 2669 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | Grazoprevir (MK-5172) | B2337 MSRP: Was: Now: £576 - £1,788 Choose Options Compare Quick view Details Biovision | GPNA (monohydrate) | B2150 MSRP: Was: Now: £380 - £904 Choose Options Compare Quick view Details Biovision | Gossypin | 2374 MSRP: Was: Now: £444 - £3,700 Choose Options Compare Quick view Details Biovision | GNE 477 | B1657 MSRP: Was: Now: £658 - £2,032 Choose Options Compare Quick view Details Biovision | GN25 | 9430 MSRP: Was: Now: £444 - £1,262 Choose Options Compare Quick view Details Biovision | GLYX13 | B2287 MSRP: Was: Now: £708 - £2,296 Choose Options Compare Quick view Details Biovision | GLX-351322 | B2340 MSRP: Was: Now: £640 - £2,048 Choose Options Compare Quick view Details Biovision | Glutathione ethyl ester | B2307 MSRP: Was: Now: £410 - £904 Choose Options Compare Quick view Details Biovision | Glutaminase C-IN-1 (968) | B1198 MSRP: Was: Now: £606 - £1,918 Choose Options Compare Quick view Details Biovision | GLPG-1690 | B1850 MSRP: Was: Now: £542 - £1,656 Choose Options Compare Previous 74 75 76 77 78 79 80 81 82 83 84 Next Previous 74 75 76 77 78 79 80 81 82 83 84 Next Compare Selected
Quick view Details Biovision | GSK-2194069 | B1571 MSRP: Was: Now: £738 - £2,444 Choose Options Compare
Quick view Details Biovision | GSK2190915 | B1891 MSRP: Was: Now: £478 - £1,362 Choose Options Compare
Quick view Details Biovision | GSK-2126458 | 1961 MSRP: Was: Now: £494 - £1,460 Choose Options Compare
Quick view Details Biovision | GSK-2118436 mesylate | 2800 MSRP: Was: Now: £444 - £1,232 Choose Options Compare
Quick view Details Biovision | GSK-2110183 | B1089 MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Details Biovision | GSK-2018682 | B1967 MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Details Biovision | GSK-199 hydrochloride | B1037 MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Details Biovision | GSK-1940029 | B2373 MSRP: Was: Now: £674 - £2,116 Choose Options Compare
Quick view Details Biovision | GSK1349572 | 2288 MSRP: Was: Now: £806 - £2,704 Choose Options Compare
Quick view Details Biovision | GSK1325756 | B1103 MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Details Biovision | GSK-1292263 | B1556 MSRP: Was: Now: £708 - £2,296 Choose Options Compare
Quick view Details Biovision | GSK1278863 | B1107 MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Details Biovision | GSK-121 trifluoroacetate | B1034 MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Details Biovision | GSK-1120212 | 1960 MSRP: Was: Now: £428 - £1,180 Choose Options Compare
Quick view Details Biovision | GSK-106 hydrochloride | B1036 MSRP: Was: Now: £410 - £576 Choose Options Compare
Quick view Details Biovision | GSK-1059615 | 9450 MSRP: Was: Now: £542 - £1,656 Choose Options Compare
Quick view Details Biovision | Grazoprevir (MK-5172) | B2337 MSRP: Was: Now: £576 - £1,788 Choose Options Compare
Quick view Details Biovision | GPNA (monohydrate) | B2150 MSRP: Was: Now: £380 - £904 Choose Options Compare
Quick view Details Biovision | GLX-351322 | B2340 MSRP: Was: Now: £640 - £2,048 Choose Options Compare
Quick view Details Biovision | Glutathione ethyl ester | B2307 MSRP: Was: Now: £410 - £904 Choose Options Compare
Quick view Details Biovision | Glutaminase C-IN-1 (968) | B1198 MSRP: Was: Now: £606 - £1,918 Choose Options Compare
Quick view Details Biovision | GLPG-1690 | B1850 MSRP: Was: Now: £542 - £1,656 Choose Options Compare