Quick view Biovision | (−)-Huperzine A | B3095 (−)-Huperzine A is a potent and reversible inhibitor of acetylcholinesterase. It shows an IC₅₀ value of 82 nM against acetylcholinesterase in the rat cortex in vitro. It also acts as an antagonist of... MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Biovision | Galantamine Hydrobromide | B3094 Galantamine is an alkaloid originally isolated from the bulbs and flowers of various Galanthus species. It inhibits acetylcholinesterase with an IC₅₀ of 800 nM. It is a potent allosteric potentiating... MSRP: Was: Now: €546 - €1,401 Choose Options Compare
Quick view Biovision | Rivastigmine tartrate | B3093 Rivastigmine is a cholinesterase (ChE) inhibitor that inhibits butyrylcholinesterase (BChE) and acetylcholinesterase (AChE) with IC₅₀ values of 0.037 μM and 4.15 μM respectively. It is used for the... MSRP: Was: Now: €546 - €1,452 Choose Options Compare
Quick view Biovision | Donepezil Hydrochloride | B3092 Donepezil is a potent acetylcholinesterase (AChE) inhibitor with an IC₅₀ value of 5.7 nM. It produces a significant increase in acetylcholine content in rat cerebral cortex at a dose of 5 mg/kg (po)... MSRP: Was: Now: €546 - €1,401 Choose Options Compare
Quick view Biovision | Chlorprothixene hydrochloride | B3091 Chlorprothixene is a thioxanthine antipsychotic drug. It is an antagonist of dopamine and histamine receptors with Ki values of 18 nM, 2.96 nM, 4.56 nM, 9 nM and 3.75 nM for hD1, hD2, hD3, hD5 and... MSRP: Was: Now: €570 - €762 Choose Options Compare
Quick view Biovision | Pentylenetetrazole | B3090 Pentylenetetrazole is a circulatory and respiratory stimulant. It is a central nervous system modulator used to experimentally induce seizures in animals. It acts as an antagonist of GABAa receptors... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | L-(–)-Norepinephrine bitartrate hydrate | B3089 Norepinephrine is a catecholamine hormone that functions as an adrenergic neurotransmitter. It increases heart rate, blood pressure, alertness and triggers the release of glucose. The levels of... MSRP: Was: Now: €546 - €762 Choose Options Compare
Quick view Biovision | Metergoline | B3088 Metergoline is a serotonin (5-HT) receptor antagonist. It is active at 5-HT1 (pKi=7.8 for 5-HT1B), 5-HT2 (pKi=8.64, 8.75 and 8.75 for 5-HT2A, 5-HT2B and 5-HT2C respectively) and 5-HT7 (pKi=16 nM)... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | Elbasvir | B3087 Elbasvir is a potent inhibitor of Hepatitis C virus (HCV), non-structural protein 5A (NS5A). It is active against many HCV genotypes with EC₅₀ values in the picomolar range (0.0003 nM-3.4 nM). It is... MSRP: Was: Now: €666 - €1,917 Choose Options Compare
Quick view Biovision | Darunavir | B3086 Darunavir is an HIV-1 protease inhibitor with an IC₅₀ of 3 nM and cytoxicity of 74.4 μM. It is also also active against wild-type and multidrug-resistant clinical isolates of HIV-1 in... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | Amastatin hydrochloride | B3085 Amastatin is an inhibitor of aminopeptidase A and leucine aminopeptidase (IC₅₀ values of 0.54 μg/ml and 0.5 μg/ml). It does not show any significant inhibition of aminopeptidase B, trypsin,... MSRP: Was: Now: €789 - €2,409 Choose Options Compare
Quick view Biovision | Trabectedin | B3084 Trabectedin is a natural product originally isolated from the sea squirt, Ecteinascidia turbinata and is currently prepared synthetically. It interferes with transcription factors, DNA‐binding... MSRP: Was: Now: €1,944 - €5,631 Choose Options Compare
Quick view Biovision | Dexmedetomidine | B3083 Dexmedetomidine is an imidazole derivate and an active d-isomer of medetomidine. Medetomidine is a racemate of the stereoisomers levomedetomidine and dexmedetomidine. Dexmedetomidine is a potent... MSRP: Was: Now: €546 - €1,329 Choose Options Compare
Quick view Biovision | BIBR-1532 | B3082 BIBR-1532 is a highly potent mixed-type non-competitive inhibitor of telomerase. It inhibits telomerase in a dose-dependent manner, with an IC₅₀ of 93 nM. It specifically targets the telomerase... MSRP: Was: Now: €762 - €2,313 Choose Options Compare
Quick view Biovision | (-)-Equol | B3081 S-equol is a metabolite of soy isoflavonoid phytoestrogen daidzein, produced by human intestinal bacteria. S-equol has a high affinity for estrogen receptor beta (ERβ) than estrogen receptor (ERα)... MSRP: Was: Now: €615 - €1,701 Choose Options Compare
Quick view Biovision | Sodium dichloroacetate | B3080 Sodium dichloroacetate is an inhibitor of pyruvate dehydrogenase kinase (PDK). It shows IC₅₀ values of 183 μM and 80 μM for PDK2 and PDK4 respectively. DCA causes apoptosis in cancer cells and... MSRP: Was: Now: €546 - €762 Choose Options Compare
Quick view Biovision | GRL-0617 | B3079 GRL-0617 is a potent inhibitor of the papain-like protease (PLpro) from the coronavirus that causes severe acute respiratory syndrome (SARS-CoV). PLpro cleaves the viral polyproteins. GRL-0617... MSRP: Was: Now: €762 - €2,313 Choose Options Compare
Quick view Biovision | Mapracorat | B3078 Mapracorat is a selective glucocorticoid receptor agonist (SEGRA) with anti-inflammatory properties. It is in clinical trials for the topical treatment of atopic dermatitis, allergic conjunctivitis... MSRP: Was: Now: €717 - €2,115 Choose Options Compare
Quick view Biovision | Sarecycline | B3077 Sarecycline is a semi-synthetic tetracycline, narrow-spectrum antibiotic, being developed to treat patients suffering from moderate to severe acne vulgaris. Sarecycline is more active than... MSRP: Was: Now: €693 - €2,019 Choose Options Compare
Quick view Biovision | GS-441524 | B3076 GS-441524 is the predominant metabolite of remdesivir in blood and is the nucleoside of the prodrug remdesivir. It is phosphorylated to the active triphosphate metabolite which incorporates into RNA... MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Biovision | ONC-201 | B3075 ONC-201 is an orally active transcriptional inducer of Tumor necrosis factor–related apoptosis-inducing ligand (TRAIL). It induces TRAIL in a p53-independent manner at concentrations of 1.25 μM-5 μM... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | EZSolution™ LDN193189 | B3074 EZSolution™ LDN193189 is a 10.9 mM (5 mg in 1.13 ml) solution of LDN193189 (Cat. No. B3067) in anhydrous DMSO.EZSolution™ LDN193189 is a 10.9 mM (5 mg in 1.13 ml) solution of LDN193189 (Cat. No... MSRP: Now: €1,062 Add to Cart Compare Quick view Biovision | LIN28 inhibitor LI71 | B3073 LIN28 is an RNA-binding protein that regulates the maturation of the let-7 microRNAs through its two distinct cold shock and zinc-knuckle domains. LIN28 inhibitor LI71 binds the cold shock domain of... MSRP: Was: Now: €717 - €2,115 Choose Options Compare Quick view Biovision | Afatinib dimaleate | B3072 Afatinib is an irreversible dual inhibitor of epidermal growth factor receptor (EGFR) and human epidermal growth factor receptor 2 (HER2) tyrosine kinase. It shows IC₅₀ values of 0.5 nM and 14 nM for... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | (S)-Crizotinib | B3071 (S)-crizotinib is a low nanomolar inhibitor of 7,8-dihydro-8-oxoguanine triphosphatase (MTH1 or NUDT1) whereas the (R)-enantiomer shows IC₅₀ values in the micromolar range. MTH1 aids in... MSRP: Was: Now: €936 - €3,099 Choose Options Compare Quick view Biovision | Golgicide A | B3070 ADP-ribosylation factor 1 (Arf1) plays an important role in regulating secretory traffic and membrane transport within the Golgi. Arf1 is activated by guanine nucleotide exchange factors (ArfGEFs)... MSRP: Was: Now: €936 - €3,003 Choose Options Compare Quick view Biovision | CHIR-124 | B3069 CHIR-124 is a quinolone-based inhibitor of Checkpoint kinase-1 (Chk1). It potently and selectively inhibits Chk1 in vitro with an IC₅₀ of 0.3 nM. It interacts synergistically with topoisomerase... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | Riluzole | B3068 Riluzole is a benzothiazole derivative which inhibits glutamatergic neurotransmission and blocks voltage-dependent sodium channels (ED₅₀ = 2.3 μM). It reduces the uptake of GABA from neuronal synapse... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | LDN-193189 | B3067 LDN-193189 inhibits the activity of the Bone Morphogenetic Protein (BMP) type I receptors ALK2 and ALK3 with IC₅₀ values of 5 nM and 30 nM respectively and shows weaker effects on activin and the... MSRP: Was: Now: €960 - €2,682 Choose Options Compare Quick view Biovision | Quisinostat hydrochloride | B3066 Quisinostat is an inhibitor of histone deacetylase (HDAC). It shows activity toward HDAC enzymes with highest potency for recombinant HDAC1 (IC₅₀ = 0.11 nM) in vitro. The IC₅₀ values for HDAC 2 and 3... MSRP: Was: Now: €1,083 - €3,591 Choose Options Compare Quick view Biovision | GSA 10 | B3065 GSA 10 is a novel, potent activator of the smoothened receptor (Smo). GSA 10 acts at Smo and promotes the differentiation of multipotent mesenchymal progenitor cells into osteoblasts (EC₅₀ = 1.2 µM)... MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Biovision | JTE-607 | B3064 JTE-607 is a multiple cytokine inhibitor. It inhibits cytokine production specifically in human peripheral blood mononuclear cells without causing immunosuppression. It inhibits tumor necrosis... MSRP: Was: Now: €864 - €2,682 Choose Options Compare Quick view Biovision | R-7050 | B3063 R-7050 is a cell-permeable inhibitor of signaling through the TNFα receptor (TNFαR) complex. It blocks the formation of signal-initiating complexes that consist of TNFα receptor (TNFαR) I, TNFαR... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | C87 | B3062 C87 is an inhibitor of Tumor Necrosis Factor α (TNFα). It binds to human TNFα with a KD of 110 nM and potently inhibits TNFα-induced cytotoxicity in L929 cells with an IC₅₀ of 8.73 μM. It effectively... MSRP: Was: Now: €1,035 - €3,393 Choose Options Compare Quick view Biovision | BAY-678 | B3061 BAY-678 is a potent, selective, cell-permeable inhibitor of human neutrophil elastase (HNE).The activity of HNE is increased in inflammatory diseases. BAY-678 shows Ki values of 15 nM and 600 nM for... MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Biovision | BAY-677 | B3060 BAY-677 is a negative control for BAY-678. BAY-678 is a potent, selective and cell-permeable inhibitor of human neutrophil elastase (HNE) with an IC₅₀ of 20 nM. The S-enantiomer BAY-677 inhibits HNE... MSRP: Was: Now: €1,134 - €3,762 Choose Options Compare Quick view Biovision | Tucidinostat | B3059 Tucidinostat is an inhibitor of histone deacetylases (HDACs) with IC₅₀ values of 95 nM, 160 nM, 67 nM and 78 nM for HDAC1, HDAC2, HDAC3 and HDAC10 respectively. It shows potent antitumor activity. It... MSRP: Was: Now: €693 - €2,019 Choose Options Compare Quick view Biovision | Gabexate mesylate | B3058 Gabexate is an inhibitor of serine proteases. It inhibits plasma kallikrein, thrombin, plasmin, factor Xa with Ki values of 0.2 μM, 0.97 μM, 1.6 μM and 8.5 μM. It exerts an anticoagulant effect on... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | E-64d | B3057 E-64d is a synthetic analog of E-64 which is a membrane permeable inhibitor of lysosomal and cytosolic cysteine proteases. It inhibits cathepsins B and L in intact lysosomes and cells. It (20-200... MSRP: Was: Now: €909 - €2,877 Choose Options Compare Quick view Biovision | Miglustat hydrochloride | B3056 Miglustat is an inhibitor of the N-linked oligosaccharide processing enzymes α-glucosidase I and II. It inhibits rat testicular enzymes ceramide-glucosyltransferase and β-glucosidase 2 with IC50... MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Biovision | Prazosin | B3055 Prazosin is an antagonist of α1-adrenergic receptors (α1-ARs). The affinity estimates (pKi) for inhibition of [3H]-prazosin binding to CHO-K1 cells expressing cloned human α1A, α1B and α1D... MSRP: Was: Now: €546 - €1,401 Choose Options Compare Quick view Biovision | FITC-Tyramide | B3054 Tyramide signal amplification is an enzyme-catalyzed deposition of tyramide on or near a protein or nucleic acid in situ. The enzyme horseradish peroxidase (HRP) converts the labelled tyramide... MSRP: Was: Now: €1,107 - €1,701 Choose Options Compare Quick view Biovision | Siramesine | B3053 Siramesine is an agonist for sigma-2 (σ2) receptor. It is selective for σ2 over σ1 with IC₅₀ values of 0.12 nM and 17 nM respectively. It shows potent anxiolytic-like effects in rodents. The minimal... MSRP: Was: Now: €666 - €1,893 Choose Options Compare Quick view Biovision | Omeprazole | B3052 Omeprazole is a proton pump inhibitor (PPI). It inhibits gastric H+/K+ ATPase with an IC₅₀ of 1.1 μM. It shows competitive inhibition of cytochrome P450 enzyme CYP2C19 activity with a Ki of 2-6 μM... MSRP: Was: Now: €546 - €762 Choose Options Compare Quick view Biovision | RIPA-56 | B3051 RIPA-56 is a highly potent, selective, and metabolically stable inhibitor of Receptor-Interacting Protein 1 (RIP1) kinase with an IC₅₀ of 13 nM. It protects HT-29 cells against TNFα-induced... MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Biovision | Astemizole | B3050 Astemizole is a histamine H1-receptor antagonist, with an IC₅₀ of 4 nM. Astemizole also shows potent hERG potassium channel blocking activity with an IC₅₀ of 0.9 nM. Astemizole shows synergistic... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | PRE-084 Hydrochloride | B3049 PRE-084 is a high affinity sigma receptor 1 (σ1) agonist. It shows Ki values of 2.2 and 13,091 nM for σ1 and σ2 receptors, respectively and an IC₅₀ of 44 nM in the sigma receptor assay. It does not... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | S1RA (E-52862) | B3048 S1RA is a highly selective sigma-1 (σ1) receptor antagonist. It shows high affinity for σ1 receptors with Ki values of 17 nM and 23.5 nM for human and guinea pig σ1 receptors respectively but no... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | NE-100 hydrochloride | B3047 NE-100 is a potent antagonist of sigma-1 (σ1) receptor. It inhibits binding of (+)-pentazocine binding to sigma-1 binding sites with an IC₅₀ value of 1.54 nM. NE-100 attenuates phencyclidin induced... MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Biovision | SA4503 dihydrochloride | B3046 SA4503 is a potent sigma-1 (σ1 receptor) agonist. It shows 100 fold higher affinity for σ1 than σ2 receptor with IC₅₀ values of 17.4 nM and 1784 nM against 200 nM (+)-pentazocine for binding σ... MSRP: Was: Now: €813 - €2,484 Choose Options Compare Quick view Biovision | Pridopidine | B3045 Pridopidine is a phenylpiperidine dopaminergic stabilizer. It is a low affinity dopamine D2 receptor antagonist and a potent sigma-1 receptor (S1R) agonist. The affinity of pridopidine for S1R is... MSRP: Was: Now: €546 - €1,209 Choose Options Compare Quick view Biovision | Ditolylguanidine | B3044 Ditolylguanidine is a sigma receptor (σR) agonist with neuroprotective activity. It shows Kd values of 21.9 nM and 57.4 nM for σ2 and σ1 receptor respectively. Combined treatment with... MSRP: Was: Now: €546 - €1,209 Choose Options Compare Quick view Details Biovision | (−)-Huperzine A | B3095 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | Galantamine Hydrobromide | B3094 MSRP: Was: Now: €546 - €1,401 Choose Options Compare Quick view Details Biovision | Rivastigmine tartrate | B3093 MSRP: Was: Now: €546 - €1,452 Choose Options Compare Quick view Details Biovision | Donepezil Hydrochloride | B3092 MSRP: Was: Now: €546 - €1,401 Choose Options Compare Quick view Details Biovision | Chlorprothixene hydrochloride | B3091 MSRP: Was: Now: €570 - €762 Choose Options Compare Quick view Details Biovision | Pentylenetetrazole | B3090 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | L-(–)-Norepinephrine bitartrate hydrate | B3089 MSRP: Was: Now: €546 - €762 Choose Options Compare Quick view Details Biovision | Metergoline | B3088 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | Elbasvir | B3087 MSRP: Was: Now: €666 - €1,917 Choose Options Compare Quick view Details Biovision | Darunavir | B3086 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | Amastatin hydrochloride | B3085 MSRP: Was: Now: €789 - €2,409 Choose Options Compare Quick view Details Biovision | Trabectedin | B3084 MSRP: Was: Now: €1,944 - €5,631 Choose Options Compare Quick view Details Biovision | Dexmedetomidine | B3083 MSRP: Was: Now: €546 - €1,329 Choose Options Compare Quick view Details Biovision | BIBR-1532 | B3082 MSRP: Was: Now: €762 - €2,313 Choose Options Compare Quick view Details Biovision | (-)-Equol | B3081 MSRP: Was: Now: €615 - €1,701 Choose Options Compare Quick view Details Biovision | Sodium dichloroacetate | B3080 MSRP: Was: Now: €546 - €762 Choose Options Compare Quick view Details Biovision | GRL-0617 | B3079 MSRP: Was: Now: €762 - €2,313 Choose Options Compare Quick view Details Biovision | Mapracorat | B3078 MSRP: Was: Now: €717 - €2,115 Choose Options Compare Quick view Details Biovision | Sarecycline | B3077 MSRP: Was: Now: €693 - €2,019 Choose Options Compare Quick view Details Biovision | GS-441524 | B3076 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | ONC-201 | B3075 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | EZSolution™ LDN193189 | B3074 MSRP: Now: €1,062 Add to Cart Compare Quick view Details Biovision | LIN28 inhibitor LI71 | B3073 MSRP: Was: Now: €717 - €2,115 Choose Options Compare Quick view Details Biovision | Afatinib dimaleate | B3072 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | (S)-Crizotinib | B3071 MSRP: Was: Now: €936 - €3,099 Choose Options Compare Quick view Details Biovision | Golgicide A | B3070 MSRP: Was: Now: €936 - €3,003 Choose Options Compare Quick view Details Biovision | CHIR-124 | B3069 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | Riluzole | B3068 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | LDN-193189 | B3067 MSRP: Was: Now: €960 - €2,682 Choose Options Compare Quick view Details Biovision | Quisinostat hydrochloride | B3066 MSRP: Was: Now: €1,083 - €3,591 Choose Options Compare Quick view Details Biovision | GSA 10 | B3065 MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Details Biovision | JTE-607 | B3064 MSRP: Was: Now: €864 - €2,682 Choose Options Compare Quick view Details Biovision | R-7050 | B3063 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | C87 | B3062 MSRP: Was: Now: €1,035 - €3,393 Choose Options Compare Quick view Details Biovision | BAY-678 | B3061 MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Details Biovision | BAY-677 | B3060 MSRP: Was: Now: €1,134 - €3,762 Choose Options Compare Quick view Details Biovision | Tucidinostat | B3059 MSRP: Was: Now: €693 - €2,019 Choose Options Compare Quick view Details Biovision | Gabexate mesylate | B3058 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | E-64d | B3057 MSRP: Was: Now: €909 - €2,877 Choose Options Compare Quick view Details Biovision | Miglustat hydrochloride | B3056 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | Prazosin | B3055 MSRP: Was: Now: €546 - €1,401 Choose Options Compare Quick view Details Biovision | FITC-Tyramide | B3054 MSRP: Was: Now: €1,107 - €1,701 Choose Options Compare Quick view Details Biovision | Siramesine | B3053 MSRP: Was: Now: €666 - €1,893 Choose Options Compare Quick view Details Biovision | Omeprazole | B3052 MSRP: Was: Now: €546 - €762 Choose Options Compare Quick view Details Biovision | RIPA-56 | B3051 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | Astemizole | B3050 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | PRE-084 Hydrochloride | B3049 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | S1RA (E-52862) | B3048 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | NE-100 hydrochloride | B3047 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | SA4503 dihydrochloride | B3046 MSRP: Was: Now: €813 - €2,484 Choose Options Compare Quick view Details Biovision | Pridopidine | B3045 MSRP: Was: Now: €546 - €1,209 Choose Options Compare Quick view Details Biovision | Ditolylguanidine | B3044 MSRP: Was: Now: €546 - €1,209 Choose Options Compare Previous 3 4 5 6 7 8 9 10 11 12 13 Next Previous 3 4 5 6 7 8 9 10 11 12 13 Next Compare Selected
Quick view Biovision | LIN28 inhibitor LI71 | B3073 LIN28 is an RNA-binding protein that regulates the maturation of the let-7 microRNAs through its two distinct cold shock and zinc-knuckle domains. LIN28 inhibitor LI71 binds the cold shock domain of... MSRP: Was: Now: €717 - €2,115 Choose Options Compare
Quick view Biovision | Afatinib dimaleate | B3072 Afatinib is an irreversible dual inhibitor of epidermal growth factor receptor (EGFR) and human epidermal growth factor receptor 2 (HER2) tyrosine kinase. It shows IC₅₀ values of 0.5 nM and 14 nM for... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | (S)-Crizotinib | B3071 (S)-crizotinib is a low nanomolar inhibitor of 7,8-dihydro-8-oxoguanine triphosphatase (MTH1 or NUDT1) whereas the (R)-enantiomer shows IC₅₀ values in the micromolar range. MTH1 aids in... MSRP: Was: Now: €936 - €3,099 Choose Options Compare
Quick view Biovision | Golgicide A | B3070 ADP-ribosylation factor 1 (Arf1) plays an important role in regulating secretory traffic and membrane transport within the Golgi. Arf1 is activated by guanine nucleotide exchange factors (ArfGEFs)... MSRP: Was: Now: €936 - €3,003 Choose Options Compare
Quick view Biovision | CHIR-124 | B3069 CHIR-124 is a quinolone-based inhibitor of Checkpoint kinase-1 (Chk1). It potently and selectively inhibits Chk1 in vitro with an IC₅₀ of 0.3 nM. It interacts synergistically with topoisomerase... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | Riluzole | B3068 Riluzole is a benzothiazole derivative which inhibits glutamatergic neurotransmission and blocks voltage-dependent sodium channels (ED₅₀ = 2.3 μM). It reduces the uptake of GABA from neuronal synapse... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | LDN-193189 | B3067 LDN-193189 inhibits the activity of the Bone Morphogenetic Protein (BMP) type I receptors ALK2 and ALK3 with IC₅₀ values of 5 nM and 30 nM respectively and shows weaker effects on activin and the... MSRP: Was: Now: €960 - €2,682 Choose Options Compare
Quick view Biovision | Quisinostat hydrochloride | B3066 Quisinostat is an inhibitor of histone deacetylase (HDAC). It shows activity toward HDAC enzymes with highest potency for recombinant HDAC1 (IC₅₀ = 0.11 nM) in vitro. The IC₅₀ values for HDAC 2 and 3... MSRP: Was: Now: €1,083 - €3,591 Choose Options Compare
Quick view Biovision | GSA 10 | B3065 GSA 10 is a novel, potent activator of the smoothened receptor (Smo). GSA 10 acts at Smo and promotes the differentiation of multipotent mesenchymal progenitor cells into osteoblasts (EC₅₀ = 1.2 µM)... MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare
Quick view Biovision | JTE-607 | B3064 JTE-607 is a multiple cytokine inhibitor. It inhibits cytokine production specifically in human peripheral blood mononuclear cells without causing immunosuppression. It inhibits tumor necrosis... MSRP: Was: Now: €864 - €2,682 Choose Options Compare
Quick view Biovision | R-7050 | B3063 R-7050 is a cell-permeable inhibitor of signaling through the TNFα receptor (TNFαR) complex. It blocks the formation of signal-initiating complexes that consist of TNFα receptor (TNFαR) I, TNFαR... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | C87 | B3062 C87 is an inhibitor of Tumor Necrosis Factor α (TNFα). It binds to human TNFα with a KD of 110 nM and potently inhibits TNFα-induced cytotoxicity in L929 cells with an IC₅₀ of 8.73 μM. It effectively... MSRP: Was: Now: €1,035 - €3,393 Choose Options Compare
Quick view Biovision | BAY-678 | B3061 BAY-678 is a potent, selective, cell-permeable inhibitor of human neutrophil elastase (HNE).The activity of HNE is increased in inflammatory diseases. BAY-678 shows Ki values of 15 nM and 600 nM for... MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare
Quick view Biovision | BAY-677 | B3060 BAY-677 is a negative control for BAY-678. BAY-678 is a potent, selective and cell-permeable inhibitor of human neutrophil elastase (HNE) with an IC₅₀ of 20 nM. The S-enantiomer BAY-677 inhibits HNE... MSRP: Was: Now: €1,134 - €3,762 Choose Options Compare
Quick view Biovision | Tucidinostat | B3059 Tucidinostat is an inhibitor of histone deacetylases (HDACs) with IC₅₀ values of 95 nM, 160 nM, 67 nM and 78 nM for HDAC1, HDAC2, HDAC3 and HDAC10 respectively. It shows potent antitumor activity. It... MSRP: Was: Now: €693 - €2,019 Choose Options Compare
Quick view Biovision | Gabexate mesylate | B3058 Gabexate is an inhibitor of serine proteases. It inhibits plasma kallikrein, thrombin, plasmin, factor Xa with Ki values of 0.2 μM, 0.97 μM, 1.6 μM and 8.5 μM. It exerts an anticoagulant effect on... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | E-64d | B3057 E-64d is a synthetic analog of E-64 which is a membrane permeable inhibitor of lysosomal and cytosolic cysteine proteases. It inhibits cathepsins B and L in intact lysosomes and cells. It (20-200... MSRP: Was: Now: €909 - €2,877 Choose Options Compare
Quick view Biovision | Miglustat hydrochloride | B3056 Miglustat is an inhibitor of the N-linked oligosaccharide processing enzymes α-glucosidase I and II. It inhibits rat testicular enzymes ceramide-glucosyltransferase and β-glucosidase 2 with IC50... MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Biovision | Prazosin | B3055 Prazosin is an antagonist of α1-adrenergic receptors (α1-ARs). The affinity estimates (pKi) for inhibition of [3H]-prazosin binding to CHO-K1 cells expressing cloned human α1A, α1B and α1D... MSRP: Was: Now: €546 - €1,401 Choose Options Compare
Quick view Biovision | FITC-Tyramide | B3054 Tyramide signal amplification is an enzyme-catalyzed deposition of tyramide on or near a protein or nucleic acid in situ. The enzyme horseradish peroxidase (HRP) converts the labelled tyramide... MSRP: Was: Now: €1,107 - €1,701 Choose Options Compare
Quick view Biovision | Siramesine | B3053 Siramesine is an agonist for sigma-2 (σ2) receptor. It is selective for σ2 over σ1 with IC₅₀ values of 0.12 nM and 17 nM respectively. It shows potent anxiolytic-like effects in rodents. The minimal... MSRP: Was: Now: €666 - €1,893 Choose Options Compare
Quick view Biovision | Omeprazole | B3052 Omeprazole is a proton pump inhibitor (PPI). It inhibits gastric H+/K+ ATPase with an IC₅₀ of 1.1 μM. It shows competitive inhibition of cytochrome P450 enzyme CYP2C19 activity with a Ki of 2-6 μM... MSRP: Was: Now: €546 - €762 Choose Options Compare
Quick view Biovision | RIPA-56 | B3051 RIPA-56 is a highly potent, selective, and metabolically stable inhibitor of Receptor-Interacting Protein 1 (RIP1) kinase with an IC₅₀ of 13 nM. It protects HT-29 cells against TNFα-induced... MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Biovision | Astemizole | B3050 Astemizole is a histamine H1-receptor antagonist, with an IC₅₀ of 4 nM. Astemizole also shows potent hERG potassium channel blocking activity with an IC₅₀ of 0.9 nM. Astemizole shows synergistic... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | PRE-084 Hydrochloride | B3049 PRE-084 is a high affinity sigma receptor 1 (σ1) agonist. It shows Ki values of 2.2 and 13,091 nM for σ1 and σ2 receptors, respectively and an IC₅₀ of 44 nM in the sigma receptor assay. It does not... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | S1RA (E-52862) | B3048 S1RA is a highly selective sigma-1 (σ1) receptor antagonist. It shows high affinity for σ1 receptors with Ki values of 17 nM and 23.5 nM for human and guinea pig σ1 receptors respectively but no... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | NE-100 hydrochloride | B3047 NE-100 is a potent antagonist of sigma-1 (σ1) receptor. It inhibits binding of (+)-pentazocine binding to sigma-1 binding sites with an IC₅₀ value of 1.54 nM. NE-100 attenuates phencyclidin induced... MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Biovision | SA4503 dihydrochloride | B3046 SA4503 is a potent sigma-1 (σ1 receptor) agonist. It shows 100 fold higher affinity for σ1 than σ2 receptor with IC₅₀ values of 17.4 nM and 1784 nM against 200 nM (+)-pentazocine for binding σ... MSRP: Was: Now: €813 - €2,484 Choose Options Compare
Quick view Biovision | Pridopidine | B3045 Pridopidine is a phenylpiperidine dopaminergic stabilizer. It is a low affinity dopamine D2 receptor antagonist and a potent sigma-1 receptor (S1R) agonist. The affinity of pridopidine for S1R is... MSRP: Was: Now: €546 - €1,209 Choose Options Compare
Quick view Biovision | Ditolylguanidine | B3044 Ditolylguanidine is a sigma receptor (σR) agonist with neuroprotective activity. It shows Kd values of 21.9 nM and 57.4 nM for σ2 and σ1 receptor respectively. Combined treatment with... MSRP: Was: Now: €546 - €1,209 Choose Options Compare
Quick view Details Biovision | (−)-Huperzine A | B3095 MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Details Biovision | Galantamine Hydrobromide | B3094 MSRP: Was: Now: €546 - €1,401 Choose Options Compare
Quick view Details Biovision | Rivastigmine tartrate | B3093 MSRP: Was: Now: €546 - €1,452 Choose Options Compare
Quick view Details Biovision | Donepezil Hydrochloride | B3092 MSRP: Was: Now: €546 - €1,401 Choose Options Compare
Quick view Details Biovision | Chlorprothixene hydrochloride | B3091 MSRP: Was: Now: €570 - €762 Choose Options Compare
Quick view Details Biovision | Pentylenetetrazole | B3090 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | L-(–)-Norepinephrine bitartrate hydrate | B3089 MSRP: Was: Now: €546 - €762 Choose Options Compare
Quick view Details Biovision | Metergoline | B3088 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | Darunavir | B3086 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | Amastatin hydrochloride | B3085 MSRP: Was: Now: €789 - €2,409 Choose Options Compare
Quick view Details Biovision | Trabectedin | B3084 MSRP: Was: Now: €1,944 - €5,631 Choose Options Compare
Quick view Details Biovision | Dexmedetomidine | B3083 MSRP: Was: Now: €546 - €1,329 Choose Options Compare
Quick view Details Biovision | BIBR-1532 | B3082 MSRP: Was: Now: €762 - €2,313 Choose Options Compare
Quick view Details Biovision | (-)-Equol | B3081 MSRP: Was: Now: €615 - €1,701 Choose Options Compare
Quick view Details Biovision | Sodium dichloroacetate | B3080 MSRP: Was: Now: €546 - €762 Choose Options Compare
Quick view Details Biovision | Mapracorat | B3078 MSRP: Was: Now: €717 - €2,115 Choose Options Compare
Quick view Details Biovision | Sarecycline | B3077 MSRP: Was: Now: €693 - €2,019 Choose Options Compare
Quick view Details Biovision | GS-441524 | B3076 MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Details Biovision | EZSolution™ LDN193189 | B3074 MSRP: Now: €1,062 Add to Cart Compare Quick view Details Biovision | LIN28 inhibitor LI71 | B3073 MSRP: Was: Now: €717 - €2,115 Choose Options Compare Quick view Details Biovision | Afatinib dimaleate | B3072 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | (S)-Crizotinib | B3071 MSRP: Was: Now: €936 - €3,099 Choose Options Compare Quick view Details Biovision | Golgicide A | B3070 MSRP: Was: Now: €936 - €3,003 Choose Options Compare Quick view Details Biovision | CHIR-124 | B3069 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | Riluzole | B3068 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | LDN-193189 | B3067 MSRP: Was: Now: €960 - €2,682 Choose Options Compare Quick view Details Biovision | Quisinostat hydrochloride | B3066 MSRP: Was: Now: €1,083 - €3,591 Choose Options Compare Quick view Details Biovision | GSA 10 | B3065 MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Details Biovision | JTE-607 | B3064 MSRP: Was: Now: €864 - €2,682 Choose Options Compare Quick view Details Biovision | R-7050 | B3063 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | C87 | B3062 MSRP: Was: Now: €1,035 - €3,393 Choose Options Compare Quick view Details Biovision | BAY-678 | B3061 MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare Quick view Details Biovision | BAY-677 | B3060 MSRP: Was: Now: €1,134 - €3,762 Choose Options Compare Quick view Details Biovision | Tucidinostat | B3059 MSRP: Was: Now: €693 - €2,019 Choose Options Compare Quick view Details Biovision | Gabexate mesylate | B3058 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | E-64d | B3057 MSRP: Was: Now: €909 - €2,877 Choose Options Compare Quick view Details Biovision | Miglustat hydrochloride | B3056 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | Prazosin | B3055 MSRP: Was: Now: €546 - €1,401 Choose Options Compare Quick view Details Biovision | FITC-Tyramide | B3054 MSRP: Was: Now: €1,107 - €1,701 Choose Options Compare Quick view Details Biovision | Siramesine | B3053 MSRP: Was: Now: €666 - €1,893 Choose Options Compare Quick view Details Biovision | Omeprazole | B3052 MSRP: Was: Now: €546 - €762 Choose Options Compare Quick view Details Biovision | RIPA-56 | B3051 MSRP: Was: Now: €570 - €1,527 Choose Options Compare Quick view Details Biovision | Astemizole | B3050 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | PRE-084 Hydrochloride | B3049 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | S1RA (E-52862) | B3048 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | NE-100 hydrochloride | B3047 MSRP: Was: Now: €546 - €1,428 Choose Options Compare Quick view Details Biovision | SA4503 dihydrochloride | B3046 MSRP: Was: Now: €813 - €2,484 Choose Options Compare Quick view Details Biovision | Pridopidine | B3045 MSRP: Was: Now: €546 - €1,209 Choose Options Compare Quick view Details Biovision | Ditolylguanidine | B3044 MSRP: Was: Now: €546 - €1,209 Choose Options Compare Previous 3 4 5 6 7 8 9 10 11 12 13 Next Previous 3 4 5 6 7 8 9 10 11 12 13 Next Compare Selected
Quick view Details Biovision | LIN28 inhibitor LI71 | B3073 MSRP: Was: Now: €717 - €2,115 Choose Options Compare
Quick view Details Biovision | Afatinib dimaleate | B3072 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | (S)-Crizotinib | B3071 MSRP: Was: Now: €936 - €3,099 Choose Options Compare
Quick view Details Biovision | Golgicide A | B3070 MSRP: Was: Now: €936 - €3,003 Choose Options Compare
Quick view Details Biovision | LDN-193189 | B3067 MSRP: Was: Now: €960 - €2,682 Choose Options Compare
Quick view Details Biovision | Quisinostat hydrochloride | B3066 MSRP: Was: Now: €1,083 - €3,591 Choose Options Compare
Quick view Details Biovision | BAY-678 | B3061 MSRP: Was: Now: €1,107 - €3,666 Choose Options Compare
Quick view Details Biovision | BAY-677 | B3060 MSRP: Was: Now: €1,134 - €3,762 Choose Options Compare
Quick view Details Biovision | Tucidinostat | B3059 MSRP: Was: Now: €693 - €2,019 Choose Options Compare
Quick view Details Biovision | Gabexate mesylate | B3058 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | Miglustat hydrochloride | B3056 MSRP: Was: Now: €570 - €1,527 Choose Options Compare
Quick view Details Biovision | FITC-Tyramide | B3054 MSRP: Was: Now: €1,107 - €1,701 Choose Options Compare
Quick view Details Biovision | Siramesine | B3053 MSRP: Was: Now: €666 - €1,893 Choose Options Compare
Quick view Details Biovision | Astemizole | B3050 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | PRE-084 Hydrochloride | B3049 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | S1RA (E-52862) | B3048 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | NE-100 hydrochloride | B3047 MSRP: Was: Now: €546 - €1,428 Choose Options Compare
Quick view Details Biovision | SA4503 dihydrochloride | B3046 MSRP: Was: Now: €813 - €2,484 Choose Options Compare
Quick view Details Biovision | Pridopidine | B3045 MSRP: Was: Now: €546 - €1,209 Choose Options Compare
Quick view Details Biovision | Ditolylguanidine | B3044 MSRP: Was: Now: €546 - €1,209 Choose Options Compare