Product Description
Cell-permeable. A potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor. Inhibits FAAH in a time-dependent manner by covalently modifying the enzyme's active site serine (IC₅₀ = 33 nM). It is highly selective for FAAH relative to other mammalian serine hydrolases.
FAAH Inhibitor, PF-622 is a potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor. Inhibits FAAH in a time-dependent manner by covalently modifying the enzyme's active site serine (IC₅₀ = 33 nM). It is highly selective for FAAH relative to other mammalian serine hydrolases.
Biovision | 1928 | FAAH Inhibitor, PF-622 DataSheet
Alternate Name/Synonyms: N-Phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carboxamide
Appearance: White soild
Formulation: N/A
CAS Number: 898235-65-9
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₂₁H₂₂N₄O
Molecular Weight: 346.43
Cell-Permeable?: Yes
Purity: ≥98% by TLC
Solubilities: DMSO (~25 mg/ml) or Ethanol (~ 3 mg/ml)
Handling: Protect from light and air
Country of Origin: USA
Tag Line: A potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor
MDL Number: N/A
PubChem CID: 11515763
SMILES: C1CN(CCN1CC2=NC3=CC=CC=C3C=C2)C(=O)NC4=CC=CC=C4
InChi: InChI=1S/C21H22N4O/c26-21(23-18-7-2-1-3-8-18)25-14-12-24(13-15-25)16-19-11-10-17-6-4-5-9-20(17)22-19/h1-11H,12-16H2,(H,23,26)
InChi Key: SNTCRRMCALVGNL-UHFFFAOYSA-N