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Product Description
LY-2795050 is a potent and selective κ-opioid Receptor (KOR) antagonist (IC₅₀ = 0.72 nM). Has the potential as a PET tracer to image KOR in vivo.
LY-2795050 is a potent and selective κ-opioid Receptor (KOR) antagonist (IC₅₀ = 0.72 nM). Has the potential as a PET tracer to image KOR in vivo.
Biovision | B2351 | LY-2795050 DataSheet
Alternate Name/Synonyms: LY279050,(S)-3-chloro-4-(4-((2-(pyridin-3-yl)pyrrolidin-1-yl)methyl)phenoxy)benzamide
Appearance: Crystalline solid
Formulation:
CAS Number: 1346133-08-1
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: N/A
Molecular Formula: C₂₃H₂₂ClN₃O₂
Molecular Weight: 407.9
Cell-Permeable?: TRUE
Purity: ≥98% by HPLC
Solubilities: >50 mg/ml (DMSO) in 0
Handling: Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
Country of Origin: USA
Tag Line: A selective κ-opioid Receptor (KOR) antagonist
MDL Number:
PubChem CID: 56851583
SMILES: C1CC(N(C1)CC2=CC=C(C=C2)OC3=C(C=C(C=C3)C(=O)N)Cl)C4=CN=CC=C4
InChi: LOOCZNLSXJHWTG-NRFANRHFSA-N
InChi Key: InChI=1S/C23H22ClN3O2/c24-20-13-17(23(25)28)7-10-22(20)29-19-8-5-16(6-9-19)15-27-12-2-4-21(27)18-3-1-11-26-14-18/h1,3,5-11,13-14,21H,2,4,12,15H2,(H2,25,28)/t21-/m0/s1
