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Product Description
TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2. Displays low-nanomolar antagonist activity against only EP2, >300-fold selectivity over human EP3, EP4, and IP receptors, 100-fold selectivity over EP1 receptors.
TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2. Displays low-nanomolar antagonist activity against only EP2, >300-fold selectivity over human EP3, EP4, and IP receptors, 100-fold selectivity over EP1 receptors.
Biovision | 9646 | TG6-10-1 DataSheet
Alternate Name/Synonyms: (E)-N-(2-(2-(trifluoromethyl)-1H-indol-1-yl)ethyl)-3-(3,4,5-trimethoxyphenyl)acrylamide
Appearance: Crystalline solid
Formulation: N/A
CAS Number: 1415716-58-3
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₂₃H₂₃F₃N₂O₄
Molecular Weight: 448.43
Cell-Permeable?: Yes
Purity: ≥98% by HPLC
Solubilities: DMSO (>5 mg/ml)
Handling: Protect from air and light
Country of Origin: USA
Tag Line: A potent and selective antagonist for the prostaglandin E2 receptor subtype EP2
MDL Number: N/A
PubChem CID: 71499384
SMILES: COC1=CC(=CC(=C1OC)OC)C=CC(=O)NCCN2C3=CC=CC=C3C=C2C(F)(F)F
InChi: InChI=1S/C23H23F3N2O4/c1-30-18-12-15(13-19(31-2)22(18)32-3)8-9-21(29)27-10-11-28-17-7-5-4-6-16(17)14-20(28)23(24,25)26/h4-9,12-14H,10-11H2,1-3H3,(H,27,29)/b9-8+
InChi Key: WUYOECAJFJFUFC-CMDGGOBGSA-N
