Product Description
Cell-permeable. A potent, slow binding dipeptidyl peptidase IV inhibitor with IC₅₀ values of 3, 5, 8, and 8 nM for rat, canine, human and monkey enzymes respectively. Acts as a long-acting hypoglycemic agent.
DPP IV Inhibitor, K 579 is a potent, slow binding dipeptidyl peptidase IV inhibitor with IC₅₀ values of 3, 5, 8, and 8 nM for rat, canine, human and monkey enzymes respectively. Acts as a long-acting hypoglycemic agent.
Biovision | 1963 | DPP IV Inhibitor, K 579 DataSheet
Alternate Name/Synonyms: (2S)-1-[[[4-Methyl-1-(2-pyrimidinyl)-4-piperidinyl]amino]acetyl]-2-pyrrolidinecarbonitrile
Appearance: Light brown solid
Formulation: N/A
CAS Number: 440100-64-1
Structure Available?: Yes
Peptide sequence: N/A
Salt Form: No
Molecular Formula: C₁₇H₂₄N₆O
Molecular Weight: 328.41
Cell-Permeable?: Yes
Purity: ≥98% by HPLC
Solubilities: DMSO (~100 mM) or EtOH (~ 20 mM) or 1 eq. HCl (50 mM)
Handling: Protect from light and air
Country of Origin: USA
Tag Line: A potent DPP IV Inhibitor,
MDL Number: MFCD07364044
PubChem CID: 9818824
SMILES: CC1(CCN(CC1)C2=NC=CC=N2)NCC(=O)N3CCCC3C#N
InChi: InChI=1S/C17H24N6O/c1-17(21-13-15(24)23-9-2-4-14(23)12-18)5-10-22(11-6-17)16-19-7-3-8-20-16/h3,7-8,14,21H,2,4-6,9-11,13H2,1H3/t14-/m0/s1
InChi Key: JERPHRNGJBSFAP-AWEZNQCLSA-N