Quick view Biovision | QS11 | 1680 Inhibits the GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) as well as synergizes the Wnt/β-catenin signaling pathway. The Wnt/β-catenin signaling pathway regulates cell fate and... MSRP: Now: NULL386.00 Add to Cart Compare Quick view Biovision | ML141 | 2267 Cell-permeable. A potent, selective, reversible and non-competitive inhibitor of Cdc42 GTPase (IC₅₀ = 2.6 and 5.4 μM for Cdc42 wild type and activated mutant, respectively). No appreciable inhibitory... MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare Quick view Biovision | genz-123346 | B2286 Genz-123346 is a potent and selective glucosylceramide synthase inhibitor with potential anticancer activity. Does not affect the activities of other related glycosidase, such as 1-O-acylceramide... MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare Quick view Biovision | Tautomycin | B1237 Tautomycin is a potent protein phosphatase inhibitor that inhibits PP1 completely at 3 nM and PP2 at 30 nM. Acts as a weak inhibitor of PP2B and does not inhibit PP2C. Its cell permeability and... MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Biovision | Liproxstatin-1 | B2312 A potent inhibitor of ferroptosis. Liproxstatin-1 suppresses ferroptosis in human cells and in an ischemia/reperfusion-induced tissue injury model in mice. Knockout of glutathione peroxidase 4 (Gpx4)... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Biovision | ITD-1 | 2879 ITD-1 is a potent and highly selective TGFβ pathway inhibitor (IC₅₀ = 0.85 µM). ITD-1 promotes cardiomyocyte differentiation specifically via degradation of the TGFβ type II receptor (TGFBR2),... MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Biovision | 10058-F4 | 2739 10058-F4 is a c-Myc inhibitor that inhibits the c-Myc-Max associationn and function. It prevents the growth of fibroblasts in a c-Myc-dependent manner. Downregulates human telomerase reverse... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Biovision | CH-223191 | 2723 CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist. It blocks activation by 2,3,7,8-Tetrachlorodibenzo-p-dioxin (TCDD) (IC₅₀ = 0.03 µM). It also blocks TCDD-mediated... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Biovision | BPTES | B2165 BPTES is an allosteric glutaminase (GLS1) inhibitor (IC₅₀ = 3.3 μM). Displays selectivity for GLS1 over GLS2 and γ-glutamyl transpeptidase. Induces cell death of P493 human lymphoma B cells in vitro... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Biovision | Entrectinib | B1324 Entrectinib is an inhibitor of TrkA (IC₅₀ = 1.7 nM), TrkB (IC₅₀ = 0.1 nM), and TrkC (IC₅₀ = 0.1 nM), as well as C-ros oncogene 1 (ROS1; IC₅₀ = 0.2 nM) and anaplastic lymphoma kinase (ALK; IC₅₀ = 1.6... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | MPI-0479605 | 9589 MPI-0479605 is a potent, selective, ATP-competitive small-molecule inhibitor of the Mitotic kinase Mps1 (IC₅₀ = 1.8 nM).MPI-0479605 is a potent, selective, ATP-competitive small-molecule inhibitor of... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | Acalisib | B1666 Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12.7 nM.Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12.7 nM.Biovision | B1666... MSRP: Was: Now: NULL247.00 - NULL739.00 Choose Options Compare Quick view Biovision | URMC-099 | 9443 URMC-099 is a brain-permeable, mixed lineage kinase (MLK) inhibitor with IC₅₀ values of 19 nM, 42 nM, 14 nM, and 150 nM, for MLK1, MLK2, MLK3, and DLK, respectively. In vitro, URMC-099 treatment... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Biovision | A-366 | 2859 A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC₅₀ = 3.3 nM). It displays >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. A-366 has been... MSRP: Was: Now: NULL254.00 - NULL714.00 Choose Options Compare Quick view Biovision | Velpatasvir | B1194 Velpatasvir (formerly GS-5816) is a novel NS5A inhibitor that has potent in vitro anti-HCV activity across all genotypes at the picomolar level.Velpatasvir (formerly GS-5816) is a novel NS5A... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Biovision | RO-3306 | 2039 Cell-permeable. A selective CDK 1 inhibitor (Cdk1/B1 and Cdk1/A). Arrests cell cycle at G1, S, and G2/M and induces apoptosis in embryonic stem cells. Actively enhances downstream p53 signaling to... MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Biovision | Pyridoclax | B1817 Pyridoclax(MR-29072) is a potent Mcl-1 inhibitor (Kd = 25 nM). Pyridoclax is able to disrupt BimL/Mcl-1 interaction in whole living cells.Pyridoclax(MR-29072) is a potent Mcl-1 inhibitor (Kd = 25 nM)... MSRP: Was: Now: NULL303.00 - NULL967.00 Choose Options Compare Quick view Biovision | Bikinin | 2034 Cell-permeable. A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase that activates brassinosteroid (BR) signaling downstream of the BR receptor. Bikinin directly binds the GSK3 BIN2... MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Biovision | OF-1 | 9592 OF-1 is a selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500 nM respectively). OF-1 displays 39-fold selectivity for BRPF1B and BRPF2 over BRD4. It increases thermal... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Biovision | LY3023414 | B1759 LY3023414 is a small molecule that has been shown in vitro to be a selective ATP-competitive inhibitor of PI3Kα and mTOR, DNA-PK, and other class I PI3K family members.LY3023414 is a small molecule... MSRP: Was: Now: NULL205.00 - NULL567.00 Choose Options Compare Quick view Biovision | SKF-86002 | 2894 SKF-86002 is a p38 MAP kinase inhibitor (IC₅₀ = 0.1 - 1 μM). Potently inhibits LPS-induced IL-1 and TNF-α production in human monocytes (IC₅₀ = 1 μM). Also acts as an inhibitor of both cyclooxygenase... MSRP: Was: Now: NULL320.00 - NULL1,009.00 Choose Options Compare Quick view Biovision | GV-58 | 2616 GV-58 is a Roscovitine (Cat. No. 1950) derivative that acts as a selective N- and P/Q-type Ca²⁺-channel agonist. These Ca2²⁺-channels regulate transmitter release in synapses. Potential lead compound... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | ANA-12 | 2878 ANA-12 is a potent and selective TrkB antagonist that prevents activation of the receptor by BDNF with a high potency. It binds selectively to TrkB and inhibits processes downstream of TrkB without... MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Biovision | NS-1619 | B1303 NS-1619 is a calcium-dependent activator of large-conductance Ca²⁺-activated K⁺ (BKCa) channels in vascular smooth muscle. Induces a concentration-dependent decrease in mitochondrial membrane... MSRP: Was: Now: NULL271.00 - NULL779.00 Choose Options Compare Quick view Biovision | PF-06447475 | 9447 PF-06447475 is a highly potent, selective, brain-permeable, and in vivo active LRRK2 (Leucine rich repeat kinase 2) kinase inhibitor. Could be potentially useful in the treatment of Parkinson’s... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | OTS-964 | B1964 OTS-964 is a potent inhibitor of lymphokine-activated killer T cell-originated protein kinase (TOPK; IC₅₀ = 28 nM). It specifically blocks cytokinesis, leading to apoptosis, in a broad range of... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Biovision | Z-DEVD-FMK | 1143 A synthetic peptide that irreversibly inhibits activity of DEVD-dependent caspases (e.g., caspase-3 and caspase-7) and blocks apoptosis. The inhibitor is designed as a methyl ester to facilitate cell... MSRP: Was: Now: NULL484.00 - NULL1,222.00 Choose Options Compare Quick view Biovision | WS3 | 2799 WS3 is a novel small molecule that promotes β cell proliferation with EC50 of 28 nM (induced R7T1 proliferation). More recently, WS3 has been found to mediate proliferation of primary retinal pigment... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | WS6 | 2711 WS6 is a novel Inducer of β cell proliferation. Inthe RIP-DTA mouse model of β cell ablation, WS6 normalizes blood glucose and induces concomitant increases in β cell proliferation and β cell number... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | Y15 | B1252 Y15 is a selective focal adhesion kinase (FAK) inhibitor preventing FAK autophosphorylation at IC₅₀ of 1 μM. It does not have any significant activity against a range of other kinases like EGFR,... MSRP: Was: Now: NULL222.00 - NULL567.00 Choose Options Compare Quick view Biovision | Gilteritinib | B1294 Gilteritinib is a potent FLT3 (FMS-like tyrosine kinase 3) inhibitor which shows potent antileukemic activity against AML with either or both FLT3-ITD and FLT3-D835 mutations.Gilteritinib is a potent... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Biovision | Zotarolimus | 9530 Zotarolimus is a semi-synthetic derivative of Sirolimus (Cat. No. 1568) that acts as an immunosuppressant. Zotarolimus displays meachanism similar to sirolimus in having high-affinity binding to the... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | PFI-3 | 2895 PFI-3 is a potent and selective polybromo 1 (PB1) and SMARCA4 (SWI/SNF related, Matrix associated, Actin dependent Regulator of Chromatin, subfamily A, member 4) inhibitor (Kd values are 48 and 89 nM... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Biovision | BAY 41-2272 | 9429 BAY 41-2272 is a soluble guanylyl cyclase (sGC) activator; acts at a nitric oxide (NO)-independent regulatory site in the sGC α1 subunit. Inhibits platelet aggregation (IC₅₀ = 36 nM) and... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | Ro 61-8048 | 1912 Cell-permeable. A high-affinity small molecule inhibitor of KMO (kynurenine 3-monoxygenase or kynurenine 3-hydroxylase)(Ki = 4.8 nM, IC₅₀ = 37 nM).Ro 61-8048 is a high-affinity small molecule... MSRP: Was: Now: NULL247.00 - NULL1,250.00 Choose Options Compare Quick view Biovision | UNC0379 | 9588 UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SET8 (IC₅₀ = 7.3 µM; Kd = 18.3 µM). It is selective for SET8 over 15 other methyltransferases, including G9a... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | HTH-01-015 | 2887 HTH-01-015 is a potent and selective inhibitor of NUAK1 kinase (IC₅₀ =100 nM); only weakly inhibits NUAK2 (IC₅₀ of >10 μM) and does not significantly inhibit the activity of 139 other kinases that... MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Biovision | G-749 | B2213 G-749 is a potent FLT3 kinase inhibitor that displays potent and sustained inhibition of the FLT3 wild type and mutants including FLT3-ITD, FLT3-D835Y, FLT3-ITD/N676D, and FLT3-ITD/F691L in cellular... MSRP: Was: Now: NULL205.00 - NULL533.00 Choose Options Compare Quick view Biovision | (-)-Indolactam V | 2197 Cell-permeable. A protein kinase C (PKC) activator and a tumor promoter. Directs differentiation of human embryonic stem cells (ESCs) into pancreatic progenitors.(-)-Indolactam is a protein kinase C... MSRP: Was: Now: NULL263.00 - NULL616.00 Choose Options Compare Quick view Biovision | Q-VD-OPh | 1170 A synthetic peptide that is potent, cell permeable, nontoxic and irreversibly inhibits caspase activity to blocks apoptosis. The new generation of caspase inhibitor is more stable in aqueous... MSRP: Was: Now: NULL378.00 - NULL10,854.00 Choose Options Compare Quick view Biovision | OAC1 | B1079 OAC1 is an Oct4-activating compound that activates expression through the Oct4 gene promoter. In cells expressing Oct4 with Sox2, Klf4, and c-Myc, OAC1 (1 μM) enhances reprogramming efficiency by... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | Kenpaullone | 1904 Cell-permeable. A potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases. In addition, it has been found to be a... MSRP: Now: NULL214.00 Add to Cart Compare Quick view Biovision | WH-4-023 | 2827 WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC₅₀ of 2 nM and 6 nM for Lck and Src kinase respectively; little inhibition on p38α and KDR.WH-4-023 is a potent and selective dual... MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare Quick view Biovision | IM-12 | 2822 IM-12 is a potent and selective GSK-3β inhibitor (IC₅₀ = 53 nM). It significantly increases β-catenin levels, leads to TCF-induction and promotes neuronal differentiation in human neural progenitor... MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare Quick view Biovision | Ozanimod | B1196 Ozanimod (RPC1063) is an orally bioavailable agonist of the sphingosine-1-phosphate receptor subtypes 1 (S1P1) and 5 (S1P5). S1P receptors belong to the family of G-protein-coupled receptor which... MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare Quick view Biovision | YH239-EE | B1229 YH239-EE is potent p53-MDM2 interaction inhibitor that induces cell cycle arrest leading to potential apoptosis by p53 activation and downstream target in AML cells with p53 mutationYH239-EE is... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | Serabelisib | B1930 Serabelisib is a potent inhibitor of phosphoinositide 3-kinase α (PI3Kα) that is selective for p110α in vitro (IC₅₀ = 15 nM for PI3Kα vs. >1 µM for other isoforms, as well as for mTOR). MLN1117... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | K02288 | B2321 A potent and selective inhibitor of type I bone morphogenic protein (BMP) receptors (IC₅₀ values are 1.1, 1.8, 6.4, 34.4, 220, 302 and 321 nM for ALK2, ALK1, ALK6, ALK3, ActRIIA, ALK4 and ALK5... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | DMH-1 | 9542 DMH-1 is an analog of Dorsomorphin (Cat. No. 1686) that acts as a highly selective Bone morphogenetic protein (BMP) inhibitor. DMH-1 exclusively targets the BMP but not the VEGF pathway. Blocks... MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare Quick view Biovision | T-5224 | 9546 T-5224 is a selective inhibitor of c-Fos/activator protein (AP)-1 that ameliorates liver injury and improves survival through decreasing production of pro-inflammatory cytokines and chemokines in... MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare Quick view Biovision | XEN445 | 2681 XEN445 is a potent and selective endothelial lipase (EL) inhibitor. It displays good ADME and PK properties and shows in vivo efficacy in raising plasma HDL cholesterol concentration in mice.XEN445... MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare Quick view Biovision | PI-3065 | B1674 PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value of 1.5nM and IC50 value of 5nM.PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value... MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare Quick view Details Biovision | QS11 | 1680 MSRP: Now: NULL386.00 Add to Cart Compare Quick view Details Biovision | ML141 | 2267 MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare Quick view Details Biovision | genz-123346 | B2286 MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare Quick view Details Biovision | Tautomycin | B1237 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | Liproxstatin-1 | B2312 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | ITD-1 | 2879 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | 10058-F4 | 2739 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | CH-223191 | 2723 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | BPTES | B2165 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Entrectinib | B1324 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | MPI-0479605 | 9589 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Acalisib | B1666 MSRP: Was: Now: NULL247.00 - NULL739.00 Choose Options Compare Quick view Details Biovision | URMC-099 | 9443 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | A-366 | 2859 MSRP: Was: Now: NULL254.00 - NULL714.00 Choose Options Compare Quick view Details Biovision | Velpatasvir | B1194 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | RO-3306 | 2039 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | Pyridoclax | B1817 MSRP: Was: Now: NULL303.00 - NULL967.00 Choose Options Compare Quick view Details Biovision | Bikinin | 2034 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | OF-1 | 9592 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | LY3023414 | B1759 MSRP: Was: Now: NULL205.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | SKF-86002 | 2894 MSRP: Was: Now: NULL320.00 - NULL1,009.00 Choose Options Compare Quick view Details Biovision | GV-58 | 2616 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | ANA-12 | 2878 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | NS-1619 | B1303 MSRP: Was: Now: NULL271.00 - NULL779.00 Choose Options Compare Quick view Details Biovision | PF-06447475 | 9447 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | OTS-964 | B1964 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | Z-DEVD-FMK | 1143 MSRP: Was: Now: NULL484.00 - NULL1,222.00 Choose Options Compare Quick view Details Biovision | WS3 | 2799 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | WS6 | 2711 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Y15 | B1252 MSRP: Was: Now: NULL222.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | Gilteritinib | B1294 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Zotarolimus | 9530 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | PFI-3 | 2895 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | BAY 41-2272 | 9429 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Ro 61-8048 | 1912 MSRP: Was: Now: NULL247.00 - NULL1,250.00 Choose Options Compare Quick view Details Biovision | UNC0379 | 9588 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | HTH-01-015 | 2887 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | G-749 | B2213 MSRP: Was: Now: NULL205.00 - NULL533.00 Choose Options Compare Quick view Details Biovision | (-)-Indolactam V | 2197 MSRP: Was: Now: NULL263.00 - NULL616.00 Choose Options Compare Quick view Details Biovision | Q-VD-OPh | 1170 MSRP: Was: Now: NULL378.00 - NULL10,854.00 Choose Options Compare Quick view Details Biovision | OAC1 | B1079 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Kenpaullone | 1904 MSRP: Now: NULL214.00 Add to Cart Compare Quick view Details Biovision | WH-4-023 | 2827 MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | IM-12 | 2822 MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare Quick view Details Biovision | Ozanimod | B1196 MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare Quick view Details Biovision | YH239-EE | B1229 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Serabelisib | B1930 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | K02288 | B2321 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | DMH-1 | 9542 MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare Quick view Details Biovision | T-5224 | 9546 MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | XEN445 | 2681 MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare Quick view Details Biovision | PI-3065 | B1674 MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare Previous 187 188 189 190 191 192 193 194 195 196 197 Next Previous 187 188 189 190 191 192 193 194 195 196 197 Next Compare Selected × OK
Quick view Biovision | ML141 | 2267 Cell-permeable. A potent, selective, reversible and non-competitive inhibitor of Cdc42 GTPase (IC₅₀ = 2.6 and 5.4 μM for Cdc42 wild type and activated mutant, respectively). No appreciable inhibitory... MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare
Quick view Biovision | genz-123346 | B2286 Genz-123346 is a potent and selective glucosylceramide synthase inhibitor with potential anticancer activity. Does not affect the activities of other related glycosidase, such as 1-O-acylceramide... MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare
Quick view Biovision | Tautomycin | B1237 Tautomycin is a potent protein phosphatase inhibitor that inhibits PP1 completely at 3 nM and PP2 at 30 nM. Acts as a weak inhibitor of PP2B and does not inhibit PP2C. Its cell permeability and... MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare
Quick view Biovision | Liproxstatin-1 | B2312 A potent inhibitor of ferroptosis. Liproxstatin-1 suppresses ferroptosis in human cells and in an ischemia/reperfusion-induced tissue injury model in mice. Knockout of glutathione peroxidase 4 (Gpx4)... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Biovision | ITD-1 | 2879 ITD-1 is a potent and highly selective TGFβ pathway inhibitor (IC₅₀ = 0.85 µM). ITD-1 promotes cardiomyocyte differentiation specifically via degradation of the TGFβ type II receptor (TGFBR2),... MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare
Quick view Biovision | 10058-F4 | 2739 10058-F4 is a c-Myc inhibitor that inhibits the c-Myc-Max associationn and function. It prevents the growth of fibroblasts in a c-Myc-dependent manner. Downregulates human telomerase reverse... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Biovision | CH-223191 | 2723 CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist. It blocks activation by 2,3,7,8-Tetrachlorodibenzo-p-dioxin (TCDD) (IC₅₀ = 0.03 µM). It also blocks TCDD-mediated... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Biovision | BPTES | B2165 BPTES is an allosteric glutaminase (GLS1) inhibitor (IC₅₀ = 3.3 μM). Displays selectivity for GLS1 over GLS2 and γ-glutamyl transpeptidase. Induces cell death of P493 human lymphoma B cells in vitro... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare
Quick view Biovision | Entrectinib | B1324 Entrectinib is an inhibitor of TrkA (IC₅₀ = 1.7 nM), TrkB (IC₅₀ = 0.1 nM), and TrkC (IC₅₀ = 0.1 nM), as well as C-ros oncogene 1 (ROS1; IC₅₀ = 0.2 nM) and anaplastic lymphoma kinase (ALK; IC₅₀ = 1.6... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | MPI-0479605 | 9589 MPI-0479605 is a potent, selective, ATP-competitive small-molecule inhibitor of the Mitotic kinase Mps1 (IC₅₀ = 1.8 nM).MPI-0479605 is a potent, selective, ATP-competitive small-molecule inhibitor of... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | Acalisib | B1666 Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12.7 nM.Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12.7 nM.Biovision | B1666... MSRP: Was: Now: NULL247.00 - NULL739.00 Choose Options Compare
Quick view Biovision | URMC-099 | 9443 URMC-099 is a brain-permeable, mixed lineage kinase (MLK) inhibitor with IC₅₀ values of 19 nM, 42 nM, 14 nM, and 150 nM, for MLK1, MLK2, MLK3, and DLK, respectively. In vitro, URMC-099 treatment... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare
Quick view Biovision | A-366 | 2859 A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC₅₀ = 3.3 nM). It displays >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. A-366 has been... MSRP: Was: Now: NULL254.00 - NULL714.00 Choose Options Compare
Quick view Biovision | Velpatasvir | B1194 Velpatasvir (formerly GS-5816) is a novel NS5A inhibitor that has potent in vitro anti-HCV activity across all genotypes at the picomolar level.Velpatasvir (formerly GS-5816) is a novel NS5A... MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Biovision | RO-3306 | 2039 Cell-permeable. A selective CDK 1 inhibitor (Cdk1/B1 and Cdk1/A). Arrests cell cycle at G1, S, and G2/M and induces apoptosis in embryonic stem cells. Actively enhances downstream p53 signaling to... MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare
Quick view Biovision | Pyridoclax | B1817 Pyridoclax(MR-29072) is a potent Mcl-1 inhibitor (Kd = 25 nM). Pyridoclax is able to disrupt BimL/Mcl-1 interaction in whole living cells.Pyridoclax(MR-29072) is a potent Mcl-1 inhibitor (Kd = 25 nM)... MSRP: Was: Now: NULL303.00 - NULL967.00 Choose Options Compare
Quick view Biovision | Bikinin | 2034 Cell-permeable. A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase that activates brassinosteroid (BR) signaling downstream of the BR receptor. Bikinin directly binds the GSK3 BIN2... MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare
Quick view Biovision | OF-1 | 9592 OF-1 is a selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500 nM respectively). OF-1 displays 39-fold selectivity for BRPF1B and BRPF2 over BRD4. It increases thermal... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare
Quick view Biovision | LY3023414 | B1759 LY3023414 is a small molecule that has been shown in vitro to be a selective ATP-competitive inhibitor of PI3Kα and mTOR, DNA-PK, and other class I PI3K family members.LY3023414 is a small molecule... MSRP: Was: Now: NULL205.00 - NULL567.00 Choose Options Compare
Quick view Biovision | SKF-86002 | 2894 SKF-86002 is a p38 MAP kinase inhibitor (IC₅₀ = 0.1 - 1 μM). Potently inhibits LPS-induced IL-1 and TNF-α production in human monocytes (IC₅₀ = 1 μM). Also acts as an inhibitor of both cyclooxygenase... MSRP: Was: Now: NULL320.00 - NULL1,009.00 Choose Options Compare
Quick view Biovision | GV-58 | 2616 GV-58 is a Roscovitine (Cat. No. 1950) derivative that acts as a selective N- and P/Q-type Ca²⁺-channel agonist. These Ca2²⁺-channels regulate transmitter release in synapses. Potential lead compound... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | ANA-12 | 2878 ANA-12 is a potent and selective TrkB antagonist that prevents activation of the receptor by BDNF with a high potency. It binds selectively to TrkB and inhibits processes downstream of TrkB without... MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare
Quick view Biovision | NS-1619 | B1303 NS-1619 is a calcium-dependent activator of large-conductance Ca²⁺-activated K⁺ (BKCa) channels in vascular smooth muscle. Induces a concentration-dependent decrease in mitochondrial membrane... MSRP: Was: Now: NULL271.00 - NULL779.00 Choose Options Compare
Quick view Biovision | PF-06447475 | 9447 PF-06447475 is a highly potent, selective, brain-permeable, and in vivo active LRRK2 (Leucine rich repeat kinase 2) kinase inhibitor. Could be potentially useful in the treatment of Parkinson’s... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | OTS-964 | B1964 OTS-964 is a potent inhibitor of lymphokine-activated killer T cell-originated protein kinase (TOPK; IC₅₀ = 28 nM). It specifically blocks cytokinesis, leading to apoptosis, in a broad range of... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare
Quick view Biovision | Z-DEVD-FMK | 1143 A synthetic peptide that irreversibly inhibits activity of DEVD-dependent caspases (e.g., caspase-3 and caspase-7) and blocks apoptosis. The inhibitor is designed as a methyl ester to facilitate cell... MSRP: Was: Now: NULL484.00 - NULL1,222.00 Choose Options Compare
Quick view Biovision | WS3 | 2799 WS3 is a novel small molecule that promotes β cell proliferation with EC50 of 28 nM (induced R7T1 proliferation). More recently, WS3 has been found to mediate proliferation of primary retinal pigment... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | WS6 | 2711 WS6 is a novel Inducer of β cell proliferation. Inthe RIP-DTA mouse model of β cell ablation, WS6 normalizes blood glucose and induces concomitant increases in β cell proliferation and β cell number... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | Y15 | B1252 Y15 is a selective focal adhesion kinase (FAK) inhibitor preventing FAK autophosphorylation at IC₅₀ of 1 μM. It does not have any significant activity against a range of other kinases like EGFR,... MSRP: Was: Now: NULL222.00 - NULL567.00 Choose Options Compare
Quick view Biovision | Gilteritinib | B1294 Gilteritinib is a potent FLT3 (FMS-like tyrosine kinase 3) inhibitor which shows potent antileukemic activity against AML with either or both FLT3-ITD and FLT3-D835 mutations.Gilteritinib is a potent... MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare
Quick view Biovision | Zotarolimus | 9530 Zotarolimus is a semi-synthetic derivative of Sirolimus (Cat. No. 1568) that acts as an immunosuppressant. Zotarolimus displays meachanism similar to sirolimus in having high-affinity binding to the... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | PFI-3 | 2895 PFI-3 is a potent and selective polybromo 1 (PB1) and SMARCA4 (SWI/SNF related, Matrix associated, Actin dependent Regulator of Chromatin, subfamily A, member 4) inhibitor (Kd values are 48 and 89 nM... MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare
Quick view Biovision | BAY 41-2272 | 9429 BAY 41-2272 is a soluble guanylyl cyclase (sGC) activator; acts at a nitric oxide (NO)-independent regulatory site in the sGC α1 subunit. Inhibits platelet aggregation (IC₅₀ = 36 nM) and... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | Ro 61-8048 | 1912 Cell-permeable. A high-affinity small molecule inhibitor of KMO (kynurenine 3-monoxygenase or kynurenine 3-hydroxylase)(Ki = 4.8 nM, IC₅₀ = 37 nM).Ro 61-8048 is a high-affinity small molecule... MSRP: Was: Now: NULL247.00 - NULL1,250.00 Choose Options Compare
Quick view Biovision | UNC0379 | 9588 UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SET8 (IC₅₀ = 7.3 µM; Kd = 18.3 µM). It is selective for SET8 over 15 other methyltransferases, including G9a... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | HTH-01-015 | 2887 HTH-01-015 is a potent and selective inhibitor of NUAK1 kinase (IC₅₀ =100 nM); only weakly inhibits NUAK2 (IC₅₀ of >10 μM) and does not significantly inhibit the activity of 139 other kinases that... MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare
Quick view Biovision | G-749 | B2213 G-749 is a potent FLT3 kinase inhibitor that displays potent and sustained inhibition of the FLT3 wild type and mutants including FLT3-ITD, FLT3-D835Y, FLT3-ITD/N676D, and FLT3-ITD/F691L in cellular... MSRP: Was: Now: NULL205.00 - NULL533.00 Choose Options Compare
Quick view Biovision | (-)-Indolactam V | 2197 Cell-permeable. A protein kinase C (PKC) activator and a tumor promoter. Directs differentiation of human embryonic stem cells (ESCs) into pancreatic progenitors.(-)-Indolactam is a protein kinase C... MSRP: Was: Now: NULL263.00 - NULL616.00 Choose Options Compare
Quick view Biovision | Q-VD-OPh | 1170 A synthetic peptide that is potent, cell permeable, nontoxic and irreversibly inhibits caspase activity to blocks apoptosis. The new generation of caspase inhibitor is more stable in aqueous... MSRP: Was: Now: NULL378.00 - NULL10,854.00 Choose Options Compare
Quick view Biovision | OAC1 | B1079 OAC1 is an Oct4-activating compound that activates expression through the Oct4 gene promoter. In cells expressing Oct4 with Sox2, Klf4, and c-Myc, OAC1 (1 μM) enhances reprogramming efficiency by... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | Kenpaullone | 1904 Cell-permeable. A potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases. In addition, it has been found to be a... MSRP: Now: NULL214.00 Add to Cart Compare Quick view Biovision | WH-4-023 | 2827 WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC₅₀ of 2 nM and 6 nM for Lck and Src kinase respectively; little inhibition on p38α and KDR.WH-4-023 is a potent and selective dual... MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare Quick view Biovision | IM-12 | 2822 IM-12 is a potent and selective GSK-3β inhibitor (IC₅₀ = 53 nM). It significantly increases β-catenin levels, leads to TCF-induction and promotes neuronal differentiation in human neural progenitor... MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare Quick view Biovision | Ozanimod | B1196 Ozanimod (RPC1063) is an orally bioavailable agonist of the sphingosine-1-phosphate receptor subtypes 1 (S1P1) and 5 (S1P5). S1P receptors belong to the family of G-protein-coupled receptor which... MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare Quick view Biovision | YH239-EE | B1229 YH239-EE is potent p53-MDM2 interaction inhibitor that induces cell cycle arrest leading to potential apoptosis by p53 activation and downstream target in AML cells with p53 mutationYH239-EE is... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | Serabelisib | B1930 Serabelisib is a potent inhibitor of phosphoinositide 3-kinase α (PI3Kα) that is selective for p110α in vitro (IC₅₀ = 15 nM for PI3Kα vs. >1 µM for other isoforms, as well as for mTOR). MLN1117... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Biovision | K02288 | B2321 A potent and selective inhibitor of type I bone morphogenic protein (BMP) receptors (IC₅₀ values are 1.1, 1.8, 6.4, 34.4, 220, 302 and 321 nM for ALK2, ALK1, ALK6, ALK3, ActRIIA, ALK4 and ALK5... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Biovision | DMH-1 | 9542 DMH-1 is an analog of Dorsomorphin (Cat. No. 1686) that acts as a highly selective Bone morphogenetic protein (BMP) inhibitor. DMH-1 exclusively targets the BMP but not the VEGF pathway. Blocks... MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare Quick view Biovision | T-5224 | 9546 T-5224 is a selective inhibitor of c-Fos/activator protein (AP)-1 that ameliorates liver injury and improves survival through decreasing production of pro-inflammatory cytokines and chemokines in... MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare Quick view Biovision | XEN445 | 2681 XEN445 is a potent and selective endothelial lipase (EL) inhibitor. It displays good ADME and PK properties and shows in vivo efficacy in raising plasma HDL cholesterol concentration in mice.XEN445... MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare Quick view Biovision | PI-3065 | B1674 PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value of 1.5nM and IC50 value of 5nM.PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value... MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare Quick view Details Biovision | QS11 | 1680 MSRP: Now: NULL386.00 Add to Cart Compare Quick view Details Biovision | ML141 | 2267 MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare Quick view Details Biovision | genz-123346 | B2286 MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare Quick view Details Biovision | Tautomycin | B1237 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | Liproxstatin-1 | B2312 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | ITD-1 | 2879 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | 10058-F4 | 2739 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | CH-223191 | 2723 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | BPTES | B2165 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Entrectinib | B1324 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | MPI-0479605 | 9589 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Acalisib | B1666 MSRP: Was: Now: NULL247.00 - NULL739.00 Choose Options Compare Quick view Details Biovision | URMC-099 | 9443 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | A-366 | 2859 MSRP: Was: Now: NULL254.00 - NULL714.00 Choose Options Compare Quick view Details Biovision | Velpatasvir | B1194 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | RO-3306 | 2039 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | Pyridoclax | B1817 MSRP: Was: Now: NULL303.00 - NULL967.00 Choose Options Compare Quick view Details Biovision | Bikinin | 2034 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | OF-1 | 9592 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | LY3023414 | B1759 MSRP: Was: Now: NULL205.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | SKF-86002 | 2894 MSRP: Was: Now: NULL320.00 - NULL1,009.00 Choose Options Compare Quick view Details Biovision | GV-58 | 2616 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | ANA-12 | 2878 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | NS-1619 | B1303 MSRP: Was: Now: NULL271.00 - NULL779.00 Choose Options Compare Quick view Details Biovision | PF-06447475 | 9447 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | OTS-964 | B1964 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | Z-DEVD-FMK | 1143 MSRP: Was: Now: NULL484.00 - NULL1,222.00 Choose Options Compare Quick view Details Biovision | WS3 | 2799 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | WS6 | 2711 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Y15 | B1252 MSRP: Was: Now: NULL222.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | Gilteritinib | B1294 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Zotarolimus | 9530 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | PFI-3 | 2895 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | BAY 41-2272 | 9429 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Ro 61-8048 | 1912 MSRP: Was: Now: NULL247.00 - NULL1,250.00 Choose Options Compare Quick view Details Biovision | UNC0379 | 9588 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | HTH-01-015 | 2887 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | G-749 | B2213 MSRP: Was: Now: NULL205.00 - NULL533.00 Choose Options Compare Quick view Details Biovision | (-)-Indolactam V | 2197 MSRP: Was: Now: NULL263.00 - NULL616.00 Choose Options Compare Quick view Details Biovision | Q-VD-OPh | 1170 MSRP: Was: Now: NULL378.00 - NULL10,854.00 Choose Options Compare Quick view Details Biovision | OAC1 | B1079 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Kenpaullone | 1904 MSRP: Now: NULL214.00 Add to Cart Compare Quick view Details Biovision | WH-4-023 | 2827 MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | IM-12 | 2822 MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare Quick view Details Biovision | Ozanimod | B1196 MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare Quick view Details Biovision | YH239-EE | B1229 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Serabelisib | B1930 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | K02288 | B2321 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | DMH-1 | 9542 MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare Quick view Details Biovision | T-5224 | 9546 MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | XEN445 | 2681 MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare Quick view Details Biovision | PI-3065 | B1674 MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare Previous 187 188 189 190 191 192 193 194 195 196 197 Next Previous 187 188 189 190 191 192 193 194 195 196 197 Next Compare Selected × OK
Quick view Biovision | WH-4-023 | 2827 WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC₅₀ of 2 nM and 6 nM for Lck and Src kinase respectively; little inhibition on p38α and KDR.WH-4-023 is a potent and selective dual... MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare
Quick view Biovision | IM-12 | 2822 IM-12 is a potent and selective GSK-3β inhibitor (IC₅₀ = 53 nM). It significantly increases β-catenin levels, leads to TCF-induction and promotes neuronal differentiation in human neural progenitor... MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare
Quick view Biovision | Ozanimod | B1196 Ozanimod (RPC1063) is an orally bioavailable agonist of the sphingosine-1-phosphate receptor subtypes 1 (S1P1) and 5 (S1P5). S1P receptors belong to the family of G-protein-coupled receptor which... MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare
Quick view Biovision | YH239-EE | B1229 YH239-EE is potent p53-MDM2 interaction inhibitor that induces cell cycle arrest leading to potential apoptosis by p53 activation and downstream target in AML cells with p53 mutationYH239-EE is... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | Serabelisib | B1930 Serabelisib is a potent inhibitor of phosphoinositide 3-kinase α (PI3Kα) that is selective for p110α in vitro (IC₅₀ = 15 nM for PI3Kα vs. >1 µM for other isoforms, as well as for mTOR). MLN1117... MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
Quick view Biovision | K02288 | B2321 A potent and selective inhibitor of type I bone morphogenic protein (BMP) receptors (IC₅₀ values are 1.1, 1.8, 6.4, 34.4, 220, 302 and 321 nM for ALK2, ALK1, ALK6, ALK3, ActRIIA, ALK4 and ALK5... MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare
Quick view Biovision | DMH-1 | 9542 DMH-1 is an analog of Dorsomorphin (Cat. No. 1686) that acts as a highly selective Bone morphogenetic protein (BMP) inhibitor. DMH-1 exclusively targets the BMP but not the VEGF pathway. Blocks... MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare
Quick view Biovision | T-5224 | 9546 T-5224 is a selective inhibitor of c-Fos/activator protein (AP)-1 that ameliorates liver injury and improves survival through decreasing production of pro-inflammatory cytokines and chemokines in... MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare
Quick view Biovision | XEN445 | 2681 XEN445 is a potent and selective endothelial lipase (EL) inhibitor. It displays good ADME and PK properties and shows in vivo efficacy in raising plasma HDL cholesterol concentration in mice.XEN445... MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare
Quick view Biovision | PI-3065 | B1674 PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value of 1.5nM and IC50 value of 5nM.PI-3065 is a small molecule and selective inhibitor of p110δkinase with an Ki value... MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare
Quick view Details Biovision | QS11 | 1680 MSRP: Now: NULL386.00 Add to Cart Compare Quick view Details Biovision | ML141 | 2267 MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare Quick view Details Biovision | genz-123346 | B2286 MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare Quick view Details Biovision | Tautomycin | B1237 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | Liproxstatin-1 | B2312 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | ITD-1 | 2879 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | 10058-F4 | 2739 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | CH-223191 | 2723 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | BPTES | B2165 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Entrectinib | B1324 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | MPI-0479605 | 9589 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Acalisib | B1666 MSRP: Was: Now: NULL247.00 - NULL739.00 Choose Options Compare Quick view Details Biovision | URMC-099 | 9443 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | A-366 | 2859 MSRP: Was: Now: NULL254.00 - NULL714.00 Choose Options Compare Quick view Details Biovision | Velpatasvir | B1194 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare Quick view Details Biovision | RO-3306 | 2039 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | Pyridoclax | B1817 MSRP: Was: Now: NULL303.00 - NULL967.00 Choose Options Compare Quick view Details Biovision | Bikinin | 2034 MSRP: Was: Now: NULL197.00 - NULL518.00 Choose Options Compare Quick view Details Biovision | OF-1 | 9592 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | LY3023414 | B1759 MSRP: Was: Now: NULL205.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | SKF-86002 | 2894 MSRP: Was: Now: NULL320.00 - NULL1,009.00 Choose Options Compare Quick view Details Biovision | GV-58 | 2616 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | ANA-12 | 2878 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare Quick view Details Biovision | NS-1619 | B1303 MSRP: Was: Now: NULL271.00 - NULL779.00 Choose Options Compare Quick view Details Biovision | PF-06447475 | 9447 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | OTS-964 | B1964 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | Z-DEVD-FMK | 1143 MSRP: Was: Now: NULL484.00 - NULL1,222.00 Choose Options Compare Quick view Details Biovision | WS3 | 2799 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | WS6 | 2711 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Y15 | B1252 MSRP: Was: Now: NULL222.00 - NULL567.00 Choose Options Compare Quick view Details Biovision | Gilteritinib | B1294 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare Quick view Details Biovision | Zotarolimus | 9530 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | PFI-3 | 2895 MSRP: Was: Now: NULL320.00 - NULL1,024.00 Choose Options Compare Quick view Details Biovision | BAY 41-2272 | 9429 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Ro 61-8048 | 1912 MSRP: Was: Now: NULL247.00 - NULL1,250.00 Choose Options Compare Quick view Details Biovision | UNC0379 | 9588 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | HTH-01-015 | 2887 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare Quick view Details Biovision | G-749 | B2213 MSRP: Was: Now: NULL205.00 - NULL533.00 Choose Options Compare Quick view Details Biovision | (-)-Indolactam V | 2197 MSRP: Was: Now: NULL263.00 - NULL616.00 Choose Options Compare Quick view Details Biovision | Q-VD-OPh | 1170 MSRP: Was: Now: NULL378.00 - NULL10,854.00 Choose Options Compare Quick view Details Biovision | OAC1 | B1079 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | Kenpaullone | 1904 MSRP: Now: NULL214.00 Add to Cart Compare Quick view Details Biovision | WH-4-023 | 2827 MSRP: Was: Now: NULL320.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | IM-12 | 2822 MSRP: Was: Now: NULL222.00 - NULL648.00 Choose Options Compare Quick view Details Biovision | Ozanimod | B1196 MSRP: Was: Now: NULL320.00 - NULL975.00 Choose Options Compare Quick view Details Biovision | YH239-EE | B1229 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | Serabelisib | B1930 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare Quick view Details Biovision | K02288 | B2321 MSRP: Was: Now: NULL239.00 - NULL697.00 Choose Options Compare Quick view Details Biovision | DMH-1 | 9542 MSRP: Was: Now: NULL288.00 - NULL935.00 Choose Options Compare Quick view Details Biovision | T-5224 | 9546 MSRP: Was: Now: NULL337.00 - NULL1,041.00 Choose Options Compare Quick view Details Biovision | XEN445 | 2681 MSRP: Was: Now: NULL271.00 - NULL837.00 Choose Options Compare Quick view Details Biovision | PI-3065 | B1674 MSRP: Was: Now: NULL247.00 - NULL771.00 Choose Options Compare Previous 187 188 189 190 191 192 193 194 195 196 197 Next Previous 187 188 189 190 191 192 193 194 195 196 197 Next Compare Selected
Quick view Details Biovision | ML141 | 2267 MSRP: Was: Now: NULL222.00 - NULL730.00 Choose Options Compare
Quick view Details Biovision | genz-123346 | B2286 MSRP: Was: Now: NULL222.00 - NULL656.00 Choose Options Compare
Quick view Details Biovision | Tautomycin | B1237 MSRP: Was: Now: NULL354.00 - NULL1,148.00 Choose Options Compare
Quick view Details Biovision | Liproxstatin-1 | B2312 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Details Biovision | ITD-1 | 2879 MSRP: Was: Now: NULL303.00 - NULL959.00 Choose Options Compare
Quick view Details Biovision | 10058-F4 | 2739 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Details Biovision | CH-223191 | 2723 MSRP: Was: Now: NULL222.00 - NULL631.00 Choose Options Compare
Quick view Details Biovision | BPTES | B2165 MSRP: Was: Now: NULL271.00 - NULL828.00 Choose Options Compare
Quick view Details Biovision | Entrectinib | B1324 MSRP: Was: Now: NULL288.00 - NULL894.00 Choose Options Compare
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